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Taxchinin A

PubChem CID: 5319881

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Compound Synonyms Taxchinin A, [(2S,4R,5R,5aS,6S,8S,9aR,10S,10aS)-5,6,10-triacetyloxy-2,8-dihydroxy-10a-(2-hydroxypropan-2-yl)-3,5a-dimethyl-9-methylidene-2,4,5,6,7,8,9a,10-octahydro-1H-benzo[g]azulen-4-yl] benzoate, ((2S,4R,5R,5aS,6S,8S,9aR,10S,10aS)-5,6,10-triacetyloxy-2,8-dihydroxy-10a-(2-hydroxypropan-2-yl)-3,5a-dimethyl-9-methylidene-2,4,5,6,7,8,9a,10-octahydro-1H-benzo(g)azulen-4-yl) benzoate, CHEMBL434246, NS00093875, 146621-74-1
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 166.0
Hydrogen Bond Donor Count 3.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CC1CC2CCCC(C)C2CC2CCCC12)C1CCCCC1
Np Classifier Class Taxane diterpenoids
Deep Smiles CC=O)O[C@H]C[C@H]O)C=C)[C@@H][C@]6C)[C@@H]OC=O)C)))[C@H]OC=O)cccccc6))))))))C=CC)[C@H]C[C@]5[C@H]%10OC=O)C))))CO)C)C))))O
Heavy Atom Count 44.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level CC1CCCC2CC(OC(O)C3CCCCC3)C3CCCC3CC12
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1230.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 9.0
Uniprot Id n.a.
Iupac Name [(2S,4R,5R,5aS,6S,8S,9aR,10S,10aS)-5,6,10-triacetyloxy-2,8-dihydroxy-10a-(2-hydroxypropan-2-yl)-3,5a-dimethyl-9-methylidene-2,4,5,6,7,8,9a,10-octahydro-1H-benzo[g]azulen-4-yl] benzoate
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 1.3
Gsk 4 400 Rule False
Molecular Formula C33H42O11
Scaffold Graph Node Bond Level C=C1CCCC2CC(OC(=O)c3ccccc3)C3=CCCC3CC12
Prediction Swissadme 0.0
Inchi Key VETCXRGMQJYOHM-JGYXPHOZSA-N
Silicos It Class Moderately soluble
Fcsp3 0.5757575757575758
Logs -4.221
Rotatable Bond Count 10.0
Logd 2.082
Synonyms taxchinin a
Esol Class Soluble
Functional Groups C=C(C)C, CC(=O)OC, CC(C)=C(C)C, CO, cC(=O)OC
Compound Name Taxchinin A
Prediction Hob Swissadme 0.0
Exact Mass 614.273
Formal Charge 0.0
Monoisotopic Mass 614.273
Hydrogen Bond Acceptor Count 11.0
Molecular Weight 614.7
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Esol -3.9109746909090926
Inchi InChI=1S/C33H42O11/c1-16-22(37)14-24(41-18(3)34)32(8)26(16)28(42-19(4)35)33(31(6,7)40)15-23(38)17(2)25(33)27(29(32)43-20(5)36)44-30(39)21-12-10-9-11-13-21/h9-13,22-24,26-29,37-38,40H,1,14-15H2,2-8H3/t22-,23-,24-,26-,27+,28-,29-,32+,33-/m0/s1
Smiles CC1=C2[C@H]([C@@H]([C@@]3([C@H](C[C@@H](C(=C)[C@H]3[C@@H]([C@@]2(C[C@@H]1O)C(C)(C)O)OC(=O)C)O)OC(=O)C)C)OC(=O)C)OC(=O)C4=CC=CC=C4
Nring 4.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Diterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Equisetum Hyemale (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Taxus Baccata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Taxus Chinensis (Plant) Rel Props:Source_db:npass_chem_all
  • 4. Outgoing r'ship FOUND_IN to/from Taxus Wallichiana (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all