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Neoandrographolide

PubChem CID: 9848024

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Compound Synonyms Neoandrographolide, 27215-14-1, Neoandrographiside, (-)-neoandrographolide, UNII-XBY0Z806J2, XBY0Z806J2, DTXSID80904895, 3-(2-((1R,4aS,5R,8aS)-5,8a-dimethyl-2-methylene-5-((((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)oxy)methyl)decahydronaphthalen-1-yl)ethyl)furan-2(5H)-one, 4-[2-[(1R,4aS,5R,8aS)-5,8a-dimethyl-2-methylidene-5-[[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]-3,4,4a,6,7,8-hexahydro-1H-naphthalen-1-yl]ethyl]-2H-furan-5-one, NEOANDROGRAPHOLIDE (CONSTITUENT OF ANDROGRAPHIS) [DSC], 2(5H)-FURANONE, 3-(2-((1R,4AS,5R,8AS)-5-((.BETA.-D-GLUCOPYRANOSYLOXY)METHYL)DECAHYDRO-5,8A-DIMETHYL-2-METHYLENE-1-NAPHTHALENYL)ETHYL)-, 2(5H)-FURANONE, 3-(2-(5-((.BETA.-D-GLUCOPYRANOSYLOXY)METHYL)DECAHYDRO-5,8A-DIMETHYL-2-METHYLENE-1-NAPHTHALENYL)ETHYL)-, (1R-(1.ALPHA.,4A.BETA.,5.ALPHA.,8A.ALPHA.))-, 2(5H)-Furanone, 3-(2-(5-((beta-D-glucopyranosyloxy)methyl)decahydro-5,8a-dimethyl-2-methylene-1-naphthalenyl)ethyl)-, (1R-(1alpha,4abeta,5alpha,8aalpha))-, 5.BETA.,9.BETA.H,10.ALPHA.-LABDA-8(20),13-DIEN-16-OIC ACID, 18-(GLUCOSYLOXY)-15-HYDROXY-, .GAMMA.-LACTONE, 4-(2-((1R,4aS,5R,8aS)-5,8a-dimethyl-2-methylidene-5-(((2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl)oxymethyl)-3,4,4a,6,7,8-hexahydro-1H-naphthalen-1-yl)ethyl)-2H-furan-5-one, Neoandrographolide (Standard), CHEMBL480853, MEGxp0_000981, SCHEMBL2225354, ACon1_000667, HY-N0721R, CHEBI:228890, DTXCID001334004, HY-N0721, s9157, AKOS030526126, Neoandrographolide, analytical standard, CCG-269552, CS-3656, MN11576, NCGC00169477-01, NCGC00169477-02, 2(5H)-Furanone, 3-(2-((1R,4aS,5R,8aS)-5-((beta-D-glucopyranosyloxy)methyl)decahydro-5,8a-dimethyl-2-methylene-1-naphthalenyl)ethyl)-, 3-[2-[(1R,4a,4aS,5R,8aS)-5-[(b-D-Glucopyranosyloxy)methyl]decanhydro-5,8a-dimethyl-2-methylene-1-naphthalenyl]ethyl]-2(5H)-furanone, AS-56986, DA-56094, 1ST157228, BRD-K66516195-001-01-4, Q27293767, NEOANDROGRAPHOLIDE (CONSTITUENT OF ANDROGRAPHIS), 4-[2-[(1R,4aS,5R,8aS)-5,8a-dimethyl-2-methylidene-5-[[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]-3,4,4a,6,7,8-hexahydro-1H-naphthalen-1-yl]ethyl]-2H-uran-5-one, 5BETA,9BETAH,10ALPHA-LABDA-8(20),13-DIEN-16-OIC ACID, 18-(GLUCOSYLOXY)-15-HYDROXY-, GAMMA-LACTONE
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 126.0
Hydrogen Bond Donor Count 4.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCCC1CCC1C(C)CCC2C(CCC3CCCCC3)CCCC12
Np Classifier Class Labdane diterpenoids
Deep Smiles OC[C@H]O[C@@H]OC[C@]C)CCC[C@@][C@@H]6CCC=C)[C@H]6CCC=CCOC5=O)))))))))))))C))))))))[C@@H][C@H][C@@H]6O))O))O
Heavy Atom Count 34.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level CC1CCC2C(COC3CCCCO3)CCCC2C1CCC1CCOC1O
Classyfire Subclass Terpene glycosides
Isotope Atom Count 0.0
Molecular Complexity 811.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name 4-[2-[(1R,4aS,5R,8aS)-5,8a-dimethyl-2-methylidene-5-[[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxymethyl]-3,4,4a,6,7,8-hexahydro-1H-naphthalen-1-yl]ethyl]-2H-furan-5-one
Prediction Hob 0.0
Veber Rule True
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 2.6
Gsk 4 400 Rule False
Molecular Formula C26H40O8
Scaffold Graph Node Bond Level C=C1CCC2C(COC3CCCCO3)CCCC2C1CCC1=CCOC1=O
Prediction Swissadme 1.0
Inchi Key YGCYRQKJYWQXHG-RDNQFMDVSA-N
Silicos It Class Soluble
Fcsp3 0.8076923076923077
Logs -3.412
Rotatable Bond Count 7.0
Logd 2.784
Synonyms neoandrographolide
Esol Class Moderately soluble
Functional Groups C=C(C)C, CC1=CCOC1=O, CO, CO[C@@H](C)OC
Compound Name Neoandrographolide
Prediction Hob Swissadme 0.0
Exact Mass 480.272
Formal Charge 0.0
Monoisotopic Mass 480.272
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 480.6
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -4.0146076000000015
Inchi InChI=1S/C26H40O8/c1-15-5-8-19-25(2,14-33-24-22(30)21(29)20(28)18(13-27)34-24)10-4-11-26(19,3)17(15)7-6-16-9-12-32-23(16)31/h9,17-22,24,27-30H,1,4-8,10-14H2,2-3H3/t17-,18-,19-,20-,21+,22-,24-,25+,26+/m1/s1
Smiles C[C@]1(CCC[C@@]2([C@@H]1CCC(=C)[C@H]2CCC3=CCOC3=O)C)CO[C@H]4[C@@H]([C@H]([C@@H]([C@H](O4)CO)O)O)O
Nring 4.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Diterpenoids