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Monocrotaline

PubChem CID: 9415

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Compound Synonyms monocrotaline, Crotaline, 315-22-0, Monocrotalin, (-)-Monocrotaline, NCI-C56462, CCRIS 416, CHEBI:6980, HSDB 3513, A 6080, Retronecine cyclic 2,3-dihydroxy-2,3,4-trimethylglutarate, UNII-73077K8HYV, BRN 0048732, MLS002153902, DTXSID9020902, 73077K8HYV, (13-alpha,14-alpha)-14,19-Dihydro-12,13-dihydroxy-20-norcrotalanan-11,15-dione, MONOCROTALINE [MI], 14,19-Dihydro-12,13-dihydroxy-20-norcrotolanan-11,15-dione, MONOCROTALINE [HSDB], MONOCROTALINE [IARC], NSC 28693, DTXCID50902, 20-Norcrotalanan-11,15-dione, 14,19-dihydro-12,13-dihydroxy-, (13alpha,14alpha)-, (3R,4R,5R,13aR,13bR)-4,5-dihydroxy-3,4,5-trimethyl-4,5,8,10,12,13,13a,13b-octahydro-2H-[1,6]dioxacycloundecino[2,3,4-gh]pyrrolizine-2,6(3H)-dione, 4-27-00-06660 (Beilstein Handbook Reference), 12-beta,13-beta-Dihydroxy-12-alpha,13-alpha,14-alpha-trimethylcrotal-1-enine, NSC-28693, 14,19-Dihydro-12,13-dihydroxy(13-alpha,14-alpha)-20-norcrotalanan-11,15-dione, (2,3,4-gh)pyrrolizine-2,6(3H)-dione, (4,5,8,10,12,13,13a,13b)-octahydro-4,5-dihydroxy-3,4,5-trimethyl-2H-(1,6)dioxacycloundecino-, NCGC00164256-01, 20-Norcrotalanan-11,15-dione, 14,19-dihydro-12,13-dihydroxy-, (13-alpha,14-alpha)-, MONOCROTALINE (IARC), (1R,4R,5R,6R,16R)-5,6-dihydroxy-4,5,6-trimethyl-2,8-dioxa-13-azatricyclo[8.5.1.013,16]hexadec-10-ene-3,7-dione, 2H-(1,6)Dioxacycloundecino(2,3,4-gh)pyrrolizine-2,6(3H)-dione, 4,5,8,10,12,13,13a,13b-octahydro-4,5-dihydroxy-3,4,5-trimethyl-, (3R,4R,5R,13aR,13bR)-, 2H-[1,6]Dioxacycloundecino[2,3,4-gh]pyrrolizine-2,6(3H)-dione, 4,5,8,10,12,13,13a,13b-octahydro-4,5-dihydroxy-3,4,5-trimethyl-, (3R,4R,5R,13aR,13bR)-, 2H-(1,6)DIOXACYCLOUNDECINO(2,3,4-GH)PYRROLIZINE-2,6(3H)-DIONE, 4,5,8,10,12,13,13A,13B-OCTAHYDRO-4,5-DIHYDROXY-3,4,5-TRIMETHYL-, (3R-(3R*,4R*,5R*,13AR*,13BR*))-, 20-Norcrotalanan-11,15-dione, 14,19-dihydro-12,13-dihydroxy-, (13.alpha.,14.alpha.)-, SR-01000838886, (1R,4R,5R,6R,16R)-5,6-dihydroxy-4,5,6-trimethyl-2,8-dioxa-13-azatricyclo(8.5.1.013,16)hexadec-10-ene-3,7-dione, (3R,4R,5R,13aR,13bR)-4,5-dihydroxy-3,4,5-trimethyl-4,5,8,10,12,13,13a,13b-octahydro-2H-(1,6)dioxacycloundecino(2,3,4-gh)pyrrolizine-2,6(3H)-dione, 2H-(1,6)DIOXACYCLOUNDECINO(2,3,4-gh)PYRROLIZINE-2,6(3H)-DIONE, 4,5,8,10,12,13,13a,13b-OCTAHYDRO-4,5-DIHYDROXY-3,4,5-TRIMETHYL-,(3R,4R,5R,13aR,13bR)-, 2H-[1,6]DIOXACYCLOUNDECINO[2,3,4-gh]PYRROLIZINE-2,6(3H)-DIONE, 4,5,8,10,12,13,13a,13b-OCTAHYDRO-4,5-DIHYDROXY-3,4,5-TRIMETHYL-,(3R,4R,5R,13aR,13bR)-, CAS-315-22-0, Prestwick_338, MFCD00084656, Spectrum_001224, Prestwick0_000603, Prestwick1_000603, Prestwick2_000603, Prestwick3_000603, Spectrum2_000906, Spectrum3_000947, Spectrum4_001057, Spectrum5_001233, BSPBio_000506, KBioGR_001354, KBioSS_001704, DivK1c_000959, SCHEMBL164486, SPECTRUM1502252, SPBio_000752, SPBio_002725, BPBio1_000558, CHEMBL521035, MEGxp0_001899, ACon0_000305, ACon1_000179, HMS502P21, KBio1_000959, KBio2_001704, KBio2_004272, KBio2_006840, KBio3_002014, (13-.alpha.,14-.alpha.)-14,19-Dihydro-12,13-dihydroxy-20-norcrotalanan-11,15-dione, 12.beta.,13.beta.-Dihydroxy-12.alpha.,13.alpha.,14.alpha.-trimethylcrotal-1-enine, 14,19-Dihydro-12,13-dihydroxy(13.alpha.,14.alpha.)-20-norcrotalanan-11,15-dione, 2H-(1,6)Dioxacycloundecino(2,3,4-gh)pyrrolizine, 20-norcrotalanan-11,15-dione deriv., 2H-[1,6]Dioxacycloundecino[2,3,4-gh]pyrrolizine, 20-norcrotalanan-11,15-dione deriv., Monocrotaline, analytical standard, NINDS_000959, HMS1569J08, HMS1921P04, HMS2096J08, HMS2235J12, HY-N0750, Tox21_112094, Tox21_201509, Tox21_302874, BDBM50480309, CCG-39621, s3812, AKOS015969712, AKOS032962048, Tox21_112094_1, CS-6164, FM64904, FS-5652, SDCCGMLS-0066675.P001, IDI1_000959, NCGC00179538-01, NCGC00179538-02, NCGC00179538-03, NCGC00256518-01, NCGC00259060-01, NCGC00262539-03, 1ST14173, AC-34918, SMR001233251, JACS 72: 158 (1950), SR-01000838886-3, SR-01000838886-4, BRD-K65508953-001-05-5, BRD-K65508953-001-08-9, Q27107379, Retronecine cyclic 2,3dihydroxy2,3,4trimethylglutarate, 12beta,13betaDihydroxy12alpha,13alpha,14alphatrimethylcrotal1enine, (13alpha,14alpha)14,19Dihydro12,13dihydroxy20norcrotalanan11,15dione, 12beta,13beta-Dihydroxy-12alpha,13alpha,14alpha-trimethylcrotal-1-enine, 14,19Dihydro12,13dihydroxy(13alpha,14alpha)20norcrotalanan11,15dione, (13alpha, 14alpha)-14,19-Dihydro-12,13-dihydroxy-20-norcrotolanan-11,15-dione, 14,19-Dihydro-12,13-dihydroxy(13alpha,14alpha)-20-norcrotalanan-11,15-dione, 20Norcrotalanan11,15dione, 14,19dihydro12,13dihydroxy, (13alpha,14alpha), (1R,4R,5R,6R,16R)-5,6-dihydroxy-4,5,6-trimethyl-2,8-dioxa-13-azatricyclo[8.5.1.0??,??]hexadec-10-ene-3,7-dione, (2,3,4-GH)PYRROLIZINE-2,6(3H)-DIONE, (4,5,8,10,12,13,13A,13B-OCTAHYDRO-4,5-DIHYDROXY-3,4,5-TRIMETHYL-2H-(1,6)DIOXACYCLOUNDECINO-, (3R,4R,5R,8a1R,13aR)-4,5-Dihydroxy-3,4,5-trimethyl-4,5,8,8a1,10,12,13,13a-octahydro-2H-[1,6]dioxacycloundecino[2,3,4-gh]pyrrolizine-2,6(3H)-dione, (3R,4R,8a1R,13aR)-4,5-Dihydroxy-3,4,5-trimethyl-4,5,8,8a1,10,12,13,13a-octahydro-2H-[1,6]dioxacycloundecino[2,3,4-gh]pyrrolizine-2,6(3H)-dione, 109525-74-8, 20-Norcrotalanan-11,15-dione, 14,19-dihydro-12,13-dihydroxy-, (13-alpha,14-alpha)-(9CI), 628-506-2, rel-(3R,4R,5R,8a1R,13aR)-4,5-Dihydroxy-3,4,5-trimethyl-4,5,8,8a1,10,12,13,13a-octahydro-2H-[1,6]dioxacycloundecino[2,3,4-gh]pyrrolizine-2,6(3H)-dione
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 96.3
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCCC(C)CC2CCC3CCC(CC1)C32
Np Classifier Class Pyrrolizidine alkaloids
Deep Smiles O=CO[C@@H]CCN[C@@H]5C=CC5))COC=O)[C@][C@][C@H]%14C))C)O))C)O
Heavy Atom Count 23.0
Classyfire Class Pyrrolizines
Scaffold Graph Node Level OC1CCCC(O)OC2CCN3CCC(CO1)C23
Isotope Atom Count 0.0
Molecular Complexity 575.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 5.0
Uniprot Id Q72547, P00811, P10828, O75496, P04637, O42275, P81908, Q9NUW8, Q9Y6L6, Q9NPD5, n.a., P04792
Iupac Name (1R,4R,5R,6R,16R)-5,6-dihydroxy-4,5,6-trimethyl-2,8-dioxa-13-azatricyclo[8.5.1.013,16]hexadec-10-ene-3,7-dione
Prediction Hob 1.0
Veber Rule True
Classyfire Superclass Organoheterocyclic compounds
Xlogp -0.7
Gsk 4 400 Rule True
Molecular Formula C16H23NO6
Scaffold Graph Node Bond Level O=C1CCCC(=O)OC2CCN3CC=C(CO1)C23
Prediction Swissadme 0.0
Inchi Key QVCMHGGNRFRMAD-XFGHUUIASA-N
Silicos It Class Soluble
Fcsp3 0.75
Logs -1.96
Rotatable Bond Count 0.0
Logd 0.907
Synonyms crotaline, monocrotaline, pyrrolizidine alkaloid
Esol Class Very soluble
Functional Groups CC=C(C)C, CN(C)C, CO, COC(C)=O
Compound Name Monocrotaline
Prediction Hob Swissadme 0.0
Exact Mass 325.153
Formal Charge 0.0
Monoisotopic Mass 325.153
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 325.36
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -1.3973382000000005
Inchi InChI=1S/C16H23NO6/c1-9-13(18)23-11-5-7-17-6-4-10(12(11)17)8-22-14(19)16(3,21)15(9,2)20/h4,9,11-12,20-21H,5-8H2,1-3H3/t9-,11+,12+,15+,16-/m0/s1
Smiles C[C@H]1C(=O)O[C@@H]2CCN3[C@@H]2C(=CC3)COC(=O)[C@]([C@]1(C)O)(C)O
Nring 3.0
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Ornithine alkaloids

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