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(3H)methyllycaconitine

PubChem CID: 5288811

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Compound Synonyms Methyllycaconitine, [3H]methyllycaconitine, CHEMBL4454983, (3H)methyllycaconitine, Delartine, [(1S,2R,3R,4S,5R,6S,8R,9S,10S,13S,16S,17R,18S)-11-Ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-13-yl]methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate, 21019-30-7, [(1S,2R,3R,4S,5R,6S,8R,9S,10S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo[7.7.2.1^{2,5}.0^{1,10}.0^{3,8}.0^{13,17}]nonadecan-13-yl]methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate, Methyllycaconitin, 2byr, ((1S,2R,3R,4S,5R,6S,8R,9S,10S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo(7.7.2.1^(2,5).0^(1,10).0^(3,8).0^(13,17))nonadecan-13-yl)methyl 2-((3S)-3-methyl-2,5-dioxopyrrolidin-1-yl)benzoate, ((1S,2R,3R,4S,5R,6S,8R,9S,10S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo(7.7.2.12,5.01,10.03,8.013,17)nonadecan-13-yl)methyl 2-((3S)-3-methyl-2,5-dioxopyrrolidin-1-yl)benzoate, GTPL3980, GTPL4005, CHEBI:43931, 1356-60-1, BDBM50530219, XM183142, MLA, BRD-K43192255-048-03-6, (20-ethyl-7,8-dihydroxy-1alpha,6beta,14alpha,16beta-tetramethoxyaconitan-4-yl)methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate, [(1beta,5alpha,6alpha,8alpha,9alpha,13alpha,14beta,16alpha)-20-ethyl-7,8-dihydroxy-1,6,14,16-tetramethoxyaconitan-4-yl]methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 144.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CCC12CCCC34C(CC1)C(CC23)C1CCC2CC1C4C2)C1CCCCC1C1C(C)CCC1C
Np Classifier Class Terpenoid alkaloids
Deep Smiles CCNC[C@@]CC[C@@H][C@][C@H]8[C@]O)[C@H][C@H]95)OC)))[C@@][C@@H][C@H]6C[C@@H][C@@H]5OC)))[C@H]C7)OC)))))))O)))))OC)))))COC=O)cccccc6NC=O)C[C@@H]C5=O))C
Heavy Atom Count 49.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC(OCC12CCCC34C5CC6CCC(C5C6)C(CC13)C4NC2)C1CCCCC1N1C(O)CCC1O
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1380.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 14.0
Iupac Name [(1S,2R,3R,4S,5R,6S,8R,9S,10S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-13-yl]methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 1.0
Gsk 4 400 Rule False
Molecular Formula C37H50N2O10
Scaffold Graph Node Bond Level O=C(OCC12CCCC34C5CC6CCC(C5C6)C(CC13)C4NC2)c1ccccc1N1C(=O)CCC1=O
Inchi Key XLTANAWLDBYGFU-VTLKBQQISA-N
Silicos It Class Moderately soluble
Rotatable Bond Count 10.0
Synonyms delsemidine, methyllycaconitine
Esol Class Moderately soluble
Functional Groups CN(C)C, CO, COC, cC(=O)OC, cN1C(=O)CCC1=O
Compound Name (3H)methyllycaconitine
Exact Mass 682.347
Formal Charge 0.0
Monoisotopic Mass 682.347
Hydrogen Bond Acceptor Count 11.0
Molecular Weight 682.8
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 14.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Inchi InChI=1S/C37H50N2O10/c1-7-38-17-34(18-49-32(42)20-10-8-9-11-23(20)39-26(40)14-19(2)31(39)41)13-12-25(46-4)36-22-15-21-24(45-3)16-35(43,27(22)28(21)47-5)37(44,33(36)38)30(48-6)29(34)36/h8-11,19,21-22,24-25,27-30,33,43-44H,7,12-18H2,1-6H3/t19-,21+,22+,24-,25-,27+,28-,29+,30-,33-,34-,35+,36-,37+/m0/s1
Smiles CCN1C[C@@]2(CC[C@@H]([C@@]34[C@@H]2[C@@H]([C@@]([C@H]31)([C@]5(C[C@@H]([C@H]6C[C@@H]4[C@@H]5[C@H]6OC)OC)O)O)OC)OC)COC(=O)C7=CC=CC=C7N8C(=O)C[C@@H](C8=O)C
Np Classifier Biosynthetic Pathway Alkaloids, Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Pseudoalkaloids

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