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Pyrethrosin

PubChem CID: 5281496

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Compound Synonyms Pyrethrosin, 28272-18-6, CHEBI:8661, Z13OX0769A, [(1S,3R,5R,8E,10R,11R)-3,8-dimethyl-12-methylidene-13-oxo-4,14-dioxatricyclo[9.3.0.03,5]tetradec-8-en-10-yl] acetate, CHEMBL517337, NSC22070, UNII-Z13OX0769A, NSC-22070, OXIRENO(8,9)CYCLODECA(1,2-B)FURAN-8(2H)-ONE, 6-(ACETYLOXY)-1A,3,6,6A,7,9A,10,10A-OCTAHYDRO-4,10A-DIMETHYL-7-METHYLENE-, (1AR,4E,6R,6AR,9AS,10AR)-, Oxireno[8,9]cyclodeca[1,2-b]furan-8(2H)-one, 6-(acetyloxy)-1a,3,6,6a,7,9a,10,10a-octahydro-4,10a-dimethyl-7-methylene-, (1aR,4E,6R,6aR,9aS,10aR)-, NSC 22070, C09536, AI3-31868, PYRETHROSIN [MI], SCHEMBL5188143, DTXSID701018639, Q27108132, Germacra-4,11(13)-dien-12-oic acid, 1-beta,10-epoxy-6-alpha,8-alpha-dihydroxy-, 12,8-lactone, acetate, (E)-, Germacra-4,11(13)-dien-12-oic acid, 1.beta.,10-epoxy-6.alpha.,8.alpha.-dihydroxy-, 12,8-lactone, acetate, (E)-, Germacra-4,11(13)-dien-12-oic acid, 1alpha,10alpha-epoxy-6,8beta-dihydroxy-, 12,8-lactone, acetate, Oxireno(8,9)cyclodeca(1,2-b)furan-8(2H)-one, 6-(acetyloxy)-1a,3,6,6a,7,9a,10,10a-octahydro-4,10a-dimethyl-7-methylene-, (1aR-(1aR*,4E,6R*,6aR*,9aS*,10aR*))-
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 65.099
Hydrogen Bond Donor Count 0.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC1CC2CC3CC3CCCCCC2C1C
Np Classifier Class Germacrane sesquiterpenoids
Deep Smiles CC=O)O[C@@H]/C=CC)/CC[C@@H][C@]C[C@H][C@H]%10C=C)C=O)O5))))))C)O3
Heavy Atom Count 22.0
Classyfire Class Lactones
Scaffold Graph Node Level CC1C(O)OC2CC3OC3CCCCCC21
Classyfire Subclass Gamma butyrolactones
Isotope Atom Count 0.0
Molecular Complexity 563.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name [(1S,3R,5R,8E,10R,11R)-3,8-dimethyl-12-methylidene-13-oxo-4,14-dioxatricyclo[9.3.0.03,5]tetradec-8-en-10-yl] acetate
Veber Rule True
Classyfire Superclass Organoheterocyclic compounds
Xlogp 1.8
Gsk 4 400 Rule True
Molecular Formula C17H22O5
Scaffold Graph Node Bond Level C=C1C(=O)OC2CC3OC3CCC=CCC12
Inchi Key JJMLQAVFDJXJAL-AWZCNKNJSA-N
Silicos It Class Soluble
Rotatable Bond Count 2.0
Synonyms pyrethrosin
Esol Class Soluble
Functional Groups C/C(C)=C/C, C=C1CCOC1=O, CC(=O)OC, C[C@H]1O[C@@]1(C)C
Compound Name Pyrethrosin
Exact Mass 306.147
Formal Charge 0.0
Monoisotopic Mass 306.147
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 306.4
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 1.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C17H22O5/c1-9-5-6-14-17(4,22-14)8-13-15(10(2)16(19)21-13)12(7-9)20-11(3)18/h7,12-15H,2,5-6,8H2,1,3-4H3/b9-7+/t12-,13+,14-,15+,17-/m1/s1
Smiles C/C/1=C\[C@H]([C@H]2[C@H](C[C@@]3([C@H](O3)CC1)C)OC(=O)C2=C)OC(=O)C
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 1.0
Egan Rule True
Np Classifier Superclass Sesquiterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Tanacetum Cinerariifolium (Plant) Rel Props:Reference:https://www.ncbi.nlm.nih.gov/pubmed/5045949