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19-Hydroxybaccatin III

PubChem CID: 5318151

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Compound Synonyms 19-Hydroxybaccatin III, 78432-78-7, NSC 330754, 19-hydroxy-baccatin III, [(1S,2S,3R,4S,7R,9S,10R,12R,15S)-4,12-diacetyloxy-1,9,15-trihydroxy-10-(hydroxymethyl)-14,17,17-trimethyl-11-oxo-6-oxatetracyclo[11.3.1.03,10.04,7]heptadec-13-en-2-yl] benzoate, 7,11-Methano-5H-cyclodeca(3,4)benz(1,2-b)oxet-5-one, 6,12b-bis(acetyloxy)-12-(benzoyloxy)-1,2a,3,4,4a,6,9,10,11,12,12a,12b-dodecahydro-4,9,11-trihydroxy-4a-(hydroxymethyl)-8,13,13-trimethyl-, (2aR-(2aalpha,4beta,4abeta,6beta,9alpha,11alpha,12alpha,12aalpha,12balpha))-, ((1S,2S,3R,4S,7R,9S,10R,12R,15S)-4,12-diacetyloxy-1,9,15-trihydroxy-10-(hydroxymethyl)-14,17,17-trimethyl-11-oxo-6-oxatetracyclo(11.3.1.03,10.04,7)heptadec-13-en-2-yl) benzoate, CHEMBL447792, DDA43278, AKOS040760958, FS-9037, DA-49137, NS00093868, 7,11-Methano-5H-cyclodeca[3,4]benz[1,2-b]oxet-5-one,6,12b-bis(acetyloxy)-12-(benzoyloxy)-1,2a,3,4,4a,6,9,10,11,12,12a,12b-dodecahydro-4,9,11-trihydroxy-4a-(hydroxymethyl)-8,13,13-trimethyl-,(2aR,4S,4aR,6R,9S,11S,12S,12aR,12bS)-
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 186.0
Hydrogen Bond Donor Count 4.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CC1C2CCCC(CC(C)C3CCC4CCC4C31)C2)C1CCCCC1
Np Classifier Class Taxane diterpenoids, Tetracyclic diterpenoids
Deep Smiles OC[C@@][C@@H]O)C[C@@H][C@][C@H]6[C@H]OC=O)cccccc6))))))))[C@]CC=CC)[C@H]C6)O)))[C@H]C%12=O))OC=O)C)))))C)C))O))))CO4))OC=O)C
Heavy Atom Count 43.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC1CC2CCCC(C2)C(OC(O)C2CCCCC2)C2C1CCC1OCC12
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1220.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name [(1S,2S,3R,4S,7R,9S,10R,12R,15S)-4,12-diacetyloxy-1,9,15-trihydroxy-10-(hydroxymethyl)-14,17,17-trimethyl-11-oxo-6-oxatetracyclo[11.3.1.03,10.04,7]heptadec-13-en-2-yl] benzoate
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 0.5
Gsk 4 400 Rule False
Molecular Formula C31H38O12
Scaffold Graph Node Bond Level O=C(OC1C2CCC=C(CC(=O)C3CCC4OCC4C31)C2)c1ccccc1
Prediction Swissadme 0.0
Inchi Key SYDMVWLQJZBPIU-VHLOTGQHSA-N
Silicos It Class Soluble
Fcsp3 0.6129032258064516
Logs -3.928
Rotatable Bond Count 8.0
Logd 1.417
Synonyms 19-hydroxybaccatin iii
Esol Class Soluble
Functional Groups CC(=O)OC, CC(C)=C(C)C, CC(C)=O, CO, COC, cC(=O)OC
Compound Name 19-Hydroxybaccatin III
Prediction Hob Swissadme 0.0
Exact Mass 602.236
Formal Charge 0.0
Monoisotopic Mass 602.236
Hydrogen Bond Acceptor Count 12.0
Molecular Weight 602.6
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Esol -3.485480413953491
Inchi InChI=1S/C31H38O12/c1-15-19(35)12-31(39)26(42-27(38)18-9-7-6-8-10-18)24-29(13-32,20(36)11-21-30(24,14-40-21)43-17(3)34)25(37)23(41-16(2)33)22(15)28(31,4)5/h6-10,19-21,23-24,26,32,35-36,39H,11-14H2,1-5H3/t19-,20-,21+,23+,24-,26-,29+,30-,31+/m0/s1
Smiles CC1=C2[C@H](C(=O)[C@@]3([C@H](C[C@@H]4[C@]([C@H]3[C@@H]([C@@](C2(C)C)(C[C@@H]1O)O)OC(=O)C5=CC=CC=C5)(CO4)OC(=O)C)O)CO)OC(=O)C
Nring 5.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Diterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Taxus Baccata (Plant) Rel Props:Reference:ISBN:9788171360536
  • 2. Outgoing r'ship FOUND_IN to/from Taxus Sumatrana (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Taxus Wallichiana (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all