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cleistanthin E

PubChem CID: 86583369

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Compound Synonyms cleistanthin E, CHEBI:84416, 9-(1,3-benzodioxol-5-yl)-6,7-dimethoxy-1-oxo-1,3-dihydronaphtho[2,3-c]furan-4-yl 2,3,5-tri-O-methyl-beta-D-xylofuranosyl-(1->4)-2,3-di-O-methyl-beta-D-xylopyranosyl-(1->4)-beta-D-glucopyranoside, 9-(1,3-benzodioxol-5-yl)-4-((2S,3R,4R,5S,6R)-5-((2S,3R,4S,5R)-5-((2S,3R,4S,5R)-3,4-dimethoxy-5-(methoxymethyl)oxolan-2-yl)oxy-3,4-dimethoxyoxan-2-yl)oxy-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl)oxy-6,7-dimethoxy-3H-benzo(f)(2)benzofuran-1-one, 9-(1,3-benzodioxol-5-yl)-4-[(2S,3R,4R,5S,6R)-5-[(2S,3R,4S,5R)-5-[(2S,3R,4S,5R)-3,4-dimethoxy-5-(methoxymethyl)oxolan-2-yl]oxy-3,4-dimethoxyoxan-2-yl]oxy-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-6,7-dimethoxy-3H-benzo[f][2]benzofuran-1-one, 9-(1,3-benzodioxol-5-yl)-6,7-dimethoxy-1-oxo-1,3-dihydronaphtho(2,3-c)furan-4-yl 2,3,5-tri-O-methyl-beta-D-xylofuranosyl-(1->4)-2,3-di-O-methyl-beta-D-xylopyranosyl-(1->4)-beta-D-glucopyranoside, Q27157743
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 225.0
Hydrogen Bond Donor Count 3.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCC2C(CC3CCC(CC4CCC(CC5CCCC5)CC4)CC3)C3CCCCC3C(C3CCC4CCCC4C3)C12
Np Classifier Class Arylnaphthalene and aryltetralin lignans
Deep Smiles COC[C@H]O[C@H][C@@H][C@H]5OC)))OC)))O[C@@H]CO[C@H][C@@H][C@H]6OC)))OC)))O[C@@H][C@@H]CO))O[C@H][C@@H][C@H]6O))O))OccCOC=O)c5ccc9ccOC))cc6)OC)))))))cccccc6)OCO5
Heavy Atom Count 62.0
Classyfire Class Organooxygen compounds
Scaffold Graph Node Level OC1OCC2C(OC3CCC(OC4CCC(OC5CCCO5)CO4)CO3)C3CCCCC3C(C3CCC4OCOC4C3)C12
Classyfire Subclass Carbohydrates and carbohydrate conjugates
Isotope Atom Count 0.0
Molecular Complexity 1450.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 13.0
Iupac Name 9-(1,3-benzodioxol-5-yl)-4-[(2S,3R,4R,5S,6R)-5-[(2S,3R,4S,5R)-5-[(2S,3R,4S,5R)-3,4-dimethoxy-5-(methoxymethyl)oxolan-2-yl]oxy-3,4-dimethoxyoxan-2-yl]oxy-3,4-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-6,7-dimethoxy-3H-benzo[f][2]benzofuran-1-one
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Organic oxygen compounds
Xlogp 0.9
Gsk 4 400 Rule False
Molecular Formula C42H52O20
Scaffold Graph Node Bond Level O=C1OCc2c1c(-c1ccc3c(c1)OCO3)c1ccccc1c2OC1CCC(OC2CCC(OC3CCCO3)CO2)CO1
Prediction Swissadme 0.0
Inchi Key VBUYDYFOLFVYET-YSGUZRDFSA-N
Silicos It Class Moderately soluble
Fcsp3 0.5952380952380952
Logs -4.998
Rotatable Bond Count 16.0
Logd 2.093
Synonyms cleistanthin e
Esol Class Moderately soluble
Functional Groups CO, COC, CO[C@@H](C)OC, CO[C@H](C)OC, c1cOCO1, cC(=O)OC, cOC, cO[C@@H](C)OC
Compound Name cleistanthin E
Prediction Hob Swissadme 0.0
Exact Mass 876.305
Formal Charge 0.0
Monoisotopic Mass 876.305
Hydrogen Bond Acceptor Count 20.0
Molecular Weight 876.8
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 13.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Esol -4.978487341935484
Inchi InChI=1S/C42H52O20/c1-47-15-27-35(50-4)38(53-7)42(59-27)60-28-16-55-41(37(52-6)36(28)51-5)62-34-26(13-43)58-40(32(45)31(34)44)61-33-20-12-24(49-3)23(48-2)11-19(20)29(30-21(33)14-54-39(30)46)18-8-9-22-25(10-18)57-17-56-22/h8-12,26-28,31-32,34-38,40-45H,13-17H2,1-7H3/t26-,27-,28-,31-,32-,34-,35+,36+,37-,38-,40+,41+,42+/m1/s1
Smiles COC[C@@H]1[C@@H]([C@H]([C@@H](O1)O[C@@H]2CO[C@H]([C@@H]([C@H]2OC)OC)O[C@@H]3[C@H](O[C@H]([C@@H]([C@H]3O)O)OC4=C5COC(=O)C5=C(C6=CC(=C(C=C64)OC)OC)C7=CC8=C(C=C7)OCO8)CO)OC)OC
Nring 8.0
Np Classifier Biosynthetic Pathway Shikimates and Phenylpropanoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Lignans

  • 1. Outgoing r'ship FOUND_IN to/from Cleistanthus Collinus (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all