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Lys-(Des-Arg9,Leu8)-Bradykinin

PubChem CID: 5310951

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Compound Synonyms 71800-37-8, Lys-(Des-Arg9,Leu8)-Bradykinin, (DES-ARG10,LEU9)-KALLIDIN, CHEMBL384721, (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2S)-1-[(2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoic acid, Lys-(Des-Arg9,Leu8)-Bradykinin trifluoroacetate salt, des-Arg10-Leu9-Kallidin, Lys-[Leu...8...][des-Arg...9...]Bradykinin, GTPL3826, Lys-(des-Arg9, Leu8)-Bradykinin trifluoroacetate salt, [3H]Lys-[Leu8][des-Arg9]BK, HY-P4676, [3H]-Lys-[Leu8][des-Arg9]BK, BDBM50233905, [3H]-Lys-[Leu8][des-Arg9]-bradykinin, DA-75216, FL108717, CS-0655859, [Leu8]des-Arg10-Kallidin (Lys-[Leu8]des-Arg9-Bradykinin), H-Lys-Arg-Pro-Pro-Gly-Phe-Ser-Pro-Leu-OH, H-KRPPGFSPL-OH, Lys-(des-Arg9, Leu8)-Bradykinin trifluoroacetate salt, >=95%
Topological Polar Surface Area 380.0
Hydrogen Bond Donor Count 11.0
Heavy Atom Count 71.0
Isotope Atom Count 0.0
Molecular Complexity 1880.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name (2S)-2-[[(2S)-1-[(2S)-2-[[(2S)-2-[[2-[[(2S)-1-[(2S)-1-[(2S)-2-[[(2S)-2,6-diaminohexanoyl]amino]-5-(diaminomethylideneamino)pentanoyl]pyrrolidine-2-carbonyl]pyrrolidine-2-carbonyl]amino]acetyl]amino]-3-phenylpropanoyl]amino]-3-hydroxypropanoyl]pyrrolidine-2-carbonyl]amino]-4-methylpentanoic acid
Prediction Hob 0.0
Target Id NPT6127
Xlogp -4.1
Molecular Formula C47H75N13O11
Prediction Swissadme 0.0
Inchi Key AGTPZUQKOYEAOH-MDKUUQCZSA-N
Fcsp3 0.6595744680851063
Logs -2.352
Rotatable Bond Count 27.0
Logd -1.584
Compound Name Lys-(Des-Arg9,Leu8)-Bradykinin
Prediction Hob Swissadme 0.0
Exact Mass 997.571
Formal Charge 0.0
Monoisotopic Mass 997.571
Hydrogen Bond Acceptor Count 14.0
Molecular Weight 998.2
Covalent Unit Count 1.0
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 0.0
Esol -3.3712566112676
Inchi InChI=1S/C47H75N13O11/c1-28(2)24-33(46(70)71)56-42(66)36-17-10-21-58(36)44(68)34(27-61)57-40(64)32(25-29-12-4-3-5-13-29)54-38(62)26-53-41(65)35-16-9-22-59(35)45(69)37-18-11-23-60(37)43(67)31(15-8-20-52-47(50)51)55-39(63)30(49)14-6-7-19-48/h3-5,12-13,28,30-37,61H,6-11,14-27,48-49H2,1-2H3,(H,53,65)(H,54,62)(H,55,63)(H,56,66)(H,57,64)(H,70,71)(H4,50,51,52)/t30-,31-,32-,33-,34-,35-,36-,37-/m0/s1
Smiles CC(C)C[C@@H](C(=O)O)NC(=O)[C@@H]1CCCN1C(=O)[C@H](CO)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)CNC(=O)[C@@H]3CCCN3C(=O)[C@@H]4CCCN4C(=O)[C@H](CCCN=C(N)N)NC(=O)[C@H](CCCCN)N
Nring 4.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Jasminum Sambac (Plant) Rel Props:Source_db:cmaup_ingredients