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methyl (1S,10R,15S,17S,18S)-17-ethyl-5-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1-carboxylate

PubChem CID: 156017391

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Compound Synonyms CHEMBL4642026
Topological Polar Surface Area 137.0
Hydrogen Bond Donor Count 3.0
Heavy Atom Count 55.0
Isotope Atom Count 0.0
Molecular Complexity 1590.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name methyl (1S,10R,15S,17S,18S)-17-ethyl-5-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1-carboxylate
Prediction Hob 0.0
Xlogp 4.1
Molecular Formula C44H54N4O7
Prediction Swissadme 0.0
Inchi Key OFCOWZWFNMOWNU-KPKAQVDPSA-N
Fcsp3 0.5681818181818182
Logs -5.064
Rotatable Bond Count 8.0
Logd 4.819
Compound Name methyl (1S,10R,15S,17S,18S)-17-ethyl-5-[(1S,12S,14R,15E,18S)-15-ethylidene-18-(hydroxymethyl)-18-methoxycarbonyl-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraen-12-yl]-10-hydroxy-6-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraene-1-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 750.399
Formal Charge 0.0
Monoisotopic Mass 750.399
Hydrogen Bond Acceptor Count 10.0
Molecular Weight 750.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 1.0
Esol -6.733727581818182
Inchi InChI=1S/C44H54N4O7/c1-7-25-17-24-20-42(40(50)54-5)38(25)48(21-24)16-15-44(52)30-13-14-33(53-4)35(37(30)46-39(42)44)29-18-31-26(8-2)22-47(3)34(43(31,23-49)41(51)55-6)19-28-27-11-9-10-12-32(27)45-36(28)29/h8-14,24-25,29,31,34,38,45,49,52H,7,15-23H2,1-6H3/b26-8-/t24-,25-,29-,31+,34-,38-,42-,43-,44+/m0/s1
Smiles CC[C@H]1C[C@H]2C[C@@]3([C@H]1N(C2)CC[C@@]4(C3=NC5=C4C=CC(=C5[C@@H]6C[C@@H]7/C(=C\C)/CN([C@H]([C@@]7(CO)C(=O)OC)CC8=C6NC9=CC=CC=C89)C)OC)O)C(=O)OC
Nring 0.0
Defined Bond Stereocenter Count 1.0