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Obliquine

PubChem CID: 443685

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Compound Synonyms Obliquine, CHEMBL4167757, (1S,13S,16S,18S)-12-[2-(4-hydroxyphenyl)ethyl]-18-methoxy-15-methyl-5,7-dioxa-12,15-diazapentacyclo[11.7.0.01,16.02,10.04,8]icosa-2,4(8),9,19-tetraen-14-one, 3S,4aS,11S,10bS-3,4,4a,13,11,5,6-heptahydro-5[2-(4-hydroxyphenyl)ethyl]-3-methoxy-13-methyl-[1,3-dioxolo[4,5-g]indolo[3,3a-c]]-isoquinolin-12-one, rel-(3R,4aR,6aR,13bR)-7-[2-(4-hydroxyphenyl)ethyl]-3-methoxy-5-methyl-3,4,4a,5,7,8-hexahydro[1,3]dioxolo[4,5-g]indolo[3,3a-c]isoquinolin-6(6aH)-one, (1S,13S,16S,18S)-12-(2-(4-hydroxyphenyl)ethyl)-18-methoxy-15-methyl-5,7-dioxa-12,15-diazapentacyclo(11.7.0.01,16.02,10.04,8)icosa-2,4(8),9,19-tetraen-14-one, 3S,4aS,11S,10bS-3,4,4a,13,11,5,6-heptahydro-5(2-(4-hydroxyphenyl)ethyl)-3-methoxy-13-methyl-(1,3-dioxolo(4,5-g)indolo(3,3a-c))-isoquinolin-12-one, rel-(3R,4aR,6aR,13bR)-7-(2-(4-hydroxyphenyl)ethyl)-3-methoxy-5-methyl-3,4,4a,5,7,8-hexahydro(1,3)dioxolo(4,5-g)indolo(3,3a-c)isoquinolin-6(6aH)-one, C12183, CHEBI:31929, BDBM50278119, Q27114728, (1S,13S,16S,18S)-12-[2-(4-hydroxyphenyl)ethyl]-18-methoxy-15-methyl-5,7-dioxa-12,15-diazapentacyclo[11.7.0.01,16.02,10.04,8]icosa-2(10),3,8,19-tetraen-14-one, 3,4,4a,5,6,11,13-heptahydro-5-(2-(4-hydroxyphenyl)ethyl)-3-methoxy-13-methyl-(1,3-dioxolo(4,5-g)indolo(3,3a-c)isoquinolin-12-one), 489433-06-9
Topological Polar Surface Area 71.5
Hydrogen Bond Donor Count 1.0
Heavy Atom Count 33.0
Isotope Atom Count 0.0
Molecular Complexity 783.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 4.0
Iupac Name (1S,13S,16S,18S)-12-[2-(4-hydroxyphenyl)ethyl]-18-methoxy-15-methyl-5,7-dioxa-12,15-diazapentacyclo[11.7.0.01,16.02,10.04,8]icosa-2,4(8),9,19-tetraen-14-one
Prediction Hob 1.0
Xlogp 3.1
Molecular Formula C26H28N2O5
Prediction Swissadme 1.0
Inchi Key MNZZTIOCKJEHEP-XVZHEKKHSA-N
Fcsp3 0.4230769230769231
Logs -2.556
Rotatable Bond Count 4.0
Logd 2.465
Compound Name Obliquine
Prediction Hob Swissadme 1.0
Exact Mass 448.2
Formal Charge 0.0
Monoisotopic Mass 448.2
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 448.5
Covalent Unit Count 1.0
Total Atom Stereocenter Count 4.0
Total Bond Stereocenter Count 0.0
Esol -4.54740870909091
Inchi InChI=1S/C26H28N2O5/c1-27-23-12-19(31-2)7-9-26(23)20-13-22-21(32-15-33-22)11-17(20)14-28(24(26)25(27)30)10-8-16-3-5-18(29)6-4-16/h3-7,9,11,13,19,23-24,29H,8,10,12,14-15H2,1-2H3/t19-,23+,24-,26+/m1/s1
Smiles CN1[C@H]2C[C@@H](C=C[C@@]23[C@@H](C1=O)N(CC4=CC5=C(C=C34)OCO5)CCC6=CC=C(C=C6)O)OC
Nring 6.0
Defined Bond Stereocenter Count 0.0