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methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate

PubChem CID: 156020220

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Compound Synonyms CHEMBL4648833
Topological Polar Surface Area 122.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 55.0
Isotope Atom Count 0.0
Molecular Complexity 1570.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob 0.0
Xlogp 5.3
Molecular Formula C44H52N4O7
Prediction Swissadme 0.0
Inchi Key OVJMPCBTOJTXQD-QKVMKJBNSA-N
Fcsp3 0.5909090909090909
Logs -4.155
Rotatable Bond Count 7.0
Logd 4.519
Compound Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 748.384
Formal Charge 0.0
Monoisotopic Mass 748.384
Hydrogen Bond Acceptor Count 9.0
Molecular Weight 748.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 11.0
Total Bond Stereocenter Count 0.0
Esol -7.621392018181818
Inchi InChI=1S/C44H52N4O7/c1-7-24-14-23-19-42(40(49)52-5)37-26(12-13-48(20-23)38(24)42)27-15-28(33(51-4)18-32(27)46-37)29-16-34-43(41(50)53-6)21-54-39(44(34)22(2)55-44)47(3)35(43)17-30-25-10-8-9-11-31(25)45-36(29)30/h8-11,15,18,22-24,29,34-35,38-39,45-46H,7,12-14,16-17,19-21H2,1-6H3/t22-,23+,24-,29-,34-,35-,38-,39-,42+,43-,44-/m0/s1
Smiles CC[C@H]1C[C@@H]2C[C@@]3([C@H]1N(C2)CCC4=C3NC5=CC(=C(C=C45)[C@@H]6C[C@H]7[C@]8(CO[C@@H]([C@]79[C@@H](O9)C)N([C@H]8CC1=C6NC2=CC=CC=C12)C)C(=O)OC)OC)C(=O)OC
Nring 13.0
Defined Bond Stereocenter Count 0.0