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Mifepristone

PubChem CID: 55245

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Compound Synonyms mifepristone, 84371-65-3, RU-486, Mifegyne, Mifeprex, Korlym, RU 486, RU486, Mifepristona, Mifepriston, Corlux, RU 38486, RU-38486, Mifepristonum, Mifepristonum [Latin], C29H35NO2, HSDB 6841, (11beta,17beta)-11-[4-(Dimethylamino)phenyl]-17-hydroxy-17-(1-propyn-1-yl)estra-4,9-dien-3-one, UNII-320T6RNW1F, BRN 5779404, 320T6RNW1F, CCRIS 9332, DTXSID5023322, RU 486-6, CHEBI:50692, Mifepristone (Standard), NSC-759862, MLS000069785, DTXCID303322, VGX-410C, VGX-410, 11beta-(4-(Dimethylamino)phenyl)-17-hydroxy-21-methyl-19-nor-17alpha-pregna-4,9-dien-20-m-3-on, 11beta-(4-(Dimethylamino)phenyl)-17beta-hydroxy-17-(1-propynyl)estra-4,9-dien-3-on, 11beta-(4-(N,N-Dimethylamino)phenyl)-17alpha-(prop-1-ynyl)-delta4,9-estradiene-17beta-ol-3-one, 17-beta-Hydroxy-11-beta-(4-dimethylaminophenyl-1)-17-alpha-(prop-1-ynyl)oestra-4,9-dien-3-one, NSC 759862, Mifepristonum (Latin), NCGC00025179-05, SMR000058481, Mifepristona [Spanish], 11beta-(p-(Dimethylamino)phenyl)-17beta-hydroxy-17-(1-propynyl)estra-4,9-dien-3-one, MIFEPRISTONE (MART.), MIFEPRISTONE [MART.], (11beta,17beta)-11-(4-(Dimethylamino)phenyl)-17-hydroxy-17-(1-propynyl)-estra-4,9-dien-3-one, (8S,11R,13S,14S,17S)-11-(4-(dimethylamino)phenyl)-17-hydroxy-13-methyl-17-(prop-1-yn-1-yl)-1,2,6,7,8,11,12,13,14,15,16,17-dodecahydro-3H-cyclopenta[a]phenanthren-3-one, (8S,11R,13S,14S,17S)-11-(4-dimethylaminophenyl)-17-hydroxy-13-methyl-17-prop-1-ynyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one, 11-(4-DIMETHYLAMINO-PHENYL)-17-HYDROXY-13-METHYL-17-PROP-1-YNYL-1,2,6,7,8,11,12,13,14,15,16,17-DODEC AHYDRO-CYCLOPENTA[A]PHENANTHREN-3-ONE, Estra-4,9-dien-3-one, 11-(4-(dimethylamino)phenyl)-17-hydroxy-17-(1-propynyl)-, (11-beta,17-beta)-, MIFEPRISTONE (USP-RS), MIFEPRISTONE [USP-RS], (10S,11S,14S,15S,17R)-17-[4-(dimethylamino)phenyl]-14-hydroxy-15-methyl-14-(prop-1-yn-1-yl)tetracyclo[8.7.0.0^{2,7}.0^{11,15}]heptadeca-1,6-dien-5-one, (11beta,17beta)-11-[4-(dimethylamino)phenyl]-17-hydroxy-17-prop-1-yn-1-ylestra-4,9-dien-3-one, RU486 (tetramethyl-rhodamine conjugated), Mifepristone [USAN:INN:BAN], SR-01000076011, R 38486, Pictovir, NSC652104, 1nhz, Mifeprex (TN), Pictovir (TM), (11beta,17beta)-11-[4-(Dimethylamino)phenyl]-17-hydroxy-17-(1-propynyl)-estra-4,9-dien-3-one, 11-(4-DIMETHYLAMINO-PHENYL)-17-HYDROXY-13-METHYL-17-PROP-1-YNYL-1,2,6,7,8,11,12,13,14,15,16,17-DODEC AHYDRO-CYCLOPENTA(A)PHENANTHREN-3-ONE, Prestwick_570, CAS-84371-65-3, Korlym (TN), MFCD00867226, 2w8y, Mifepristone (Mifeprex), Opera_ID_562, Mifepristone, >=98%, Prestwick0_000299, Prestwick1_000299, Prestwick2_000299, Prestwick3_000299, Spectrum5_002045, MIFEPRISTONE [MI], MIFEPRISTONE [INN], MIFEPRISTONE [JAN], MIFEPRISTONE [HSDB], MIFEPRISTONE [USAN], MIFEPRISTONE [VANDF], BIDD:PXR0123, Lopac0_000801, SCHEMBL16087, BSPBio_000238, Estra-4,9-dien-3-one, 11-(4-(dimethylamino)phenyl)-17-hydroxy-17-(1-propynyl)-, (11beta,17beta)-, MLS001074115, MLS001424271, MIFEPRISTONE [WHO-DD], SPBio_002457, RU-486, MIFEPRISTONE, BPBio1_000262, CHEMBL438575, GTPL2805, Mifepristone (JAN/USAN/INN), CHEMBL1276308, BDBM18627, G03XB01, HMS1568L20, HMS2052L05, HMS2090L22, HMS2095L20, HMS2230P21, HMS3262B03, HMS3412D17, HMS3649J08, HMS3676D17, HMS3712L20, HMS3884D12, MIFEPRISTONE [ORANGE BOOK], BCP02145, Tox21_110952, Tox21_301841, Tox21_500801, BDBM50072024, HB2783, HSCI1_000369, HY-13683R, s2606, VX-410, AKOS015895416, Tox21_110952_1, CCG-101164, CI-1073, CS-1435, DB00834, FM26002, LP00801, NC00414, SDCCGSBI-0050778.P002, Mifepristone 1.0 mg/ml in Acetonitrile, NCGC00025179-06, NCGC00025179-07, NCGC00025179-08, NCGC00025179-09, NCGC00025179-12, NCGC00025179-13, NCGC00025179-23, NCGC00179632-01, NCGC00255152-01, NCGC00261486-01, (8S,11R,13S,14S,17S)-11-[4-(dimethylamino)phenyl]-17-hydroxy-13-methyl-17-prop-1-ynyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one, AS-13938, CPD000058481, HY-13683, RU486, C-1073, CS-0694789, EU-0100801, C-1073, C07652, D00585, EN300-117256, M 8046, Q411240, SR-01000721888, SR-01000076011-1, SR-01000076011-3, SR-01000076011-5, SR-01000076011-9, SR-01000721888-4, BRD-K37270826-001-04-5, BRD-K37270826-001-26-8, BRD-K37270826-001-27-6, BRD-K37270826-001-31-8, Z1501480424, Mifepristone, United States Pharmacopeia (USP) Reference Standard, 11-((4-dimethylamino) phenyl)-17-Hydroxy-17-(1-propynyl) Estra-4,9-dien-3-one, 11.beta.-[4-(Dimethylamino)phenyl]-17.beta.-hydroxy-17-(1-propynyl)estra-4,9-dien-3-one, 11b-(4-Dimethyl-amino)-phenyl-17b-hydroxy-17-(1-propynyl)-estra-4,9-dien-3-one, 11beta-(4-(Dimethylamino)phenyl)-17beta-hydroxy-17-(prop-1-yn-1-yl)estra-4,9-dien-3-one, 11beta-(4-Dimethyl-amino)-phenyl-17beta-hydroxy-17-(1-propynyl)-estra-4,9-dien-3-one, 11beta-(4-Dimethylamino)phenyl-17beta-hydroxy-17-(1-propynyl)estra-4,9-dien-3-one, 11ss-[p-(Dimethylamino)fenyl]-17ss-hydroxy- 17-(1-propynyl)estra-4,9-dien-3-on, (11beta,17beta)-11-(4-(Dimethylamino)-phenyl)-17-hydroxy-17-(1-propynyl)estra- 4,9-dien-3-one(O'Neil, M.J. (ed.). The Merck Index - An Encyclopedia of Chemicals, Drugs, and Biologicals. 13th Edition, Whitehouse Station, NJ: Merck and Co., Inc., 2001., p. 1103), (11R,13S,14S,17S)-11-(4-Dimethylamino-phenyl)-17-hydroxy-13-methyl-17-prop-1-ynyl-1,2,6,7,8,11,12,13,14,15,16,17-dodecahydro-cyclopenta[a]phenanthren-3-one, (1S,3aS,3bS,10R,11aS)-10-[4-(dimethylamino)phenyl]-1-hydroxy-11a-methyl-1-(prop-1-yn-1-yl)-1H,2H,3H,3aH,3bH,4H,5H,7H,8H,9H,10H,11H,11aH-cyclopenta[a]phenanthren-7-one, (aa Beta, 17 beta)-11-(4-(dimethylamino)-phenyl)-17-hydroxy-17-(1-propynyl)estra-4,9-dien-3-one, 11 Beta-(4-(N,N-dimethylamino)phenyl)-17alpha-(propyl-1-ynyl)-delta-4,9-estradiene-17 beta-ol-3-one, 11beta-(4-(dimethylamino)phenyl)-17beta-hydroxy-17alpha-(prop-1-yn-1-yl)estra-4,9-dien-3-one, 11beta-(4-(N,N-dimethylamino)phenyl)-17alpha-(prop-1-ynyl)-delta 4,9-estradiene- 17beta-ol-3-one(O'Neil, M.J. (ed.). The Merck Index - An Encyclopedia of Chemicals, Drugs, and Biologicals. 13th Edition, Whitehouse Station, NJ: Merck and Co., Inc., 2001., p. 1103), 122742-25-0, 17beta-Hydroxy-11beta-[4-(dimethylamino)-phenyl]-17alpha-(prop-1-ynyl)-estra-4,9-dien-3-one, 83203-42-3, Estra-4,9-dien-3-one, 11-[4-(dimethylamino)phenyl]-17-hydroxy-17-(1-propyn-1-yl)-, (11.beta.,17.beta.)-, Estra-4,9-dien-3-one, 11-[4-(dimethylamino)phenyl]-17-hydroxy-17-(1-propyn-1-yl)-, (11beta,17beta)-, Estra-4,9-dien-3-one, 11-[4-(dimethylamino)phenyl]-17-hydroxy-17-(1-propynyl)-, (11b,17b)-, Mifegyne(O'Neil, M.J. (ed.). The Merck Index - An Encyclopedia of Chemicals, Drugs, and Biologicals. 13th Edition, Whitehouse Station, NJ: Merck and Co., Inc., 2001., p. 1103), RU 38486(O'Neil, M.J. (ed.). The Merck Index - An Encyclopedia of Chemicals, Drugs, and Biologicals. 13th Edition, Whitehouse Station, NJ: Merck and Co., Inc., 2001., p. 1103)
Topological Polar Surface Area 40.5
Hydrogen Bond Donor Count 1.0
Heavy Atom Count 32.0
Isotope Atom Count 0.0
Molecular Complexity 921.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name (8S,11R,13S,14S,17S)-11-[4-(dimethylamino)phenyl]-17-hydroxy-13-methyl-17-prop-1-ynyl-1,2,6,7,8,11,12,14,15,16-decahydrocyclopenta[a]phenanthren-3-one
Prediction Hob 1.0
Target Id NPT542, NPT153, NPT249, NPT541, NPT108, NPT248, NPT109, NPT713, NPT628, NPT212
Xlogp 3.8
Molecular Formula C29H35NO2
Prediction Swissadme 1.0
Inchi Key VKHAHZOOUSRJNA-GCNJZUOMSA-N
Fcsp3 0.5517241379310345
Logs -5.333
Rotatable Bond Count 3.0
Logd 3.75
Compound Name Mifepristone
Prediction Hob Swissadme 1.0
Exact Mass 429.267
Formal Charge 0.0
Monoisotopic Mass 429.267
Hydrogen Bond Acceptor Count 3.0
Molecular Weight 429.6
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Esol -4.885394800000001
Inchi InChI=1S/C29H35NO2/c1-5-15-29(32)16-14-26-24-12-8-20-17-22(31)11-13-23(20)27(24)25(18-28(26,29)2)19-6-9-21(10-7-19)30(3)4/h6-7,9-10,17,24-26,32H,8,11-14,16,18H2,1-4H3/t24-,25+,26-,28-,29-/m0/s1
Smiles CC#C[C@@]1(CC[C@@H]2[C@@]1(C[C@@H](C3=C4CCC(=O)C=C4CC[C@@H]23)C5=CC=C(C=C5)N(C)C)C)O
Nring 5.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Trifolium Pratense (Plant) Rel Props:Source_db:cmaup_ingredients