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methyl (12R,13R,15S,17S)-13-ethyl-4-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-5-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2,4,6,8(18)-tetraene-17-carboxylate

PubChem CID: 90680618

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Compound Synonyms CHEMBL3286757
Topological Polar Surface Area 118.0
Hydrogen Bond Donor Count 3.0
Heavy Atom Count 54.0
Isotope Atom Count 0.0
Molecular Complexity 1480.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name methyl (12R,13R,15S,17S)-13-ethyl-4-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-5-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2,4,6,8(18)-tetraene-17-carboxylate
Prediction Hob 0.0
Xlogp 4.6
Molecular Formula C44H54N4O6
Prediction Swissadme 0.0
Inchi Key BRLRROSLMJEGJL-SIFBDTQASA-N
Fcsp3 0.5454545454545454
Logs -4.373
Rotatable Bond Count 8.0
Logd 4.797
Compound Name methyl (12R,13R,15S,17S)-13-ethyl-4-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-5-methoxy-1,11-diazapentacyclo[13.3.1.02,7.08,18.012,17]nonadeca-2,4,6,8(18)-tetraene-17-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 734.404
Formal Charge 0.0
Monoisotopic Mass 734.404
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 734.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 1.0
Esol -7.025882266666668
Inchi InChI=1S/C44H54N4O6/c1-7-25-15-24-20-43(41(50)53-5)39(25)45-14-13-28-29-18-36(52-4)30(17-35(29)48(21-24)40(28)43)31-16-33-26(8-2)22-47(3)37(44(33,23-49)42(51)54-6)19-32-27-11-9-10-12-34(27)46-38(31)32/h8-12,17-18,24-25,31,33,37,39,45-46,49H,7,13-16,19-23H2,1-6H3/b26-8-/t24-,25+,31-,33+,37-,39+,43-,44-/m0/s1
Smiles CC[C@@H]1C[C@H]2C[C@@]3([C@@H]1NCCC4=C3N(C2)C5=CC(=C(C=C45)OC)[C@@H]6C[C@@H]7/C(=C\C)/CN([C@H]([C@@]7(CO)C(=O)OC)CC8=C6NC9=CC=CC=C89)C)C(=O)OC
Nring 9.0
Defined Bond Stereocenter Count 1.0