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Febrifugine

PubChem CID: 9851692

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Compound Synonyms Febrifugine, 24159-07-7, Ferbifrugin, beta-Dichroine, .beta.-Dichroine, 89UWD0FH2I, DICHROIN B, .BETA.-DICHROIN, FEBRIFUGINE [MI], UNII-89UWD0FH2I, Dichroin, TRANS-(+)-FEBRIFUGINE, CHEMBL322782, 3-(3-(3-Hydroxy-2-piperidinyl)-2-oxopropyl)-4(3H)-quinazolinone, NSC 315535, NSC-315535, 3-[3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl]quinazolin-4-one, (E)-3-(3-(3-Hydroxy-2-piperidinyl)acetonyl)-4-(3H)-quinazolinone, trans-3-(beta-Keto-gamma-(3-hydroxy-2-piperidyl)propyl)-4-quinazolone, (E)-3-(3-(3-Hydroxy-2-piperidinyl)-2-oxopropyl)-4(3H)-quinazolinone, 3-[3-[(2R,3S)-3-Hydroxy-2-piperidinyl]-2-oxopropyl]-4(3H)-quinazolinone, 3-{3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl}quinazolin-4(3H)-one, 3-(3-((2R,3S)-3-HYDROXY-2-PIPERIDINYL)-2-OXOPROPYL)-4(3H)-QUINAZOLINONE, 4(3H)-Quinazolinone, 3-(3-(3-hydroxy-2-piperidinyl)-2-oxopropyl)-, (2S-trans)-, 3-(3-((2R,3S)-3-hydroxypiperidin-2-yl)-2-oxopropyl)quinazolin-4(3H)-one, 3-(3-((2R,3S)-3-hydroxypiperidin-2-yl)-2-oxopropyl)quinazolin-4-one, 9SF, Febrifugine (8CI), BETA-DICHROIN, SCHEMBL9542831, 3-(3-((2S,3R)-3-hydroxy-2-piperidyl)-2-oxo-propyl)quinazolin-4-one, 3-[3-[(2S,3R)-3-hydroxy-2-piperidyl]-2-oxo-propyl]quinazolin-4-one, DTXSID30946987, HY-N2384, BDBM50606503, AKOS040760109, AC-34102, DA-63399, MS-24342, CS-0022587
Topological Polar Surface Area 82.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 22.0
Isotope Atom Count 0.0
Molecular Complexity 466.0
Database Name cmaup_ingredients;npass_chem_all;pubchem
Defined Atom Stereocenter Count 2.0
Iupac Name 3-[3-[(2R,3S)-3-hydroxypiperidin-2-yl]-2-oxopropyl]quinazolin-4-one
Prediction Hob 1.0
Xlogp 0.1
Molecular Formula C16H19N3O3
Prediction Swissadme 1.0
Inchi Key FWVHWDSCPKXMDB-CABCVRRESA-N
Fcsp3 0.4375
Logs -0.844
Rotatable Bond Count 4.0
Logd -0.296
Compound Name Febrifugine
Prediction Hob Swissadme 1.0
Exact Mass 301.143
Formal Charge 0.0
Monoisotopic Mass 301.143
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 301.34
Covalent Unit Count 1.0
Total Atom Stereocenter Count 2.0
Total Bond Stereocenter Count 0.0
Esol -2.7194088363636353
Inchi InChI=1S/C16H19N3O3/c20-11(8-14-15(21)6-3-7-17-14)9-19-10-18-13-5-2-1-4-12(13)16(19)22/h1-2,4-5,10,14-15,17,21H,3,6-9H2/t14-,15+/m1/s1
Smiles C1C[C@@H]([C@H](NC1)CC(=O)CN2C=NC3=CC=CC=C3C2=O)O
Nring 3.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Dichroa Febrifuga (Plant) Rel Props:Source_db:npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Hydrangea Umbellata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all