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methyl (3S,4S,10E,11R,13S)-10-ethylidene-13-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate

PubChem CID: 156011559

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Compound Synonyms CHEMBL4636746
Topological Polar Surface Area 126.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 55.0
Isotope Atom Count 0.0
Molecular Complexity 1590.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name methyl (3S,4S,10E,11R,13S)-10-ethylidene-13-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob 1.0
Xlogp 4.8
Molecular Formula C44H50N4O7
Prediction Swissadme 0.0
Inchi Key FGSMSNKIWGRJOM-PIHUVOOSSA-N
Fcsp3 0.5227272727272727
Logs -5.263
Rotatable Bond Count 7.0
Logd 4.977
Compound Name methyl (3S,4S,10E,11R,13S)-10-ethylidene-13-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 746.368
Formal Charge 0.0
Monoisotopic Mass 746.368
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 746.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 1.0
Esol -7.262392818181819
Inchi InChI=1S/C44H50N4O7/c1-6-23-16-25-19-43(41(50)53-4)38-28(14-15-48(39(23)43)40(25)49)27-12-13-33(52-3)35(37(27)46-38)30-17-31-24(7-2)20-47-22-55-21-44(31,42(51)54-5)34(47)18-29-26-10-8-9-11-32(26)45-36(29)30/h7-13,23,25,30-31,34,39,45-46H,6,14-22H2,1-5H3/b24-7-/t23-,25+,30-,31+,34-,39-,43+,44-/m0/s1
Smiles CC[C@H]1C[C@@H]2C[C@@]3([C@H]1N(C2=O)CCC4=C3NC5=C4C=CC(=C5[C@@H]6C[C@@H]7/C(=C\C)/CN8COC[C@]7([C@@H]8CC9=C6NC1=CC=CC=C91)C(=O)OC)OC)C(=O)OC
Nring 11.0
Defined Bond Stereocenter Count 1.0