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Aristololactam-glucoside

PubChem CID: 159819

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Compound Synonyms Aristololactam-glucoside, Aristolactam-N-beta-D-glycoside, 17413-41-1, CCRIS 2997, 6-glucopyranosyl-8-methoxybenzo(f)-1,3-benzodioxolo(6,5,4-cd)indol-5(6H)one, Benzo(f)-1,3-benzodioxolo(6,5,4-cd)indol-5(6H)-one, 6-beta-D-glucopyranosyl-8-methoxy-, 14-methoxy-10-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,5-dioxa-10-azapentacyclo[9.7.1.02,6.08,19.013,18]nonadeca-1(18),2(6),7,11(19),12,14,16-heptaen-9-one, aristololactam beta-D-glucoside, DTXSID301030980
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 138.0
Hydrogen Bond Donor Count 4.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1C2CC3CCCC3C3C4CCCCC4CC(C1C1CCCCC1)C23
Deep Smiles OC[C@H]O[C@@H][C@@H][C@H][C@@H]6O))O))O))NC=O)ccc5cccOC))cccc6c%10ccc%14)OCO5
Heavy Atom Count 33.0
Classyfire Class Aristolactams
Scaffold Graph Node Level OC1C2CC3OCOC3C3C4CCCCC4CC(C23)N1C1CCCCO1
Isotope Atom Count 0.0
Molecular Complexity 768.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 5.0
Iupac Name 14-methoxy-10-[(2S,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]-3,5-dioxa-10-azapentacyclo[9.7.1.02,6.08,19.013,18]nonadeca-1(18),2(6),7,11(19),12,14,16-heptaen-9-one
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 1.2
Gsk 4 400 Rule False
Molecular Formula C23H21NO9
Scaffold Graph Node Bond Level O=C1c2cc3c(c4c2c(cc2ccccc24)N1C1CCCCO1)OCO3
Inchi Key GIDCUQKCIZAUKW-AUJACXKFSA-N
Silicos It Class Soluble
Rotatable Bond Count 3.0
Synonyms aristolactum n-beta-glucoside
Esol Class Soluble
Functional Groups CO, c1cOCO1, cC(=O)N(c)[C@H](C)OC, cOC
Compound Name Aristololactam-glucoside
Exact Mass 455.122
Formal Charge 0.0
Monoisotopic Mass 455.122
Hydrogen Bond Acceptor Count 9.0
Molecular Weight 455.4
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C23H21NO9/c1-30-13-4-2-3-9-10(13)5-12-16-11(6-14-21(17(9)16)32-8-31-14)22(29)24(12)23-20(28)19(27)18(26)15(7-25)33-23/h2-6,15,18-20,23,25-28H,7-8H2,1H3/t15-,18-,19+,20-,23+/m1/s1
Smiles COC1=CC=CC2=C3C4=C(C=C21)N(C(=O)C4=CC5=C3OCO5)[C@@H]6[C@@H]([C@H]([C@@H]([C@H](O6)CO)O)O)O
Defined Bond Stereocenter Count 0.0
Egan Rule False

  • 1. Outgoing r'ship FOUND_IN to/from Aristolochia Indica (Plant) Rel Props:Reference:ISBN:9788171360536