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Homatropine

PubChem CID: 5282593

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Compound Synonyms HOMATROPINE, 87-00-3, Homatropin, Homoatropine, Mandelyltropeine, DL-HOMATROPINE, 8QS6WCL55Z, Homotropine, Mandelytropeine, CHEBI:5747, DTXSID6044014, 1aH,3aH-Tropan-3a-ol mandelate (ester) hydrobromide, Mandelic acid, 3d-tropanyl ester, Omatropina, Methylhomatropinum, [(1S,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] 2-hydroxy-2-phenylacetate, Omatropina [DCIT], 3alpha-Tropylmandelat, Tropinmandelsaeureester, NCGC00179630-03, Homatropine [INN:BAN], DL-Mandelsaeure-tropylester, UNII-8QS6WCL55Z, Tropine, mandelate (ester), s ethyl, EINECS 201-716-8, (+-)-Homatropine, BRN 0087959, HOMATROPINE [MI], Prestwick0_000062, Prestwick1_000062, Prestwick2_000062, Prestwick3_000062, (RS)-3alpha(1alphaH,5alphaH)-Tropanylmandelat, HOMATROPINE [VANDF], HOMATROPINE [MART.], SCHEMBL23969, BSPBio_000243, HOMATROPINE [WHO-DD], 5-21-01-00234 (Beilstein Handbook Reference), SPBio_002164, BPBio1_000269, MEGxp0_001876, CHEMBL1618018, SCHEMBL15275620, ACon1_000253, CHEBI:91858, DTXCID00809535, DTXSID00858826, (1R,3r,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl 2-hydroxy-2-phenylacetate, ZTVIKZXZYLEVOL-DGKWVBSXSA-N, ZTVIKZXZYLEVOL-MCOXGKPRSA-N, HY-B0547, Tox21_113104, AC-1301, DB11181, FS-6780, CAS-87-00-3, NCGC00179630-01, NCGC00179630-02, PD006610, CS-0009509, NS00010367, C07814, AB00694561_08, EN300-18536062, Q1038115, BRD-A74975734-004-02-4, BRD-A74975734-004-10-7, HOMATROPINE HYDROBROMIDE IMPURITY A [EP IMPURITY], 1-alpha-H,5-alpha-H-Tropan-3-alpha-ol, mandelate (ester), HOMATROPINE METHYLBROMIDE IMPURITY B [EP IMPURITY], (3-exo)-8-Methyl-8-azabicyclo[3.2.1]oct-3-yl hydroxy(phenyl)acetate, BENZENEACETIC ACID, .ALPHA.-HYDROXY-, 8-METHYL-8-AZABICYCLO(.2.1)OCT-3-YL ESTER, 16175-57-8
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 49.8
Hydrogen Bond Donor Count 1.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC(CC1CCCCC1)CC1CC2CCC(C2)C1
Np Classifier Class Tropane alkaloids
Deep Smiles OCcccccc6))))))C=O)OCC[C@@H]CC[C@H]C7)N5C
Heavy Atom Count 20.0
Classyfire Class Tropane alkaloids
Scaffold Graph Node Level OC(CC1CCCCC1)OC1CC2CCC(C1)N2
Isotope Atom Count 0.0
Molecular Complexity 340.0
Database Name cmaup_ingredients;imppat_phytochem;pubchem
Defined Atom Stereocenter Count 2.0
Iupac Name [(1S,5R)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl] 2-hydroxy-2-phenylacetate
Prediction Hob 1.0
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 1.9
Gsk 4 400 Rule True
Molecular Formula C16H21NO3
Scaffold Graph Node Bond Level O=C(Cc1ccccc1)OC1CC2CCC(C1)N2
Prediction Swissadme 1.0
Inchi Key ZTVIKZXZYLEVOL-DGKWVBSXSA-N
Silicos It Class Soluble
Fcsp3 0.5625
Logs -1.554
Rotatable Bond Count 4.0
Logd 0.887
Synonyms homatropine
Esol Class Soluble
Functional Groups CN(C)C, CO, COC(C)=O
Compound Name Homatropine
Prediction Hob Swissadme 1.0
Exact Mass 275.152
Formal Charge 0.0
Monoisotopic Mass 275.152
Hydrogen Bond Acceptor Count 4.0
Molecular Weight 275.34
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 3.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -2.7210575999999995
Inchi InChI=1S/C16H21NO3/c1-17-12-7-8-13(17)10-14(9-12)20-16(19)15(18)11-5-3-2-4-6-11/h2-6,12-15,18H,7-10H2,1H3/t12-,13+,14?,15?
Smiles CN1[C@@H]2CC[C@H]1CC(C2)OC(=O)C(C3=CC=CC=C3)O
Nring 3.0
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Ornithine alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Atropa Belladonna (Plant) Rel Props:Reference:ISBN:9788185042053
  • 2. Outgoing r'ship FOUND_IN to/from Linum Usitatissimum (Plant) Rel Props:Source_db:cmaup_ingredients