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Lamivudine

PubChem CID: 60825

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Compound Synonyms lamivudine, 134678-17-4, Epivir, Zeffix, Heptovir, Epivir-HBV, Hepitec, 136891-12-8, 2',3'-Dideoxy-3'-thiacytidine, BCH-189, 3TC, Heptodin, (-)-2'-Deoxy-3'-thiacytidine, 4-amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)pyrimidin-2(1H)-one, GR-109714X, VIROLAM, GR109714X, 3'-Thia-2',3'-dideoxycytidine, Lamivudine teva, beta-L-2',3'-Dideoxy-3'-thiacytidine, beta-L-3'-Thia-2',3'-dideoxycytidine, 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2-one, GR 109714X, (-)-BCH-189, (-)NGPB-21, Epivir (TN), BCH 189, (-)-, Lamivudina, Lamivudinum, BCH189, (-)-BCH 189, HSDB 7155, 4-Amino-1-(cis-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)pyrimidin-2(1H)-one, 4-AMINO-1-[(2R,5S)-2-(HYDROXYMETHYL)-1,3-OXATHIOLAN-5-YL]-1,2-DIHYDROPYRIMIDIN-2-ONE, 4-AMINO-1-[(2R,5S)-2-(HYDROXYMETHYL)-1,3-OXATHIOLAN-5-YL]-2(1H)-PYRIMIDINONE, (-)-1-((2R,5S)-2-(Hydroxymethyl)-1,3-oxathiolan-5-yl)cytosine, CCRIS 9274, CHEBI:63577, Lamivudine [USAN:USP:INN:BAN], LAMIVUDINE [MI], 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2(1H)-one, LAMIVUDINE [INN], LAMIVUDINE [JAN], LAMIVUDINE [HSDB], LAMIVUDINE [USAN], MFCD00869739, LAMIVUDINE [VANDF], 2T8Q726O95, NSC-760061, LAMIVUDINE [MART.], CIS-LAMIVUDINE, LAMIVUDINE [USP-RS], LAMIVUDINE [WHO-DD], LAMIVUDINE [WHO-IP], LAMIVUDINE [EMA EPAR], 2(1H)-Pyrimidinone, 4-amino-1-(2-(hydroxymethyl)-1,3-oxathiolan-5-yl)-, (2R-cis)-, DTXSID7023194, LAMIVUDINE [EP IMPURITY], LAMIVUDINE [ORANGE BOOK], LAMIVUDINE [EP MONOGRAPH], KIVEXA COMPONENT LAMIVUDINE, LAMIVUDINE [USP MONOGRAPH], (-)-1-[(2R,5S)-2-(Hydroxymethyl)-1,3-oxathiolan-5-yl]cytosine, EPZICOM COMPONENT LAMIVUDINE, TEMIXYS COMPONENT LAMIVUDINE, TRIUMEQ COMPONENT LAMIVUDINE, LAMIVUDINUM [WHO-IP LATIN], COMBIVIR COMPONENT LAMIVUDINE, LAMIVUDINE TEVA PHARMA B.V., TRIZIVIR COMPONENT LAMIVUDINE, 4-Amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)-2(1H)-pyrimidinone, DELSTRIGO COMPONENT LAMIVUDINE, NSC 760061, EMTRICITABINE IMPURITY C [WHO-IP], Heptivir, Lamivir, Zefix, BCH 189, LAMIVUDINE (MART.), LAMIVUDINE (USP-RS), LAMIVUDINE/ZIDOVUDINE TEVA COMPONENT LAMIVUDINE, LAMIVUDINE (EP IMPURITY), LAMIVUDINE (EP MONOGRAPH), Lamivudine [USAN:BAN:INN], LAMIVUDINE (USP MONOGRAPH), Lamivudine (USAN:USP:INN:BAN), (-)-(2'R,5'S)-1-[2'-Hydroxymethyl-5'-(1,3-oxathiolanyl)]cytosine, 3TC Lamivudine, Epivir HBV, 2(1H)-Pyrimidinone, 4-amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)-, 2(1H)-Pyrimidinone, 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-, Lamivudine, 3TC, Epivir(TM), 4-AMINO-1-((2R,5S)-2-(HYDROXYMETHYL)-1,3-OXATHIOLAN-5-YL)PYRIMIDIN-2(1H)-ONE [WHO-IP], HHA & Lamivudine, Lamivudine & GNA, SMR000466319, DTHC, CHEMBL141, 2',3' Dideoxy 3' thiacytidine, DRG-0126, 3TC and NV-01, 3TC, 2',3'-Dideoxy-3'-thiacytidine, (-)-BCH-189, (-)-SddC, Lamivudine (JAN/USP/INN), 1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)cytosine, 1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]cytosine, 3TC & GNA, 3TC & SST, HHA & 3TC, lamivudine oral, (+/-)-SddC, NSC620753, UNII-2T8Q726O95, 4-amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)-1,2-dihydropyrimidin-2-one, 4-amino-1-((2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl)pyrimidin-2-one, BCH-790, NCGC00159341-04, GG-714, MFCD00870542, Lamivudine (Standard), Lamivudine (EPIVIR), CPD000466319, (+/-)-3TC, (+/-)-BCH-189, (2R-cis)-4-Amino-1-, MLS000759424, MLS001424097, MLS006011910, BIDD:GT0033, SCHEMBL109675, EMTRICITABINE IMPURITY C, Lamivudine - Bio-X trade mark, GTPL12673, HY-B0250R, J05AF05, DTXCID001508532, HMS2051D21, HMS3259F08, HMS3713C16, HY-B0250, BBL033871, BDBM50366817, s1706, STK801940, lamivudine & TNF-alpha & IFN-gamma, TELURA COMPONENT OF LAMIVUDINE, AKOS005622556, AKOS015854841, LAMIVUDINE COMPONENT OF EPZICOM, LAMIVUDINE COMPONENT OF TEMIXYS, LAMIVUDINE COMPONENT OF TRIUMEQ, Lamivudine, >=98% (HPLC), powder, (-)-BCH189, AC-1416, CCG-100984, DB00709, KS-1073, LAMIVUDINE COMPONENT OF COMBIVIR, LAMIVUDINE COMPONENT OF DUTREBIS, LAMIVUDINE COMPONENT OF TRIZIVIR, NC00234, NC00705, NL06295, LAMIVUDINE COMPONENT OF DELSTRIGO, NCGC00159341-05, NCGC00159341-18, NCGC00159341-20, BL164607, L0217, NS00007004, rac-cis-Lamivudine ((2RS,5SR)-Lamivudine), SW197614-3, C07065, D00353, EN300-123034, Lamivudine 100 microg/mL in Acetonitrile:Water, P17147, AB00639995-06, AB00639995-08, AB00639995_09, Q422631, SR-01000759420, SR-01000759420-5, BRD-K02992638-001-11-8, LAMIVUDINE COMPONENT OF LAMIVUDINE/ZIDOVUDINE TEVA, Z1509637175, Lamivudine, British Pharmacopoeia (BP) Reference Standard, Lamivudine, European Pharmacopoeia (EP) Reference Standard, (2R,5S)-1-[2-(Hydroxymethyl)-1,3-oxathiolan-5-yl]cytosine, .beta.-L-(-)-2',3'-dideoxy-3'-thiacytidine & Sho-Saiko-To, Lamivudine, United States Pharmacopeia (USP) Reference Standard, (+/-) (Cis)-1-[2-(Hydroxymethyl)-1,3-oxathiolan-5-yl]cytosine, (-)-L-2',3'-DIDEOXY-3'-THIACYTIDINE, LAMIVUDINE, EPIVIR, Lamivudine, 1.0 mg/mL in methanol, certified reference material, Lamivudine, Pharmaceutical Secondary Standard, Certified Reference Material, (+/-)-(cis)-4-Amino-1-(2-hydroxymethyl-1,3-oxathiolan-5-yl)-(1H)-pyrimidin-2-one, 2(1H)-Pyrimidinone, 4-amino-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl], (+/-) (Cis), 2(1H)-Pyrimidinone,4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-, rel-, 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-[1,3]-oxathiolan-5-yl]-(1H)-pyrimidin-2-one, 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-Oxathiolan-5-yl]-(1H)-pyrimidin-2-one, cis(+/-)-4-amino-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl]-2(1H)-pyrimidinone, Lamivudine for system suitability 1, European Pharmacopoeia (EP) Reference Standard, Lamivudine for system suitability 2, European Pharmacopoeia (EP) Reference Standard, 1117764-41-6, 2(1H)-Pyrimidinone, 4-amino-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl], (-)(2R,5S) & Galanthus Nivalis Agglutinin (GNA), 2(1H)-Pyrimidinone, 4-amino-1-[2-(hydroxymethyl)-1,3-oxathiolan-5-yl], (-)(2R,5S) & Hippeastrum hybrid agglutinin( HHA), 603-844-3
Topological Polar Surface Area 113.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 15.0
Isotope Atom Count 0.0
Molecular Complexity 331.0
Database Name cmaup_ingredients;npass_chem_all;pubchem
Defined Atom Stereocenter Count 2.0
Uniprot Id n.a., Q72547, Q72874, P02545, P38532, P10636, O60840, P02768, O95342, Q92887, O15438, O15439, Q03732, P08684, P10635, P11712, P0DTD1
Iupac Name 4-amino-1-[(2R,5S)-2-(hydroxymethyl)-1,3-oxathiolan-5-yl]pyrimidin-2-one
Prediction Hob 1.0
Target Id NPT483, NPT51
Xlogp -0.9
Molecular Formula C8H11N3O3S
Prediction Swissadme 1.0
Inchi Key JTEGQNOMFQHVDC-NKWVEPMBSA-N
Fcsp3 0.5
Logs -0.795
Rotatable Bond Count 2.0
Logd -1.632
Compound Name Lamivudine
Prediction Hob Swissadme 1.0
Exact Mass 229.052
Formal Charge 0.0
Monoisotopic Mass 229.052
Hydrogen Bond Acceptor Count 4.0
Molecular Weight 229.26
Covalent Unit Count 1.0
Total Atom Stereocenter Count 2.0
Total Bond Stereocenter Count 0.0
Esol -1.8979182
Inchi InChI=1S/C8H11N3O3S/c9-5-1-2-11(8(13)10-5)6-4-15-7(3-12)14-6/h1-2,6-7,12H,3-4H2,(H2,9,10,13)/t6-,7+/m0/s1
Smiles C1[C@H](O[C@H](S1)CO)N2C=CC(=NC2=O)N
Nring 2.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Citrus Bergamia (Plant) Rel Props:Source_db:npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Sophora Flavescens (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Strychnos Vanprukii (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all