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Calpurnine

PubChem CID: 165547

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Compound Synonyms Calpurnine, 6874-80-2, Oroboidine, 13-hydroxy-lupanine-2-pyrrole-carbonic acid, Hoe 933, [(1S,2S,4S,9S,10R)-14-oxo-7,15-diazatetracyclo[7.7.1.02,7.010,15]heptadecan-4-yl] 1H-pyrrole-2-carboxylate, 13-hydroxylupanine-2-pyrrolecarbonic Acid, HOE-933, 13-Hydroxylupanine-2-pyrrolecarboxylic acid ester, (2S-(2alpha,7beta,7abeta,14beta,14aalpha))-1H-Pyrrole-2-carboxylic acid, dodecahydro-11-oxo-7,14-methano-2H,6H-dipyrido(1,2-a:1',2'-e)(1,5)diazocin-2-yl ester, 1H-Pyrrole-2-carboxylic acid, dodecahydro-11-oxo-7,14-methano-2H,6H-dipyrido(1,2-alpha:1',2'-e)(1,5)diazocin-2-yl ester, (2S-(2-alpha,7-beta,7a-beta,14-beta,14a-alpha))-, InChI=1/C20H27N3O3/c24-19-5-1-4-17-13-9-14(12-23(17)19)18-10-15(6-8-22(18)11-13)26-20(25)16-3-2-7-21-16/h2-3,7,13-15,17-18,21H,1,4-6,8-12H2/t13?,14?,15-,17-,18-/m0/s
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 65.6
Hydrogen Bond Donor Count 1.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC(CC1CCC2CC3CC(CC4C(C)CCCC34)C2C1)C1CCCC1
Np Classifier Class Quinolizidine alkaloids
Deep Smiles O=CCCC[C@H]N6C[C@@H]C[C@H]6CN[C@H]6C[C@H]CC6))OC=O)cccc[nH]5
Heavy Atom Count 26.0
Classyfire Class Lupin alkaloids
Scaffold Graph Node Level OC(OC1CCN2CC3CC(CN4C(O)CCCC34)C2C1)C1CCCN1
Classyfire Subclass Sparteine, lupanine, and related alkaloids
Isotope Atom Count 0.0
Molecular Complexity 583.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name [(1S,2S,4S,9S,10R)-14-oxo-7,15-diazatetracyclo[7.7.1.02,7.010,15]heptadecan-4-yl] 1H-pyrrole-2-carboxylate
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 2.0
Gsk 4 400 Rule True
Molecular Formula C20H27N3O3
Scaffold Graph Node Bond Level O=C(OC1CCN2CC3CC(CN4C(=O)CCCC34)C2C1)c1ccc[nH]1
Inchi Key YFRYJFMFQOBOSY-YDRHNJASSA-N
Silicos It Class Soluble
Rotatable Bond Count 3.0
Synonyms calpurnine, oroboidine
Esol Class Soluble
Functional Groups CC(=O)N(C)C, CN(C)C, cC(=O)OC, c[nH]c
Compound Name Calpurnine
Exact Mass 357.205
Formal Charge 0.0
Monoisotopic Mass 357.205
Hydrogen Bond Acceptor Count 4.0
Molecular Weight 357.4
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C20H27N3O3/c24-19-5-1-4-17-13-9-14(12-23(17)19)18-10-15(6-8-22(18)11-13)26-20(25)16-3-2-7-21-16/h2-3,7,13-15,17-18,21H,1,4-6,8-12H2/t13-,14-,15-,17+,18-/m0/s1
Smiles C1C[C@@H]2[C@H]3C[C@@H](CN2C(=O)C1)[C@@H]4C[C@H](CCN4C3)OC(=O)C5=CC=CN5
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Lysine alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Calpurnia Aurea (Plant) Rel Props:Reference:ISBN:9788172360481