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Lycaconitine

PubChem CID: 441745

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Compound Synonyms Lycaconitine, CHEBI:6587, CHEMBL451640, C08696, 25867-19-0, [(1S,2R,3R,4S,5R,6S,8R,9S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-13-yl]methyl 2-(2,5-dioxopyrrolidin-1-yl)benzoate, DTXSID00948756, CHEBI:564014, FL74374, NS00094350, Q27107253, (20-Ethyl-7,8-dihydroxy-1,6,14,16-tetramethoxyaconitan-4-yl)methyl 2-(2,5-dioxopyrrolidin-1-yl)benzoate
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 144.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CCC12CCCC34C(CC1)C(CC23)C1CCC2CC1C4C2)C1CCCCC1C1C(C)CCC1C
Np Classifier Class Terpenoid alkaloids
Deep Smiles CO[C@H][C@@H][C@]CC[C@@H][C@]6C[C@@]9O)[C@@]O)C[C@@H][C@H]C[C@@H]9[C@@H]7[C@H]5OC)))))))OC))))))NC8)CC)))))OC)))))COC=O)cccccc6NC=O)CCC5=O
Heavy Atom Count 48.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC(OCC12CCCC34C5CC6CCC(C5C6)C(CC13)C4NC2)C1CCCCC1N1C(O)CCC1O
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1330.0
Database Name imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 12.0
Uniprot Id Q05941, P12390
Iupac Name [(1S,2R,3R,4S,5R,6S,8R,9S,13S,16S,17R,18S)-11-ethyl-8,9-dihydroxy-4,6,16,18-tetramethoxy-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-13-yl]methyl 2-(2,5-dioxopyrrolidin-1-yl)benzoate
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 0.4
Gsk 4 400 Rule False
Molecular Formula C36H48N2O10
Scaffold Graph Node Bond Level O=C(OCC12CCCC34C5CC6CCC(C5C6)C(CC13)C4NC2)c1ccccc1N1C(=O)CCC1=O
Inchi Key KFXVNXQXPRPLQA-CPIHIRBUSA-N
Silicos It Class Moderately soluble
Rotatable Bond Count 10.0
Synonyms lycaconitine
Esol Class Soluble
Functional Groups CN(C)C, CO, COC, cC(=O)OC, cN1C(=O)CCC1=O
Compound Name Lycaconitine
Exact Mass 668.331
Formal Charge 0.0
Monoisotopic Mass 668.331
Hydrogen Bond Acceptor Count 11.0
Molecular Weight 668.8
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 13.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Inchi InChI=1S/C36H48N2O10/c1-6-37-17-33(18-48-31(41)19-9-7-8-10-22(19)38-25(39)11-12-26(38)40)14-13-24(45-3)35-21-15-20-23(44-2)16-34(42,27(21)28(20)46-4)36(43,32(35)37)30(47-5)29(33)35/h7-10,20-21,23-24,27-30,32,42-43H,6,11-18H2,1-5H3/t20-,21-,23+,24+,27-,28+,29-,30+,32?,33+,34-,35+,36-/m1/s1
Smiles CCN1C[C@@]2(CC[C@@H]([C@@]34[C@@H]2[C@@H]([C@@](C31)([C@]5(C[C@@H]([C@H]6C[C@@H]4[C@@H]5[C@H]6OC)OC)O)O)OC)OC)COC(=O)C7=CC=CC=C7N8C(=O)CCC8=O
Np Classifier Biosynthetic Pathway Alkaloids, Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Pseudoalkaloids