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12-Deoxyphorbol-13-isobutyrate-20-acetate

PubChem CID: 3035003

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Compound Synonyms 12-Deoxyphorbol-13-isobutyrate-20-acetate, 25090-71-5, 12-Deoxy-phorbol-13-isobutyrate-20-acetate, 12-Deoxy-phorbol, 20-acetate-13-isobutyrate, 12-Deoxyphorbol-13-(2-methylpropionate)-20-acetate, [(1R,2S,6R,10S,11R,13S,15R)-8-(acetyloxymethyl)-1,6-dihydroxy-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] 2-methylpropanoate, 12-DEOXYPHORBOL 13-ISOBUTYRATE 20-ACETATE, 5H-Cyclopropa(3,4)benz(1,2-e)azulen-5-one, 1,1a-alpha,1b-beta,4,4a,7a-alpha,7b,8,9,9a-decahydro-3-(acetoxymethyl)-1,1,6,8-alpha-tetramethyl-4a-beta,7b-alpha,9a-alpha-trihydroxy-, 9a-isobutyrate, Propanoic acid, 2-methyl-, 3-((acetyloxy)methyl)-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-4a,7b-dihydroxy-1,1,6,8-tetramethyl-5-oxo-9aH-cyclopropa(3,4)benz(1,2-e)azulen-9a-yl ester, (1aR-(1aalpha,1bbeta,4abeta,7aalpha,7balpha,8alpha,9aalpha))-, ((1R,2S,6R,10S,11R,13S,15R)-8-(acetyloxymethyl)-1,6-dihydroxy-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo(8.5.0.02,6.011,13)pentadeca-3,8-dienyl) 2-methylpropanoate, CHEMBL486418, DTXSID10947952, Propanoic acid,2-methyl-,(1aR,1bS,4aR,7aS,7bR,8R,9aS)-3-[(acetyloxy)methyl]-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-4a,7b-dihydroxy-1,1,6,8-tetramethyl-5-oxo-9aH-cyclopropa[3,4]benz[1,2-e]azulen-9a-ylester, 3-[(Acetyloxy)methyl]-4a,7b-dihydroxy-1,1,6,8-tetramethyl-5-oxo-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-9aH-cyclopropa[3,4]benzo[1,2-e]azulen-9a-yl 2-methylpropanoate
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 110.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CCC2C1CCCC1C3CC3CCC21
Np Classifier Class Tetracyclic diterpenoids, Tigliane diterpenoids
Deep Smiles CC=O)OCC=C[C@H][C@H][C@@]C3C)C))OC=O)CC)C))))C[C@H][C@@]6[C@H][C@@]C%11)O)C=O)C=C5)C)))))O))C
Heavy Atom Count 33.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC1CCC2C1CCCC1C3CC3CCC21
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 975.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 7.0
Iupac Name [(1R,2S,6R,10S,11R,13S,15R)-8-(acetyloxymethyl)-1,6-dihydroxy-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] 2-methylpropanoate
Prediction Hob 0.0
Veber Rule True
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 2.3
Gsk 4 400 Rule False
Molecular Formula C26H36O7
Scaffold Graph Node Bond Level O=C1C=CC2C1CC=CC1C3CC3CCC21
Prediction Swissadme 1.0
Inchi Key MTXOHECJOIIIJM-PHFLZNSYSA-N
Silicos It Class Soluble
Fcsp3 0.7307692307692307
Logs -4.355
Rotatable Bond Count 6.0
Logd 2.607
Synonyms 12-deoxyphorbol-13-isobutyrate-20-acetate
Esol Class Soluble
Functional Groups CC(=O)OC, CC(C)=CC, CC1=CCCC1=O, CO, COC(C)=O
Compound Name 12-Deoxyphorbol-13-isobutyrate-20-acetate
Prediction Hob Swissadme 0.0
Exact Mass 460.246
Formal Charge 0.0
Monoisotopic Mass 460.246
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 460.6
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 7.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -3.7611154000000013
Inchi InChI=1S/C26H36O7/c1-13(2)22(29)33-25-10-15(4)26(31)18(20(25)23(25,6)7)9-17(12-32-16(5)27)11-24(30)19(26)8-14(3)21(24)28/h8-9,13,15,18-20,30-31H,10-12H2,1-7H3/t15-,18+,19-,20-,24-,25+,26-/m1/s1
Smiles C[C@@H]1C[C@@]2([C@@H](C2(C)C)[C@H]3[C@]1([C@@H]4C=C(C(=O)[C@]4(CC(=C3)COC(=O)C)O)C)O)OC(=O)C(C)C
Nring 4.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Diterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Euphorbia Tirucalli (Plant) Rel Props:Reference:ISBN:9788185042114
  • 2. Outgoing r'ship FOUND_IN to/from Uncaria Canescens (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all