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methyl (1S,16S,17S)-3-formyl-16-[(1S)-1-hydroxyethyl]-10,12-diazapentacyclo[12.3.1.02,10.04,9.012,17]octadeca-2,4,6,8-tetraene-1-carboxylate

PubChem CID: 156010110

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Compound Synonyms CHEMBL4634059
Topological Polar Surface Area 71.8
Hydrogen Bond Donor Count 1.0
Heavy Atom Count 27.0
Isotope Atom Count 0.0
Molecular Complexity 642.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 4.0
Iupac Name methyl (1S,16S,17S)-3-formyl-16-[(1S)-1-hydroxyethyl]-10,12-diazapentacyclo[12.3.1.02,10.04,9.012,17]octadeca-2,4,6,8-tetraene-1-carboxylate
Prediction Hob 1.0
Xlogp 1.6
Molecular Formula C21H24N2O4
Prediction Swissadme 1.0
Inchi Key QRRIMMYRGDDMOA-UUAKLTOTSA-N
Fcsp3 0.5238095238095238
Logs -1.903
Rotatable Bond Count 4.0
Logd 1.82
Compound Name methyl (1S,16S,17S)-3-formyl-16-[(1S)-1-hydroxyethyl]-10,12-diazapentacyclo[12.3.1.02,10.04,9.012,17]octadeca-2,4,6,8-tetraene-1-carboxylate
Prediction Hob Swissadme 1.0
Exact Mass 368.174
Formal Charge 0.0
Monoisotopic Mass 368.174
Hydrogen Bond Acceptor Count 5.0
Molecular Weight 368.4
Covalent Unit Count 1.0
Total Atom Stereocenter Count 5.0
Total Bond Stereocenter Count 0.0
Esol -3.1023512666666675
Inchi InChI=1S/C21H24N2O4/c1-12(25)15-7-13-8-21(20(26)27-2)18(15)22(9-13)11-23-17-6-4-3-5-14(17)16(10-24)19(21)23/h3-6,10,12-13,15,18,25H,7-9,11H2,1-2H3/t12-,13?,15+,18-,21-/m0/s1
Smiles C[C@@H]([C@H]1CC2C[C@@]3([C@H]1N(C2)CN4C3=C(C5=CC=CC=C54)C=O)C(=O)OC)O
Nring 1.0
Defined Bond Stereocenter Count 0.0