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Baricitinib

PubChem CID: 44205240

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Compound Synonyms Baricitinib, 1187594-09-7, olumiant, LY3009104, INCB028050, INCB 028050, INCB-028050, 2-(3-(4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-1-(ethylsulfonyl)azetidin-3-yl)acetonitrile, UNII-ISP4442I3Y, LY-3009104, ISP4442I3Y, 1-(Ethylsulfonyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]-3-azetidineacetonitrile, Baricitinib [USAN:INN], LY 3009104, 2-(3-(4-(3H-Pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl)-1-(ethylsulfonyl)azetidin-3-yl)acetonitrile, 2-[1-ETHYLSULFONYL-3-[4-(7H-PYRROLO[2,3-D]PYRIMIDIN-4-YL)PYRAZOL-1-YL]AZETIDIN-3-YL]ACETONITRILE, 3-Azetidineacetonitrile, 1-(ethylsulfonyl)-3-(4-(7H-pyrrolo(2,3-d)pyrimidin-4-yl)-1H-pyrazol-1-yl)-, CHEBI:95341, DTXSID30152228, LY3009104 (phosphate), INCB028050 (phosphate), Baricitinib [USAN], Baricitinib (LY3009104, INCB028050), baricitinibum, C16H17N7O2S, INCB 28050, Olumiant (TN), (1-(Ethylsulfonyl)-3-(4-(7H-pyrrolo(2,3-d)pyrimidin-4-yl)-1H-pyrazol-1-yl)azetidin-3-yl)acetonitrile, {1-(ethylsulfonyl)-3-[4-(7h-pyrrolo[2,3-d]pyrimidin-4-yl)-1h-pyrazol-1-yl]azetidin-3-yl}acetonitrile, 1-(ethylsulfonyl)-3-(4-(7H-pyrrolo(2,3-d)pyrimidin-4-yl)-1H-pyrazol-1-yl)-3-azetidineacetonitrile, 2-(3-(4-(3H-pyrrolo(2,3-d)pyrimidin-4-yl)-1H-pyrazol-1-yl)-1-(ethylsulfonyl)azetidin-3-yl)acetonitrile, 3JW, MFCD21608464, Baricitinib (Standard), BARICITINIB [MI], BARICITINIB [INN], BARICITINIB [JAN], JAK inhibitors: baricitinib, BARICITINIB [WHO-DD], MLS006011247, SCHEMBL871150, Baricitinib (JAN/USAN/INN), Baricitinib (LY3009104), BARICITINIB [EMA EPAR], Baricitinib (INCB028050), GTPL7792, Baricitinib - Bio-X trade mark, CHEMBL2105759, DTXCID5074719, INCB28050, BARICITINIB [ORANGE BOOK], EX-A413, L04AA37, XUZMWHLSFXCVMG-UHFFFAOYSA-N, HMS3651L17, HMS3672M15, HMS3747G21, BCP04686, BDBM50021656, HY-15315R, NSC799357, s2851, AKOS022186127, AKOS025401933, BCP9000380, CCG-268312, CS-0724, DB11817, DS-7641, FE30357, NSC-799357, PB27275, SB10845, SDCCGSBI-0654448.P001, NCGC00345839-01, NCGC00345839-14, NCGC00345839-16, AC-27404, BB184033, DA-50940, HY-15315, SMR004703006, BCP0726000031, NS00072974, SW220096-1, Baricitinib (INCB28050, LY3009104)?, D10308, EN300-24435973, Q4860707, BRD-K53581288-001-02-9, Z2724205326, (1-(Ethylsulfonyl)-3-(4-(7H-pyrrolo(2,3-d)pyrimidin-4-yl)-1H-pyrazol-1-yl)azetidin-3-yl)ethanenitrile, 2-[1-(ethanesulfonyl)-3-(4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H-pyrazol-1-yl)azetidin-3-yl]acetonitrile, INCB 028050, 1-(Ethylsulfonyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]-3-azetidineacetonitrile, LY 3009104, INCB 028050, 1-(Ethylsulfonyl)-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)-1H-pyrazol-1-yl]-3-azetidineacetonitrile, LY 3009104
Topological Polar Surface Area 129.0
Hydrogen Bond Donor Count 1.0
Heavy Atom Count 26.0
Isotope Atom Count 0.0
Molecular Complexity 678.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 0.0
Iupac Name 2-[1-ethylsulfonyl-3-[4-(7H-pyrrolo[2,3-d]pyrimidin-4-yl)pyrazol-1-yl]azetidin-3-yl]acetonitrile
Prediction Hob 1.0
Target Id NPT1689, NPT3246, NPT3276, NPT1440
Xlogp -0.5
Molecular Formula C16H17N7O2S
Prediction Swissadme 1.0
Inchi Key XUZMWHLSFXCVMG-UHFFFAOYSA-N
Fcsp3 0.375
Logs -3.2
Rotatable Bond Count 5.0
Logd 1.054
Compound Name Baricitinib
Prediction Hob Swissadme 1.0
Exact Mass 371.116
Formal Charge 0.0
Monoisotopic Mass 371.116
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 371.4
Covalent Unit Count 1.0
Total Atom Stereocenter Count 0.0
Total Bond Stereocenter Count 0.0
Esol -1.9215027384615384
Inchi InChI=1S/C16H17N7O2S/c1-2-26(24,25)22-9-16(10-22,4-5-17)23-8-12(7-21-23)14-13-3-6-18-15(13)20-11-19-14/h3,6-8,11H,2,4,9-10H2,1H3,(H,18,19,20)
Smiles CCS(=O)(=O)N1CC(C1)(CC#N)N2C=C(C=N2)C3=C4C=CNC4=NC=N3
Nring 4.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Tabebuia Avellanedae (Plant) Rel Props:Source_db:cmaup_ingredients