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dimethyl (1S,10S,15R,17S,18S)-17-ethyl-7-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1,15-dicarboxylate

PubChem CID: 156021788

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Compound Synonyms CHEMBL4648800
Topological Polar Surface Area 163.0
Hydrogen Bond Donor Count 3.0
Heavy Atom Count 59.0
Isotope Atom Count 0.0
Molecular Complexity 1760.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name dimethyl (1S,10S,15R,17S,18S)-17-ethyl-7-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1,15-dicarboxylate
Prediction Hob 0.0
Xlogp 3.5
Molecular Formula C46H56N4O9
Prediction Swissadme 0.0
Inchi Key QSPNZYJNRJAQHY-QSYCZPBJSA-N
Fcsp3 0.5652173913043478
Logs -4.547
Rotatable Bond Count 10.0
Logd 3.346
Compound Name dimethyl (1S,10S,15R,17S,18S)-17-ethyl-7-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1,15-dicarboxylate
Prediction Hob Swissadme 0.0
Exact Mass 808.405
Formal Charge 0.0
Monoisotopic Mass 808.405
Hydrogen Bond Acceptor Count 12.0
Molecular Weight 809.0
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 1.0
Esol -6.582468193220339
Inchi InChI=1S/C46H56N4O9/c1-8-25-20-43(40(52)57-5)22-44(41(53)58-6)38(25)50(23-43)15-14-46(55)32-16-28(35(56-4)19-34(32)48-39(44)46)29-17-31-26(9-2)21-49(3)36(45(31,24-51)42(54)59-7)18-30-27-12-10-11-13-33(27)47-37(29)30/h9-13,16,19,25,29,31,36,38,47,51,55H,8,14-15,17-18,20-24H2,1-7H3/b26-9-/t25-,29-,31+,36-,38-,43+,44-,45-,46-/m0/s1
Smiles CC[C@H]1C[C@]2(C[C@@]3([C@H]1N(C2)CC[C@]4(C3=NC5=C4C=C(C(=C5)OC)[C@@H]6C[C@@H]7/C(=C\C)/CN([C@H]([C@@]7(CO)C(=O)OC)CC8=C6NC9=CC=CC=C89)C)O)C(=O)OC)C(=O)OC
Nring 10.0
Defined Bond Stereocenter Count 1.0