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Norscopolamine

PubChem CID: 92989

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Compound Synonyms Norhyoscine, norscopolamine, 4684-28-0, (S)-norscopolamine, Nor Scopolamine, G880Z17K5S, EINECS 225-139-6, NORSCOPOLAMINE [USP-RS], EC 225-139-6, NORSCOPOLAMINE [USP IMPURITY], [7(S)-(1alpha,.2beta,4beta,5alpha,7beta)]-3-oxa-9-azatricyclo[3.3.1.02,4]non-7-yl (hydroxymethyl)phenylacetate, (7(S)-(1alpha,2beta,4beta,5alpha,7beta))-3-Oxa-9-azatricyclo(3.3.1.02,4)non-7-yl (hydroxymethyl)phenylacetate, NORSCOPOLAMINE (USP-RS), NORSCOPOLAMINE (USP IMPURITY), (7(S)-(1alpha,.2beta,4beta,5alpha,7beta))-3-Oxa-9-azatricyclo(3.3.1.02,4)non-7-yl (hydroxymethyl)phenylacetate, 1.ALPHA.H,5.ALPHA.H-NORTROPAN-3.ALPHA.-OL, 6.BETA.,7.BETA.-EPOXY-, (-)-TROPATE (ESTER), BENZENEACETIC ACID, .ALPHA.-(HYDROXYMETHYL)-, (1.ALPHA.,2.BETA.,4.BETA.,5.ALPHA.,7.BETA.)-3-OXA-9-AZATRICYCLO(3.3.1.02,4)NON-7-YL ESTER, (.ALPHA.S)-, BENZENEACETIC ACID, .ALPHA.-(HYDROXYMETHYL)-, 3-OXA-9-AZATRICYCLO(3.3.1.02,4)NON-7-YL ESTER, (7(S)-(1.ALPHA.,2.BETA.,4.BETA.,5.ALPHA.,7.BETA.))-, Benzeneacetic acid, alpha-(hydroxymethyl)-, 3-oxa-9-azatricyclo(3.3.1.0(2,4))non-7-yl ester, (7(S)-(1alpha,2beta,4beta,5alpha,7beta))-, DTXSID30963679, UNII-G880Z17K5S, Benzeneacetic acid, a-(hydroxymethyl)-, (1a,2ss,4ss,5a,7ss)-3-oxa-9-azatricyclo[3.3.1.02,4]non-7-yl ester, (aS)-, 1aH,5aH-Nortropan-3a-ol, 6ss,7ss-epoxy-, (-)-tropate (ester) (8CI), Benzeneacetic acid, a-(hydroxymethyl)-, 3-oxa-9-azatricyclo[3.3.1.02,4]non-7-yl ester, [7(S)-(1a,2ss,4ss,5a,7ss)]-, Norscopolamine (7CI), Norhyoscine, DTXCID501766159, MFCD22666251, AKOS027326579, NS00003138, 1H,5H-Nortropan-3-ol, 6,7-epoxy-, (-)-tropate (ester), Norhyoscine, 1ALPHAH,5ALPHAH-NORTROPAN-3ALPHA-OL, 6BETA,7BETA-EPOXY-, (-)-TROPATE (ESTER), (1R,2R,4S,5S)-3-oxa-9-azatricyclo[3.3.1.0?,?]nonan-7-yl (2S)-3-hydroxy-2-phenylpropanoate, BENZENEACETIC ACID, ALPHA-(HYDROXYMETHYL)-, (1ALPHA,2BETA,4BETA,5ALPHA,7BETA)-3-OXA-9-AZATRICYCLO(3.3.1.02,4)NON-7-YL ESTER, (ALPHAS)-, BENZENEACETIC ACID, ALPHA-(HYDROXYMETHYL)-, 3-OXA-9-AZATRICYCLO(3.3.1.02,4)NON-7-YL ESTER, (7(S)-(1ALPHA,2BETA,4BETA,5ALPHA,7BETA))-
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 71.1
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC(CC1CCCCC1)CC1CC2CC(C1)C1CC21
Np Classifier Class Tropane alkaloids
Deep Smiles OC[C@H]cccccc6))))))C=O)OCC[C@@H]N[C@H]C6)[C@@H][C@H]5O3
Heavy Atom Count 21.0
Classyfire Class Hydroxy acids and derivatives
Scaffold Graph Node Level OC(CC1CCCCC1)OC1CC2NC(C1)C1OC21
Classyfire Subclass Beta hydroxy acids and derivatives
Isotope Atom Count 0.0
Molecular Complexity 393.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name [(1S,2S,4R,5R)-3-oxa-9-azatricyclo[3.3.1.02,4]nonan-7-yl] (2S)-3-hydroxy-2-phenylpropanoate
Veber Rule True
Classyfire Superclass Organic acids and derivatives
Xlogp 0.9
Gsk 4 400 Rule True
Molecular Formula C16H19NO4
Scaffold Graph Node Bond Level O=C(Cc1ccccc1)OC1CC2NC(C1)C1OC21
Inchi Key MOYZEMOPQDTDHA-YQYZCKNZSA-N
Silicos It Class Soluble
Rotatable Bond Count 5.0
Synonyms norhyoscine, norscopolamine
Esol Class Very soluble
Functional Groups CNC, CO, COC(C)=O, C[C@@H]1O[C@@H]1C
Compound Name Norscopolamine
Exact Mass 289.131
Formal Charge 0.0
Monoisotopic Mass 289.131
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 289.33
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C16H19NO4/c18-8-11(9-4-2-1-3-5-9)16(19)20-10-6-12-14-15(21-14)13(7-10)17-12/h1-5,10-15,17-18H,6-8H2/t10?,11-,12-,13+,14-,15+/m1/s1
Smiles C1[C@@H]2[C@@H]3[C@@H](O3)[C@@H](N2)CC1OC(=O)[C@H](CO)C4=CC=CC=C4
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Ornithine alkaloids

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