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Gitoxigenin

PubChem CID: 348482

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Compound Synonyms Gitoxigenin, 545-26-6, 16beta-Hydroxydigitoxigenin, UNII-G36K2H8SME, 16beta-Hydroxydisitoxigenin, EINECS 208-886-2, G36K2H8SME, 16-beta-Hydroxydigitoxigenin, 16.beta.-Hydroxydigitoxigenin, 3-[(3S,5R,8R,9S,10S,13R,14S,16S,17R)-3,14,16-trihydroxy-10,13-dimethyl-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta[a]phenanthren-17-yl]-2H-furan-5-one, CHEBI:38105, 3beta,14,16beta-Trihydroxy-5beta-card-20(22)-enolide, GITOXIGENIN [MI], NSC 407807, NSC-407807, BRN 0096483, 16.beta.-Hydroxydisitoxigenin, 3-beta,14,16-Trioxycarden-(20:22)-olid, 3-beta,14,16-Trioxy-digen-(20:22)-olid, DTXSID20878642, 5-18-04-00385 (Beilstein Handbook Reference), CARDOGENEN-(20:22)-TRIOL-(3-beta,14,16), NSC407807, 3-beta,14,16-Trioxy-digen-(20:22)-olid [German], 3-beta,14,16-Trioxycarden-(20:22)-olid [German], Cardogenen-(20:22)-triol-(3-beta,14,16) [German], delta(20,22)-2,14,16,21-tetrahydroxynorcholenic acid lactone, Card-20(22)-enolide, 3,14,16-trihydroxy-, (3-beta,5-beta,16-beta)-, Bigitaligenin, 5beta-Card-20(22)-enolide, 3beta,14,16beta-trihydroxy-, 5-beta-CARD-20(22)-ENOLIDE, 3-beta,14,16-beta-TRIHYDROXY-, 5.beta.-Card-20(22)-enolide, 3.beta.,14,16.beta.-trihydroxy-, Card-20(22)-enolide, 3,14,16-trihydroxy-, (3beta,5beta,16beta)-, Card-20(22)-enolide, 3,14,16-trihydroxy-, (3.beta.,5.beta.,16.beta.)-, SR-05000002231, 3-((3S,5R,8R,9S,10S,13R,14S,16S,17R)-3,14,16-trihydroxy-10,13-dimethyl-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta(a)phenanthren-17-yl)-2H-furan-5-one, 3-.beta.,14,16-Trioxycarden-(20:22)-olid, 16b-Hydroxydigitoxigenin, 3-.beta.,14,16-Trioxy-digen-(20:22)-olid, Cardogenen-(20:22)-triol-(3.beta.,14,16), 3,14,16-Trihydroxycard-20(22)-enolide, (3.beta.)-, SCHEMBL644087, CHEMBL464658, MEGxp0_001900, .delta.(20,22)-2,14,16,21-(Tetrahydroxy)norcholenic acid lactone, PVAMXWLZJKTXFW-VQMOFDJESA-N, BDBM225705, CS334, DTXCID401016684, 3-beta,14,16-beta-Trihydroxy-5-beta,14-beta-card-20(22)-enolide, LMST01120003, AKOS030490030, CCG-208473, HY-W127509, NCI60_003893, CS-0185737, NS00004870, Cardogenen-(20:22)-triol-(3beta,14,16), G89193, Q1527718, SR-05000002231-2, SR-05000002231-3, 3,14,16-Trihydroxycard-20(22)-enolide, (3beta)-, 3 beta,14,16 beta-trihydroxy-5 beta-card-20(22)-enolide, 5.beta.-Card-20(22)-enolide,14,16.beta.-trihydroxy-, .delta.(20,14,16,21-(Tetrahydroxy)norcholenic acid lactone, .delta.20,14,16,21-(Tetrahydroxy)norcholenic acid lactone, 5beta-Card-20(22)-enolide, 3beta,14,16beta-trihydroxy-(8CI), delta(20,22)-2,14,16,21-(Tetrahydroxy)norcholenic acid lactone, Card-20(22)-enolide, 3,14,16-trihydroxy-, (3beta,5beta,16beta)-(9CI), Card-20(22)-enolide,14,16-trihydroxy-, (3.beta.,5.beta.,16.beta.)-, 208-886-2
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 87.0
Hydrogen Bond Donor Count 3.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCC(C2CCC3C2CCC2C4CCCCC4CCC23)C1
Np Classifier Class Cardenolides
Deep Smiles O[C@H]CC[C@][C@@H]C6)CC[C@@H][C@@H]6CC[C@][C@]6O)C[C@@H][C@@H]5C=CC=O)OC5))))))O))))C)))))))))C
Heavy Atom Count 28.0
Classyfire Class Steroids and steroid derivatives
Scaffold Graph Node Level OC1CC(C2CCC3C2CCC2C4CCCCC4CCC23)CO1
Classyfire Subclass Steroid lactones
Isotope Atom Count 0.0
Molecular Complexity 718.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 9.0
Uniprot Id n.a., P51151, Q16236, Q96QE3, P11473, P84022, P16473, O75496, Q99700, P43220, O42275, P81908, Q9NUW8, O75874
Iupac Name 3-[(3S,5R,8R,9S,10S,13R,14S,16S,17R)-3,14,16-trihydroxy-10,13-dimethyl-1,2,3,4,5,6,7,8,9,11,12,15,16,17-tetradecahydrocyclopenta[a]phenanthren-17-yl]-2H-furan-5-one
Prediction Hob 0.0
Veber Rule True
Classyfire Superclass Lipids and lipid-like molecules
Target Id NPT537
Xlogp 1.6
Gsk 4 400 Rule True
Molecular Formula C23H34O5
Scaffold Graph Node Bond Level O=C1C=C(C2CCC3C2CCC2C4CCCCC4CCC23)CO1
Prediction Swissadme 1.0
Inchi Key PVAMXWLZJKTXFW-VQMOFDJESA-N
Silicos It Class Soluble
Fcsp3 0.8695652173913043
Logs -3.838
Rotatable Bond Count 1.0
Logd 3.169
Synonyms gitoxigenin
Esol Class Soluble
Functional Groups CC1=CC(=O)OC1, CO
Compound Name Gitoxigenin
Prediction Hob Swissadme 0.0
Exact Mass 390.241
Formal Charge 0.0
Monoisotopic Mass 390.241
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 390.5
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -3.203224000000001
Inchi InChI=1S/C23H34O5/c1-21-7-5-15(24)10-14(21)3-4-17-16(21)6-8-22(2)20(13-9-19(26)28-12-13)18(25)11-23(17,22)27/h9,14-18,20,24-25,27H,3-8,10-12H2,1-2H3/t14-,15+,16+,17-,18+,20+,21+,22-,23+/m1/s1
Smiles C[C@]12CC[C@@H](C[C@H]1CC[C@@H]3[C@@H]2CC[C@]4([C@@]3(C[C@@H]([C@@H]4C5=CC(=O)OC5)O)O)C)O
Nring 5.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Steroids

  • 1. Outgoing r'ship FOUND_IN to/from Aconitum Brevicalcaratum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Ammodendron Conollyi (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 3. Outgoing r'ship FOUND_IN to/from Angelica Archangelica (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 4. Outgoing r'ship FOUND_IN to/from Cirsium Dipsacolepis (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 5. Outgoing r'ship FOUND_IN to/from Cocculus Diversifolius (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 6. Outgoing r'ship FOUND_IN to/from Crinum Kirkii (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 7. Outgoing r'ship FOUND_IN to/from Croton Rhamnifolius (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 8. Outgoing r'ship FOUND_IN to/from Cryptostegia Grandiflora (Plant) Rel Props:Reference:ISBN:9788172360481
  • 9. Outgoing r'ship FOUND_IN to/from Cryptotaenia Japonica (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 10. Outgoing r'ship FOUND_IN to/from Cytisus Scoparius (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 11. Outgoing r'ship FOUND_IN to/from Digitalis Lanata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 12. Outgoing r'ship FOUND_IN to/from Digitalis Purpurea (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 13. Outgoing r'ship FOUND_IN to/from Eria Subsessilis (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 14. Outgoing r'ship FOUND_IN to/from Hypericum Triquetrifolium (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 15. Outgoing r'ship FOUND_IN to/from Hyssopus Officinalis (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 16. Outgoing r'ship FOUND_IN to/from Isodon Japonicus (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 17. Outgoing r'ship FOUND_IN to/from Knightia Deplanchei (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 18. Outgoing r'ship FOUND_IN to/from Lonicera Periclymenum (Plant) Rel Props:Source_db:npass_chem_all
  • 19. Outgoing r'ship FOUND_IN to/from Malva Sylvestris (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 20. Outgoing r'ship FOUND_IN to/from Mesembryanthemum Anatomicum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 21. Outgoing r'ship FOUND_IN to/from Myrica Multiflora (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 22. Outgoing r'ship FOUND_IN to/from Nerium Oleander (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 23. Outgoing r'ship FOUND_IN to/from Plantago Lanceolata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 24. Outgoing r'ship FOUND_IN to/from Ptilidium Ciliare (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 25. Outgoing r'ship FOUND_IN to/from Rhododendron Farrerae (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 26. Outgoing r'ship FOUND_IN to/from Scutellaria Seleriana (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 27. Outgoing r'ship FOUND_IN to/from Solanum Racemigerum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 28. Outgoing r'ship FOUND_IN to/from Teucrium Pestalozzae (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 29. Outgoing r'ship FOUND_IN to/from Toxicodendron Succedaneum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 30. Outgoing r'ship FOUND_IN to/from Trifolium Apertum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 31. Outgoing r'ship FOUND_IN to/from Tripodanthus Acutifolius (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 32. Outgoing r'ship FOUND_IN to/from Veronica Pectinata (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 33. Outgoing r'ship FOUND_IN to/from Viguiera Annua (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all