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Puerarin

PubChem CID: 5281807

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Compound Synonyms Puerarin, 3681-99-0, Kakonein, Puerarin 80 mm, CHEBI:8633, Daidzein 8-c-glucoside, Daidzein-8-C-glucoside, 7-hydroxy-3-(4-hydroxyphenyl)-8-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydro-2H-pyran-2-yl)-4H-chromen-4-one, NPI 031G, 7-hydroxy-3-(4-hydroxyphenyl)-8-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]chromen-4-one, PUERARIN [WHO-DD], NSC 380711, NSC-380711, 7,4'-Dihydroxy-8-C-glucosylisoflavone, BRN 0064198, Z9W8997416, 4-19-00-03200 (Beilstein Handbook Reference), 4H-1-Benzopyran-4-one, 8-beta-D-glucopyranosyl-7-hydroxy-3-(4-hydroxyphenyl)-, 8-beta-D-Glucopyranosyl-7-hydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one, Puerarin, analytical standard, 7-hydroxy-3-(4-hydroxyphenyl)-8-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-4H-chromen-4-one, 7-hydroxy-3-(4-hydroxyphenyl)-8-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl]chromen-4-one, (1S)-1,5-anhydro-1-[7-hydroxy-3-(4-hydroxyphenyl)-4-oxo-4H-1-benzopyran-8-yl]-D-glucitol, 4H-1-BENZOPYRAN-4-ONE, 8-.BETA.-D-GLUCOPYRANOSYL-7-HYDROXY-3-(4-HYDROXYPHENYL)-, AC1NQZ4N, 8-(beta-D-Glucopyranosyl)-4',7-dihydroxyisoflavone, MFCD00063399, UNII-Z9W8997416, (1S)-1,5-anhydro-1-(7-hydroxy-3-(4-hydroxyphenyl)-4-oxo-4H-1-benzopyran-8-yl)-D-glucitol, 7-hydroxy-3-(4-hydroxyphenyl)-8-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl)chromen-4-one, 7-hydroxy-3-(4-hydroxyphenyl)-8-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)tetrahydropyran-2-yl)chromen-4-one, Puerarin (Standard), PUERARIN [INCI], 7,4'-dihydroxyisoflavone-8beta-glucopyranoside, SureCN8581666, A1H6W, MLS002473178, BIDD:ER0101, CHEMBL486386, SCHEMBL8581666, GTPL12553, HKEAFJYKMMKDOR-VPRICQMDSA-, HY-N0145R, DTXSID30958020, HKEAFJYKMMKDOR-VPRICQMDSA-N, HMS2198M10, Puerarin, >=98.0% (HPLC), 7-hydroxy-3-(4-hydroxyphenyl)-8-[(3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]chromen-4-one, HY-N0145, MSK40127, BDBM50129558, AKOS007930376, AKOS015965556, CS-6158, DB12290, KS-5191, MP08125, 1ST40127, AC-20294, SMR001397270, NS00018338, 4',7-DIHYDROXY-8-C-GLUCOSYLISOFLAVONE, BRD-K89048337-001-06-9, Q63408673, Z1494829516, 8-?-D-Glucopyranosyl-7-hydroxy-3-(4-hydroxyphenyl)-4H-1-benzopyran-4-one, (1S)-1,5-Anhydro-1-[7-hydroxy-3-(4-hydroxyphenyl)-4-oxo-4H-chromen-8-yl]-D-glucitol, 4H-1-Benzopyran-4-one, 8-beta-D-glucopyranosyl-7-hydroxy-3-(4-hydroxyphenyl)-(9CI), InChI=1/C21H20O9/c22-7-14-17(26)18(27)19(28)21(30-14)15-13(24)6-5-11-16(25)12(8-29-20(11)15)9-1-3-10(23)4-2-9/h1-6,8,14,17-19,21-24,26-28H,7H2/t14-,17-,18+,19-,21+/m1/s1
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 157.0
Hydrogen Bond Donor Count 6.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1C(C2CCCCC2)CCC2C(C3CCCCC3)CCCC12
Np Classifier Class Isoflavones
Deep Smiles OC[C@H]O[C@H][C@@H][C@H][C@@H]6O))O))O))ccO)cccc6occc6=O))cccccc6))O
Heavy Atom Count 30.0
Classyfire Class Isoflavonoids
Description A polyphenol metabolite detected in biological fluids [PhenolExplorer]
Scaffold Graph Node Level OC1C(C2CCCCC2)COC2C(C3CCCCO3)CCCC12
Classyfire Subclass Isoflavonoid c-glycosides
Isotope Atom Count 0.0
Molecular Complexity 659.0
Database Name cmaup_ingredients;fooddb_chem_all;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 5.0
Uniprot Id n.a., O89049, Q99685, P00915, P00918, P22748, P43166, O43570, P0DTD1
Iupac Name 7-hydroxy-3-(4-hydroxyphenyl)-8-[(2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]chromen-4-one
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Phenylpropanoids and polyketides
Target Id NPT955, NPT949
Xlogp 0.0
Gsk 4 400 Rule False
Molecular Formula C21H20O9
Scaffold Graph Node Bond Level O=c1c(-c2ccccc2)coc2c(C3CCCCO3)cccc12
Prediction Swissadme 0.0
Inchi Key HKEAFJYKMMKDOR-VPRICQMDSA-N
Silicos It Class Soluble
Fcsp3 0.2857142857142857
Logs -3.924
Rotatable Bond Count 3.0
Logd 0.707
Synonyms puerarin
Esol Class Soluble
Functional Groups CO, COC, c=O, cO, coc
Compound Name Puerarin
Prediction Hob Swissadme 0.0
Exact Mass 416.111
Formal Charge 0.0
Monoisotopic Mass 416.111
Hydrogen Bond Acceptor Count 9.0
Molecular Weight 416.4
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -2.126835066666667
Inchi InChI=1S/C21H20O9/c22-7-14-17(26)18(27)19(28)21(30-14)15-13(24)6-5-11-16(25)12(8-29-20(11)15)9-1-3-10(23)4-2-9/h1-6,8,14,17-19,21-24,26-28H,7H2/t14-,17-,18+,19-,21+/m1/s1
Smiles C1=CC(=CC=C1C2=COC3=C(C2=O)C=CC(=C3[C@H]4[C@@H]([C@H]([C@@H]([C@H](O4)CO)O)O)O)O)O
Nring 4.0
Np Classifier Biosynthetic Pathway Shikimates and Phenylpropanoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Isoflavonoids

  • 1. Outgoing r'ship FOUND_IN to/from Astragalus Wiedemannianus (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Bertya Dimerostigma (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Bupleurum Chinense (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 4. Outgoing r'ship FOUND_IN to/from Camellia Sinensis (Plant) Rel Props:Reference:https://www.ncbi.nlm.nih.gov/pubmed/20183820
  • 5. Outgoing r'ship FOUND_IN to/from Delphinium Barbeyi (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 6. Outgoing r'ship FOUND_IN to/from Hemerocallis Fulva (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 7. Outgoing r'ship FOUND_IN to/from Pueraria Lobata (Plant) Rel Props:Source_db:npass_chem_all
  • 8. Outgoing r'ship FOUND_IN to/from Pueraria Montana (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 9. Outgoing r'ship FOUND_IN to/from Pueraria Thomsonii (Plant) Rel Props:Source_db:npass_chem_all
  • 10. Outgoing r'ship FOUND_IN to/from Pueraria Tuberosa (Plant) Rel Props:Reference:https://www.ncbi.nlm.nih.gov/pubmed/21648202
  • 11. Outgoing r'ship FOUND_IN to/from Scutellaria Baicalensis (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 12. Outgoing r'ship FOUND_IN to/from Spatholobus Suberectus (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 13. Outgoing r'ship FOUND_IN to/from Ziziphus Jujuba (Plant) Rel Props:Source_db:cmaup_ingredients