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methyl (12R,13S,15S,17S)-13-[(1S)-1-hydroxyethyl]-4-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2(7),3,5,8(18)-tetraene-17-carboxylate

PubChem CID: 90680624

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Compound Synonyms CHEMBL3286763
Topological Polar Surface Area 72.7
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 28.0
Isotope Atom Count 0.0
Molecular Complexity 630.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name methyl (12R,13S,15S,17S)-13-[(1S)-1-hydroxyethyl]-4-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2(7),3,5,8(18)-tetraene-17-carboxylate
Prediction Hob 1.0
Xlogp 1.8
Molecular Formula C22H28N2O4
Prediction Swissadme 1.0
Inchi Key QRNYDROIKQEMOH-YPQVPPDESA-N
Fcsp3 0.5909090909090909
Logs -1.746
Rotatable Bond Count 4.0
Logd 2.764
Compound Name methyl (12R,13S,15S,17S)-13-[(1S)-1-hydroxyethyl]-4-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2(7),3,5,8(18)-tetraene-17-carboxylate
Prediction Hob Swissadme 1.0
Exact Mass 384.205
Formal Charge 0.0
Monoisotopic Mass 384.205
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 384.5
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Esol -3.3190083428571437
Inchi InChI=1S/C22H28N2O4/c1-12(25)17-8-13-10-22(21(26)28-3)19(17)23-7-6-16-15-5-4-14(27-2)9-18(15)24(11-13)20(16)22/h4-5,9,12-13,17,19,23,25H,6-8,10-11H2,1-3H3/t12-,13-,17+,19+,22-/m0/s1
Smiles C[C@@H]([C@H]1C[C@H]2C[C@@]3([C@@H]1NCCC4=C3N(C2)C5=C4C=CC(=C5)OC)C(=O)OC)O
Nring 5.0
Defined Bond Stereocenter Count 0.0