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Deacetylvindoline

PubChem CID: 260534

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Compound Synonyms Deacetylvindoline, Desacetyl Vindoline, 3633-92-9, 4-Desacetylvindoline, 24ETH7DXT4, NSC-91993, UNII-24ETH7DXT4, Vindoline, deacetyl-, 17-O-Deacetylvindoline, methyl (1R,9R,10S,11R,12R,19R)-12-ethyl-10,11-dihydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2(7),3,5,13-tetraene-10-carboxylate, Desacetylvindoline, Aspidospermidine-3-carboxylic acid, 6,7-didehydro-3,4-dihydroxy-16-methoxy-1-methyl-, methyl ester, (2beta,3beta,4beta,5alpha,12beta,19alpha)-, Aspidospermidine-3-carboxylic acid, 6,7-didehydro-3,4-dihydroxy-16-methoxy-1-methyl-, methyl ester, (2beta,3beta,4beta,5alpha,12R,19alpha)-, deacetyl vindoline, (2ss,3ss,4ss,5a,12R,19a)-6,7-Didehydro-3,4-dihydroxy-16-methoxy-1-methyl-aspidospermidine-3-carboxylic Acid Methyl Ester, 4-Desacetylvindoline, Deacetylvindoline, NSC 91993, , CHEMBL4081511, SCHEMBL26693259, CHEBI:18362, ZDKMPOJNYNVYLA-PEGGBQQISA-N, DTXSID401032208, methyl 3beta,4beta-dihydroxy-16-methoxy-1-methyl-6,7-didehydro-2beta,5alpha,12beta,19alpha-aspidospermidine-3alpha-carboxylate, NSC91993, NSC814276, NSC-814276, NS00094419, C01091, Q19903931, ASPIDOSPERMIDINE-3-CARBOXYLIC ACID, 6,7-DIDEHYDRO-3,4-DIHYDROXY-16-METHOXY-1-METHYL-, METHYL ESTER, (2.BETA.,3.BETA.,4.BETA.,5.ALPHA.,12.BETA.,19.ALPHA.)-, ASPIDOSPERMIDINE-3-CARBOXYLIC ACID, 6,7-DIDEHYDRO-3,4-DIHYDROXY-16-METHOXY-1-METHYL-, METHYL ESTER, (2.BETA.,3.BETA.,4.BETA.,5.ALPHA.,12R,19.ALPHA.)-, methyl (2beta,3beta,4beta,5alpha,12beta,19alpha)-3,4-dihydroxy-16-methoxy-1-methyl-6,7-didehydroaspidospermidine-3-carboxylate
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 82.5
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule True
Scaffold Graph Level C1CCC2C(C1)CC1CCC3CCCC4CCC12C34
Np Classifier Class Aspidosperma type, Aspidosperma-Iboga hybrid type (Vinca alkaloids)
Deep Smiles COcccccc6)NC)[C@@H][C@]5CCN[C@H]5[C@@][C@H][C@]9O)C=O)OC))))O))CC))C=CC6
Heavy Atom Count 30.0
Classyfire Class Plumeran-type alkaloids
Scaffold Graph Node Level C1CCC2C(C1)NC1CCC3CCCN4CCC12C34
Isotope Atom Count 0.0
Molecular Complexity 760.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 6.0
Iupac Name methyl (1R,9R,10S,11R,12R,19R)-12-ethyl-10,11-dihydroxy-5-methoxy-8-methyl-8,16-diazapentacyclo[10.6.1.01,9.02,7.016,19]nonadeca-2(7),3,5,13-tetraene-10-carboxylate
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 2.3
Gsk 4 400 Rule False
Molecular Formula C23H30N2O5
Scaffold Graph Node Bond Level C1=CC2CCC3Nc4ccccc4C34CCN(C1)C24
Inchi Key ZDKMPOJNYNVYLA-PEGGBQQISA-N
Silicos It Class Soluble
Rotatable Bond Count 4.0
Synonyms deacetylvindoline, desacetylvindoline
Esol Class Soluble
Functional Groups CC=CC, CN(C)C, CO, COC(C)=O, cN(C)C, cOC
Compound Name Deacetylvindoline
Exact Mass 414.215
Formal Charge 0.0
Monoisotopic Mass 414.215
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 414.5
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 6.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C23H30N2O5/c1-5-21-9-6-11-25-12-10-22(17(21)25)15-8-7-14(29-3)13-16(15)24(2)18(22)23(28,19(21)26)20(27)30-4/h6-9,13,17-19,26,28H,5,10-12H2,1-4H3/t17-,18+,19+,21+,22+,23-/m0/s1
Smiles CC[C@@]12C=CCN3[C@@H]1[C@]4(CC3)[C@H]([C@]([C@@H]2O)(C(=O)OC)O)N(C5=C4C=CC(=C5)OC)C
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Tryptophan alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Catharanthus Roseus (Plant) Rel Props:Reference:https://doi.org/10.1093/database/bav075