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Pseudoaconitine

PubChem CID: 90478913

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Compound Synonyms Acraconitine, Nepaline, Nepaul aconitine, Pseudaconitine, Pseudoaconitine, Feraconitne, Nepal aconitine, 127-29-7, English aconitine, 8-ACETYL LUDACONITINE, Feraconitine, UNII-5483BY72RT, 5483BY72RT, BRN 0075720, PSEUDOACONITINE [MI], DTXSID90894011, 5-21-06-00309 (Beilstein Handbook Reference), [(1S,2R,3R,4R,5S,6S,8R,9R,10R,13R,14R,16S,17S,18R)-8-acetyloxy-11-ethyl-5,14-dihydroxy-6,16,18-trimethoxy-13-(methoxymethyl)-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-4-yl] 3,4-dimethoxybenzoate, Aconitane-3,8,13,14-tetrol, 20-ethy-4-(methoxymethyl)-1,6,16-trimethoxy, 8-acetate, 14-(3,4-dimethoxybenzoate), (1-alpha,3-alpha,6-alpha,14-alpha,16-beta)-, ACONITANE-3,8,13,14-TETROL, 20-ETHYL-1,6,16-TRIMETHOXY-4-(METHOXYMETHYL)-, 8-ACETATE 14-(3,4-DIMETHOXYBENZOATE), (1.ALPHA.,3.ALPHA.,6.ALPHA.,14.ALPHA.,16.BETA.)-, DTXCID401324055, Q27261185, ACONITANE-3,8,13,14-TETROL, 20-ETHYL-1,6,16-TRIMETHOXY-4-(METHOXYMETHYL)-, 8-ACETATE 14-(3,4-DIMETHOXYBENZOATE), (1ALPHA,3ALPHA,6ALPHA,14ALPHA,16BETA)-
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 152.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CC1C2CCC3C4CC5C6CCCC5(C4CC6)C(C2)C13)C1CCCCC1
Np Classifier Class Terpenoid alkaloids
Deep Smiles COC[C@]CNCC))[C@H][C@][C@@H]6[C@@H]OC))[C@@H]5[C@@][C@@H][C@H]7C[C@@][C@@H]5OC=O)cccccc6)OC)))OC)))))))))[C@H]C7)OC)))O)))))OC=O)C)))))))[C@H]C[C@H]8O)))OC
Heavy Atom Count 49.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC(OC1C2CCC3C4CC5C6CCCC5(C(C2)C31)C4NC6)C1CCCCC1
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1290.0
Database Name cmaup_ingredients;imppat_phytochem;pubchem
Defined Atom Stereocenter Count 14.0
Iupac Name [(1S,2R,3R,4R,5S,6S,8R,9R,10R,13R,14R,16S,17S,18R)-8-acetyloxy-11-ethyl-5,14-dihydroxy-6,16,18-trimethoxy-13-(methoxymethyl)-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-4-yl] 3,4-dimethoxybenzoate
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 1.2
Gsk 4 400 Rule False
Molecular Formula C36H51NO12
Scaffold Graph Node Bond Level O=C(OC1C2CCC3C4CC5C6CCCC5(C(C2)C31)C4NC6)c1ccccc1
Prediction Swissadme 0.0
Inchi Key YVPYMQHYESYLIR-HZKWNRCISA-N
Silicos It Class Moderately soluble
Fcsp3 0.7777777777777778
Logs -3.715
Rotatable Bond Count 13.0
Logd 1.757
Synonyms feraconitine, pseudaconitine
Esol Class Moderately soluble
Functional Groups CC(=O)OC, CN(C)C, CO, COC, cC(=O)OC, cOC
Compound Name Pseudoaconitine
Prediction Hob Swissadme 0.0
Exact Mass 689.341
Formal Charge 0.0
Monoisotopic Mass 689.341
Hydrogen Bond Acceptor Count 13.0
Molecular Weight 689.8
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 14.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Esol -4.099066044897961
Inchi InChI=1S/C36H51NO12/c1-9-37-16-33(17-42-3)23(39)13-24(45-6)36-20-14-34(41)25(46-7)15-35(49-18(2)38,27(30(36)37)28(47-8)29(33)36)26(20)31(34)48-32(40)19-10-11-21(43-4)22(12-19)44-5/h10-12,20,23-31,39,41H,9,13-17H2,1-8H3/t20-,23-,24+,25+,26-,27+,28+,29-,30-,31-,33+,34+,35-,36+/m1/s1
Smiles CCN1C[C@@]2([C@@H](C[C@@H]([C@@]34[C@@H]2[C@H]([C@@H]([C@H]31)[C@]5(C[C@@H]([C@]6(C[C@@H]4[C@@H]5[C@H]6OC(=O)C7=CC(=C(C=C7)OC)OC)O)OC)OC(=O)C)OC)OC)O)COC
Nring 7.0
Np Classifier Biosynthetic Pathway Alkaloids, Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Pseudoalkaloids

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