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Mitomycin

PubChem CID: 5746

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Compound Synonyms mitomycin C, Mitomycin, 50-07-7, Ametycine, Mutamycin, Mitomycin-C, Mitocin-C, Ametycin, Mytozytrex, Mitomycinum, Mytomycin, Mitomycinum C, Mitamycin, Mitozytrex, Mitosol, Muamycin, Mitomycyna C, 7-Amino-9alpha-methoxymitosane, Mito-C, NSC-26980, Mit-C, MMC, RCRA waste number U010, NCI-C04706, CCRIS 414, HSDB 3239, NSC26980, EINECS 200-008-6, Mitomycine, UNII-50SG953SK6, JELMYTO, DTXSID2020898, CHEBI:27504, AI3-26199, Mitocin C, 50SG953SK6, DTXCID00898, 6-Amino-1,1a,2,8,8a,8b-hexahydro-8-(hydroxymethyl)-8a-methoxy-5-methylazirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione carbamate (ester), Azirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione, 6-amino-8-(((aminocarbonyl)oxy)methyl)-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methyl-, (1aS-(1aalpha,8beta,8aalpha,8balpha))-, UGN-101, UGN-102, Mitomycin [USAN:USP:INN:BAN], Mitomycyna C [Polish], MFCD00078109, [(4S,6S,7R,8S)-11-amino-7-methoxy-12-methyl-10,13-dioxo-2,5-diazatetracyclo[7.4.0.0^{2,7}.0^{4,6}]trideca-1(9),11-dien-8-yl]methyl carbamate, Mitomicina, MITOMYCIN (MART.), MITOMYCIN [MART.], MITOMYCIN (USP-RS), MITOMYCIN [USP-RS], MITOMYCIN C (IARC), MITOMYCIN C [IARC], Mitomycin (TN), 1404-00-8, Azirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione, 6-amino-1,1a,2,8,8a,8b-hexahydro-8-(hydroxymethyl)-8a-methoxy-5-methyl-, carbamate (ester), Azirino[2',3':3,4]pyrrolo[1,2-a]indole-4,7-dione, 6-amino-8-[[(aminocarbonyl)oxy]methyl]-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methyl-, (1aS,8S,8aR,8bS)-, C15H18N4O5, MITOMYCIN (EP MONOGRAPH), MITOMYCIN [EP MONOGRAPH], MITOMYCIN (USP MONOGRAPH), MITOMYCIN [USP MONOGRAPH], Mitomycin (USAN:USP:INN:BAN), CAS-50-07-7, Muamycin (TN), NSC 26980, ((1aS,8S,8aR,8bS)-6-amino-8a-methoxy-5-methyl-4,7-dioxo-1,1a,2,4,7,8,8a,8b-octahydroazirino[2',3':3,4]pyrrolo[1,2-a]indol-8-yl)methyl carbamate, (1aS,8S,8aR,8bS)-6-Amino-8-[[(aminocarbonyl)oxy]methyl]-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methylazirino[2',3':3,4]pyrrolo[1,2-a]indole-4,7-dione, [(1aS,8S,8aR,8bS)-6-amino-8a-methoxy-5-methyl-4,7-dioxo-1,1a,2,4,7,8,8a,8b-octahydroazireno[2',3':3,4]pyrrolo[1,2-a]indol-8-yl]methyl carbamate, [(4S,6S,7R,8S)-11-amino-7-methoxy-12-methyl-10,13-dioxo-2,5-diazatetracyclo[7.4.0.02,7.04,6]trideca-1(9),11-dien-8-yl]methyl carbamate, [1aS-(1aalpha,8beta,8aalpha,8balpha)]-6-Amino-8-[[(aminocarbonyl)oxy]methyl]-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methylazirino[2',3':3,4]pyrrolo[1,2-a]indole-4,7-dione, Azirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione, 6-amino-8-(((aminocarbonyl)oxy)methyl)-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methyl-, (1aS,8S,8aR,8bS)-, Mitomycin (USP/INN), MLS002702984, (amino-methoxy-methyl-dioxo-[?]yl)methyl carbamate, RCRA waste no. U010, 7-Amino-9.alpha.-methoxymitosane, Mutamycine, Mitocin, Mitolem, Mitomycine C, Mito-Medac, Mitomycin-X, NCGC00095258-01, ((1aS,8S,8aR,8bS)-6-amino-8a-methoxy-5-methyl-4,7-dioxo-1,1a,2,4,7,8,8a,8b-octahydroazirino(2',3':3,4)pyrrolo(1,2-a)indol-8-yl)methyl carbamate, (1as,8s,8ar,8bs)-6-amino-8-(((aminocarbonyl)oxy)methyl)-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methylazirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione, [(1aS,8S,8aR,8bS)-6-amino-8a-methoxy-5-methyl-4,7-dioxo-1,1a,2,4,7,8,8a,8b-octahydroazirino[2',3':3,4]pyrrolo[1,2-a]indol-8-yl]methyl carbamate, Mitomycin, [(1aS,8S,8aR,8bS)-6-Amino-8a-methoxy-5-methyl-4,7-dioxo-1,1a,2,4,7,8,8a,8b-octahydroazirino[2'',3'':3,4]pyrrolo[1,2-a]indol-8-yl]methyl carbamate, Mitomycin C, Jelmyto (TN), MITO, Mitomycin C from Streptomyces caespitosus, MITOMYCIN [INN], Mitomycin C (JP18), MITOMYCIN [HSDB], MITOMYCIN [USAN], MITOMYCIN [VANDF], MITOMYCIN C [MI], CHEMBL105, MITOMYCIN C [JAN], MITOMYCIN [WHO-DD], Mitomycin C - High Purity, SCHEMBL3760, CBiol_001927, BSPBio_001267, KBioGR_000607, KBioSS_000607, Mitomycin C (4% in NaCl), MLS001332654, Mitozytrex (TN) (Supergene), 50-07-7 (non-salt), AMETYCIN pound notmitomycin C, GTPL7089, MITOMYCIN [ORANGE BOOK], KBio2_000607, KBio2_003175, KBio2_005743, KBio3_001073, KBio3_001074, DTXSID00858942, EX-A501, L01DC03, Mitomycin C - Bio-X trade mark, BCPP000410, Bio1_000213, Bio1_000702, Bio1_001191, Bio2_000464, Bio2_000944, HMS1362O09, HMS1792O09, HMS1990O09, HMS2089F16, HMS3403O09, Mutamycin(mitomycin for injection), AZIRINO(2',3':3,4)PYRROLO(1,2-A)INDOLE-4,7-DIONE, 6-AMINO-8-(((AMINOCARBONYL)OXY)METHYL)-1,1A,2,8,8A,8B-HEXAHYDRO-8A-METHOXY-5-METHYL-, (1AS-(1A.ALPHA.,8.BETA.,8A.ALPHA.,8B.ALPHA.))-, Tox21_111493, AC-918, BDBM50428658, GR-311, HB4458, s8146, AKOS015895703, Tox21_111493_1, AM26019, BCP9000285, CCG-208564, CS-0564, DB00305, KS-5148, 7-AMINO-9-ALPHA-METHOXYMITOSANE, IDI1_002219, SMP1_000307, Mitomycin 100 microg/mL in Acetonitrile, NCGC00163468-02, NCGC00163468-03, NCGC00163468-05, NCGC00163468-06, AM161650, BM164668, HY-13316, SMR000058401, BCP0726000181, M2320, NS00004729, C06681, D00208, D91590, AB00918689-03, AB00918689-04, EN300-7405455, BRD-K59670716-001-02-6, BRD-K59670716-001-06-7, Q19856779, WLN: T D3 B556 BN EM JV MVTTT&J GO1 H1OVZ KZ L1, Mitomycin C from Streptomyces caespitosus, >=970 mug/mg (USP XXIV), Mitomycin C from Streptomyces caespitosus, powder, BioReagent, suitable for cell culture, Mitomycin C from Streptomyces caespitosus, powder, contains NaCl as solubilizer, (1AR)-6-AMINO-8-(((AMINOCARBONYL)OXY)METHYL)-1,1A,2,8,8A,8B-HEXAHYDRO-8A-METHOXY-5-METHYLAZIRINO(2',3':3,4)PYRROLO(1,2-A)INDOLE-4,7-DIONE, (1aS,8S,8aR,8bS)-6-Amino-4,7-dioxo-8a-methoxy-5-methyl-1,1a,2,8,8a,8b-hexahydroazirino(2',3':3,4)pyrrolo(1,2-a)indol-8-ylmethyl carbamate, (1aS-(1a alpha,8beta,8a alpha,8b alpha))-6-amino-8-(((aminocarbonyl)oxy)methyl)-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methylazirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione, 1aS-(1a-a,8b,8a-a,8b-a)-6-Amino-8-(aminocarbonyl)oxymethyl-1,1a,2,8,8a,8b-hexahydro-8a-methoxy-5-methylazirino2,'3':3,4pyrrol o1,2-a indole-4,7-dione, MMC, Ametycine, 200-008-6, 6-AMINO-1,1A,2,8,8A,8B-HEXAHYDRO-8-(HYDROXYMETHYL)-8A-METHOXY-5-METHYLAZIRINO-(2',3':3,4)PYRROLO(1,2-A)INDOLE-4,7-DIONE, CARBAMATE (ESTER), AZIRINO(2',3':3,4)PYRROLO(1,2-A)INDOLE-4,7-DIONE, 6-AMINO-8-(((AMINOCARBONYL)OXY)METHYL)-1,1A,2,8,8A,8B-HEXAHYDRO-8A-METHOXY-5-METHYL-, (1AS-(1AALPHA,8BETA,8AALPHA,8B.ALPHA)).-, AZIRINO(2',3':3,4)PYRROLO(1,2-A)INDOLE-4,7-DIONE, 6-AMINO-8-(((AMINOCARBONYL)OXY)METHYL)-1,1A,2,8,8A,8B-HEXAHYDRO-8A-METHOXY-5-METHYL-,(1AR-(1AALPHA,8BETA,8AALPHA,8BALPHA))-, Azirino(2',3':3,4)pyrrolo(1,2-a)indole-4,7-dione,6-amino-8-(((aminocarbonyl)oxy) methyl)-1,1a,2,8,8a,8b-hexahydro-8-a-methoxy-5-methyl-, (1aS-(1aalpha,8beta, 8aalpha,8balpha))-, Azirino[2',4]pyrrolo[1,2-a]indole-4,7-dione, 6-amino-1,1a,2,8,8a,8b-hexahydro-8-(hydroxymethyl)-8a- methoxy-5-methyl-, carbamate (ester), Azirino[2',4]pyrrolo[1,2-a]indole-4,7-dione, 6-amino-8-[[(aminocarbonyl)oxy]methyl]-1,1a,2,8,8a,8b- hexahydro-8a-methoxy-5-methyl-, [1aR-(1a.alpha.,8.beta.,8a.alpha.,8b.alpha.)]-, Mitomycin C from Streptomyces caespitosus, >=98% (HPLC), potency: >=970 mug per mg (USP XXIV), gamma-irradiated, suitable for cell culture
Topological Polar Surface Area 147.0
Hydrogen Bond Donor Count 3.0
Heavy Atom Count 24.0
Isotope Atom Count 0.0
Molecular Complexity 757.0
Database Name cmaup_ingredients;hmdb_chem_all;npass_chem_all;pubchem
Defined Atom Stereocenter Count 4.0
Uniprot Id P16435, P08183, n.a., P00375, Q16236, Q9UNA4, O75496, O42275, P81908, P14902, Q9NUW8, P27695, P0DTD1, P10275, Q03181
Iupac Name [(4S,6S,7R,8S)-11-amino-7-methoxy-12-methyl-10,13-dioxo-2,5-diazatetracyclo[7.4.0.02,7.04,6]trideca-1(9),11-dien-8-yl]methyl carbamate
Prediction Hob 1.0
Class Indoles and derivatives
Target Id NPT1078
Xlogp -0.4
Superclass Organoheterocyclic compounds
Subclass Indolequinones
Molecular Formula C15H18N4O5
Prediction Swissadme 0.0
Inchi Key NWIBSHFKIJFRCO-WUDYKRTCSA-N
Fcsp3 0.5333333333333333
Logs -2.288
Rotatable Bond Count 4.0
State Solid
Logd 0.624
Synonyms 7-Amino-9alpha-methoxymitosane, Ametycine, Mitocin-C, MMC, Mutamycin, Mitomycin C, Muamycin, 7-Amino-9a-methoxymitosane, 7-Amino-9α-methoxymitosane, Mitamycin, Mitocin C, Mitomycin-C, MitocinC, Mitomycin
Compound Name Mitomycin
Kingdom Organic compounds
Prediction Hob Swissadme 0.0
Exact Mass 334.128
Formal Charge 0.0
Monoisotopic Mass 334.128
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 334.33
Covalent Unit Count 1.0
Total Atom Stereocenter Count 4.0
Total Bond Stereocenter Count 0.0
Molecular Framework Aliphatic heteropolycyclic compounds
Esol -1.8630584000000001
Inchi InChI=1S/C15H18N4O5/c1-5-9(16)12(21)8-6(4-24-14(17)22)15(23-2)13-7(18-13)3-19(15)10(8)11(5)20/h6-7,13,18H,3-4,16H2,1-2H3,(H2,17,22)/t6-,7+,13+,15-/m1/s1
Smiles CC1=C(C(=O)C2=C(C1=O)N3C[C@H]4[C@@H]([C@@]3([C@@H]2COC(=O)N)OC)N4)N
Nring 4.0
Defined Bond Stereocenter Count 0.0
Taxonomy Direct Parent Mitomycins

  • 1. Outgoing r'ship FOUND_IN to/from Cedrus Deodara (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Eupatorium Chinense (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Inula Racemosa (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 4. Outgoing r'ship FOUND_IN to/from Scoparia Dulcis (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all