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[(1S,3R,13R,14S,17S,18R,19R,20R,21S,22S,23R,24R,25R)-19,22,24-triacetyloxy-20-(acetyloxymethyl)-21-benzoyloxy-25-hydroxy-3,13,14,25-tetramethyl-6,15-dioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-18-yl] 1-methyl-6-oxopyridine-3-carboxylate

PubChem CID: 44567102

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Compound Synonyms Emarginatine B, CHEMBL451257
Topological Polar Surface Area 273.0
Hydrogen Bond Donor Count 1.0
Heavy Atom Count 69.0
Isotope Atom Count 0.0
Molecular Complexity 2190.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 13.0
Iupac Name [(1S,3R,13R,14S,17S,18R,19R,20R,21S,22S,23R,24R,25R)-19,22,24-triacetyloxy-20-(acetyloxymethyl)-21-benzoyloxy-25-hydroxy-3,13,14,25-tetramethyl-6,15-dioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-18-yl] 1-methyl-6-oxopyridine-3-carboxylate
Prediction Hob 0.0
Xlogp 2.0
Molecular Formula C48H52N2O19
Prediction Swissadme 0.0
Inchi Key OIYGAGDGUHYHMX-BZOAEYFQSA-N
Fcsp3 0.5
Logs -4.027
Rotatable Bond Count 15.0
Logd 1.238
Compound Name [(1S,3R,13R,14S,17S,18R,19R,20R,21S,22S,23R,24R,25R)-19,22,24-triacetyloxy-20-(acetyloxymethyl)-21-benzoyloxy-25-hydroxy-3,13,14,25-tetramethyl-6,15-dioxo-2,5,16-trioxa-11-azapentacyclo[15.7.1.01,20.03,23.07,12]pentacosa-7(12),8,10-trien-18-yl] 1-methyl-6-oxopyridine-3-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 960.316
Formal Charge 0.0
Monoisotopic Mass 960.316
Hydrogen Bond Acceptor Count 20.0
Molecular Weight 960.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 13.0
Total Bond Stereocenter Count 0.0
Esol -7.1365652782608695
Inchi InChI=1S/C48H52N2O19/c1-23-24(2)41(56)67-38-36(66-43(58)30-17-18-32(55)50(9)20-30)40(65-28(6)54)47(22-61-25(3)51)39(68-42(57)29-14-11-10-12-15-29)35(63-26(4)52)33-37(64-27(5)53)48(47,46(38,8)60)69-45(33,7)21-62-44(59)31-16-13-19-49-34(23)31/h10-20,23-24,33,35-40,60H,21-22H2,1-9H3/t23-,24+,33-,35+,36+,37-,38+,39-,40+,45+,46-,47-,48+/m1/s1
Smiles C[C@@H]1[C@@H](C(=O)O[C@H]2[C@@H]([C@@H]([C@]3([C@@H]([C@H]([C@@H]4[C@H]([C@@]3([C@]2(C)O)O[C@]4(COC(=O)C5=C1N=CC=C5)C)OC(=O)C)OC(=O)C)OC(=O)C6=CC=CC=C6)COC(=O)C)OC(=O)C)OC(=O)C7=CN(C(=O)C=C7)C)C
Nring 7.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Maytenus Emarginata (Plant) Rel Props:Source_db:cmaup_ingredients