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10-Hydroxycamptothecin

PubChem CID: 97226

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Compound Synonyms 10-Hydroxycamptothecin, 19685-09-7, (S)-10-Hydroxycamptothecin, Hydroxycamptothecin, 10-hydroxycamptothecine, 10-Hydroxy camptothecin, Hydroxycamptothecine, Camptothecin, hydroxy-, (4S)-4-Ethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione, (S)-4-Ethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione, Camptothecine, 10-hydroxy-, Camptothecin, 10-hydroxy-, 10-HCPT, NSC 107124, 10-Hydroxy-Camptothecin, (S)-10-Hydroxycamptothecin hydrate, UNII-9Z01632KRV, 9Z01632KRV, MFCD02093100, NSC107124, NSC-107124, CHEMBL273862, CHEBI:81395, (+)-10-HYDROXYCAMPTOTHECIN, Hydroxy camptothecine, 1H-Pyrano(3',4':6,7)indolizino(1,2-b)quinoline-3,14(4H,12H)-dione, 4-ethyl-4,9-dihydroxy-, hydrate, (S)-, 10-HYDROXYCAMPTOTHECIN [WHO-DD], (S)-4-ethyl-4,9-dihydroxy-1,12-dihydro-14H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H)-dione, 1H-Pyrano(3',4':6,7)indolizino(1,2-b)quinoline-3,14(4H,12H)-dione-,4-ethyl-4,9-dihydroxy-, (S)-, (19S)-19-ethyl-7,19-dihydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaene-14,18-dione, (20S)-4-Ethyl-4,9-dihydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione, (S)-4-Ethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione ((S)-10-Hydroxycamptothecin), 1H-PYRANO(3',4':6,7)INDOLIZINO(1,2-B)QUINOLINE-3,14(4H,12H)-DIONE, 4-ETHYL-4,9-DIHYDROXY-, (4S)-, CAMPTOTHECIN, 10-HYDROXY, 10-Hydroxy-CPT, Spectrum_001639, (+)-(S)-10-HYDROXYCAMPTOTHECIN, SpecPlus_000763, Spectrum2_001660, Spectrum3_001621, Spectrum4_001815, Spectrum5_000549, ethyl(dihydroxy)[?]dione, SCHEMBL25875, BSPBio_003281, KBioGR_002454, KBioSS_002119, DivK1c_006859, SPECTRUM1504123, SPBio_001819, HY-N0095R, KBio1_001803, KBio2_002119, KBio2_004687, KBio2_007255, KBio3_002501, DTXSID00941444, EX-A988, Camptothecine, 10-hydroxy-(8CI), BCP01385, HY-N0095, BDBM50008922, CCG-38770, s2423, s3898, AKOS015919293, AC-5502, BCP9000058, CS-5193, DB12385, (S)-10-Hydroxycamptothecin (Standard), NCGC00095986-01, NCGC00095986-02, NCGC00095986-03, NCGC00095986-04, NCGC00178165-01, AC-13221, AS-13196, NCI60_000173, SY010687, H1463, NS00018317, C17939, EN300-19810684, SR-05000002620, SR-05000002620-1, BRD-K63784565-001-02-1, BRD-K63784565-001-03-9, BRD-K63784565-001-05-4, BRD-K63784565-001-06-2, Q27155328, Z3093896188, 4-Ethyl-4,9-dihydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione, (19S)-19-ethyl-7,19-dihydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.0^{2,11}.0^{4,9}.0^{15,20}]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaene-14,18-dione, (S)-4-Ethyl-4,9-dihydroxy-1H-pyrano[3 inverted exclamation mark ,4 inverted exclamation mark :6,7]indolizino[1,2-b]quinoline-3,14-(4H,12H)-dione, (S)-4-Ethyl-4,9-dihydroxy-1H-pyrano[3',4':6,7]indolizino[1,2-b]quinoline-3,14-(4H,12H)-dione, 1H-Pyrano(3',4':6,7)indolizino(1,2-b)quinoline-3,14(4H,12H)-dione-,4-ethyl-4,9-dihydroxy-, (S)-(9CI), 1H-Pyrano[3',7]indolizino[1,2-b]quinoline-3,14(4H,12H)-dione-,4-ethyl-4,9-dihydroxy-, (S)-, 4-Ethyl-4,10-dihydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione, 4-Ethyl-4,9-dihydroxy-1,12-dihydro-4H-2-oxa-6,12a-diaza-dibenzo[b,h]fluorene-3,13-dione (10-hydroxycamptothecin), 613-598-9
Topological Polar Surface Area 100.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 27.0
Isotope Atom Count 0.0
Molecular Complexity 774.0
Database Name cmaup_ingredients;npass_chem_all;pubchem
Defined Atom Stereocenter Count 1.0
Uniprot Id P02768, P11387, n.a., Q03164, P55210, Q16637, P51450, P97697, P02791, P68871, P29466, P08684, Q92830, O42275, P81908, Q9NUW8, P0DTD1
Iupac Name (19S)-19-ethyl-7,19-dihydroxy-17-oxa-3,13-diazapentacyclo[11.8.0.02,11.04,9.015,20]henicosa-1(21),2(11),3,5,7,9,15(20)-heptaene-14,18-dione
Prediction Hob 1.0
Target Id NPT143, NPT1226, NPT93, NPT2930, NPT277, NPT109
Xlogp 0.6
Molecular Formula C20H16N2O5
Prediction Swissadme 0.0
Inchi Key HAWSQZCWOQZXHI-FQEVSTJZSA-N
Fcsp3 0.25
Logs -4.238
Rotatable Bond Count 1.0
Logd 1.327
Compound Name 10-Hydroxycamptothecin
Prediction Hob Swissadme 0.0
Exact Mass 364.106
Formal Charge 0.0
Monoisotopic Mass 364.106
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 364.4
Covalent Unit Count 1.0
Total Atom Stereocenter Count 1.0
Total Bond Stereocenter Count 0.0
Esol -3.9331319185185194
Inchi InChI=1S/C20H16N2O5/c1-2-20(26)14-7-16-17-11(5-10-6-12(23)3-4-15(10)21-17)8-22(16)18(24)13(14)9-27-19(20)25/h3-7,23,26H,2,8-9H2,1H3/t20-/m0/s1
Smiles CC[C@@]1(C2=C(COC1=O)C(=O)N3CC4=C(C3=C2)N=C5C=CC(=CC5=C4)O)O
Nring 5.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Camptotheca Acuminata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all