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(1R,2R,5S,10R,11R,14R,15S,18S,21R,22R,23S)-22-hydroxy-10-(hydroxymethyl)-2,14,15,21,22-pentamethyl-7-[(1S,18R,19S,20S)-18-methyl-14-oxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4,6,8,15-pentaen-19-yl]-6,8-dioxahexacyclo[12.12.0.02,11.05,10.015,24.018,23]hexacos-24-ene-18-carboxylic acid

PubChem CID: 155554987

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Compound Synonyms CHEMBL4551460
Topological Polar Surface Area 142.0
Hydrogen Bond Donor Count 4.0
Heavy Atom Count 60.0
Isotope Atom Count 0.0
Molecular Complexity 1870.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 15.0
Iupac Name (1R,2R,5S,10R,11R,14R,15S,18S,21R,22R,23S)-22-hydroxy-10-(hydroxymethyl)-2,14,15,21,22-pentamethyl-7-[(1S,18R,19S,20S)-18-methyl-14-oxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4,6,8,15-pentaen-19-yl]-6,8-dioxahexacyclo[12.12.0.02,11.05,10.015,24.018,23]hexacos-24-ene-18-carboxylic acid
Prediction Hob 0.0
Xlogp 6.6
Molecular Formula C50H66N2O8
Prediction Swissadme 0.0
Inchi Key LCZVPHZDOMBTOO-IFGBZRKBSA-N
Fcsp3 0.72
Logs -4.624
Rotatable Bond Count 3.0
Logd 4.756
Compound Name (1R,2R,5S,10R,11R,14R,15S,18S,21R,22R,23S)-22-hydroxy-10-(hydroxymethyl)-2,14,15,21,22-pentamethyl-7-[(1S,18R,19S,20S)-18-methyl-14-oxo-17-oxa-3,13-diazapentacyclo[11.8.0.02,10.04,9.015,20]henicosa-2(10),4,6,8,15-pentaen-19-yl]-6,8-dioxahexacyclo[12.12.0.02,11.05,10.015,24.018,23]hexacos-24-ene-18-carboxylic acid
Prediction Hob Swissadme 0.0
Exact Mass 822.482
Formal Charge 0.0
Monoisotopic Mass 822.482
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 823.1
Covalent Unit Count 1.0
Total Atom Stereocenter Count 16.0
Total Bond Stereocenter Count 0.0
Esol -9.007820800000001
Inchi InChI=1S/C50H66N2O8/c1-27-13-19-49(44(55)56)21-20-46(4)33(41(49)48(27,6)57)11-12-36-45(3)17-15-38-50(25-53,37(45)14-18-47(36,46)5)26-59-43(60-38)39-28(2)58-24-32-31(39)23-35-40-30(16-22-52(35)42(32)54)29-9-7-8-10-34(29)51-40/h7-11,24,27-28,31,35-39,41,43,51,53,57H,12-23,25-26H2,1-6H3,(H,55,56)/t27-,28-,31-,35+,36-,37-,38+,39-,41-,43?,45-,46-,47-,48-,49+,50-/m1/s1
Smiles C[C@@H]1CC[C@@]2(CC[C@@]3(C(=CC[C@H]4[C@]3(CC[C@@H]5[C@@]4(CC[C@H]6[C@@]5(COC(O6)[C@@H]7[C@H](OC=C8[C@H]7C[C@H]9C3=C(CCN9C8=O)C4=CC=CC=C4N3)C)CO)C)C)[C@@H]2[C@]1(C)O)C)C(=O)O
Nring 11.0
Defined Bond Stereocenter Count 0.0