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Silibinin B

PubChem CID: 1548994

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Compound Synonyms Silybin B, Silibinin B, 142797-34-0, SILYMARIN, SILYBIN (A and B)(P), 65666-07-1, UNII-853OHH1429, (2R,3R)-3,5,7-trihydroxy-2-[(2S,3S)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2,3-dihydro-1,4-benzodioxin-6-yl]-2,3-dihydrochromen-4-one, Legalon, DTXSID30858697, 853OHH1429, (2R,3R)-3,5,7-trihydroxy-2-((2S,3S)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2,3-dihydrobenzo[b][1,4]dioxin-6-yl)chroman-4-one, Flavobion, 308831-37-0, 4H-1-BENZOPYRAN-4-ONE, 2-((2S,3S)-2,3-DIHYDRO-3-(4-HYDROXY-3-METHOXYPHENYL)-2-(HYDROXYMETHYL)-1,4-BENZODIOXIN-6-YL)-2,3-DIHYDRO-3,5,7-TRIHYDROXY-, (2R,3R)-, rel-(2R,3R)-3,5,7-Trihydroxy-2-((2S,3S)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2,3-dihydrobenzo[b][1,4]dioxin-6-yl)chroman-4-one, Legalon 70, CCRIS 7096, PRX-321, Silybin A and B, 4H-1-Benzopyran-4-one, 2-[(2S,3S)-2,3-dihydro-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-1,4-benzodioxin-6-yl]-2,3-dihydro-3,5,7-trihydroxy-, (2R,3R)-, 4H-1-Benzopyran-4-one, 2-[(2S,3S)-2,3-dihydro-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-1,4-benzodioxin-6-yl]-2,3-dihydro-3,5,7-trihydroxy-, (2R,3R)-, 1,4-Benzodioxin, 4H-1-benzopyran-4-one deriv., (2R,3R)-2-[(2S,3S)-2,3-Dihydro-3-(4-hydroxy-3-metho, Milk thistle [NF], Silymarin + Melatonin, Silybin B (Standard), SILYBIN B [MI], UNII-U946SH95EE, SCHEMBL751461, Silybin B, analytical standard, CHEMBL592675, DTXCID703580, U946SH95EE, HY-N7046R, CHEBI:207762, HY-N7046, BDBM50088491, AKOS015912848, (2r,3r)-2-[(2s,3s)-2,3-dihydro-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-1,4-benzodioxin-6-yl]-2,3-dihydro-3,5,7-trihydroxy-4h-1-benzopyran-4-one, FS139048, FS180849, MS-28965, CS-0101839, SILYBIN B (CONSTITUENT OF MILK THISTLE), Q27269584, SILYBIN B (CONSTITUENT OF MILK THISTLE) [DSC], (2R,3R)-3,5,7-trihydroxy-2-[(2S,3S)-3-(4-hydroxy-3-methoxy-phenyl)-2-(hydroxymethyl)-2,3-dihydro-1,4-benzodioxin-6-yl]chroman-4-one, (2R,3R)-3,5,7-trihydroxy-2-[(2S,3S)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2,3-dihydro-1,4-benzodioxin-6-yl]-2,3-dihydro-4H-chromen-4-one
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 155.0
Hydrogen Bond Donor Count 5.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC1CC(C2CCC3CCC(C4CCCCC4)CC3C2)CC2CCCCC12
Np Classifier Class Dihydroflavonols, Flavonolignans
Deep Smiles OC[C@@H]Occcccc6O[C@H]%10cccccc6)OC)))O)))))))))[C@H]OcccO)ccc6C=O)[C@@H]%10O))))O
Heavy Atom Count 35.0
Classyfire Class Flavonolignans
Scaffold Graph Node Level OC1CC(C2CCC3OCC(C4CCCCC4)OC3C2)OC2CCCCC12
Isotope Atom Count 0.0
Molecular Complexity 750.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 4.0
Uniprot Id O42713, P11712, n.a., Q9Y6L6, Q9NPD5, O94956
Iupac Name (2R,3R)-3,5,7-trihydroxy-2-[(2S,3S)-3-(4-hydroxy-3-methoxyphenyl)-2-(hydroxymethyl)-2,3-dihydro-1,4-benzodioxin-6-yl]-2,3-dihydrochromen-4-one
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Lignans, neolignans and related compounds
Target Id NPT212, NPT73, NPT72, NPT622
Xlogp 2.4
Gsk 4 400 Rule False
Molecular Formula C25H22O10
Scaffold Graph Node Bond Level O=C1CC(c2ccc3c(c2)OC(c2ccccc2)CO3)Oc2ccccc21
Prediction Swissadme 0.0
Inchi Key SEBFKMXJBCUCAI-WAABAYLZSA-N
Silicos It Class Moderately soluble
Fcsp3 0.24
Logs -5.051
Rotatable Bond Count 4.0
Logd 2.44
Synonyms silybin b
Esol Class Moderately soluble
Functional Groups CO, cC(C)=O, cO, cOC
Compound Name Silibinin B
Prediction Hob Swissadme 0.0
Exact Mass 482.121
Formal Charge 0.0
Monoisotopic Mass 482.121
Hydrogen Bond Acceptor Count 10.0
Molecular Weight 482.4
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 4.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -4.14470562857143
Inchi InChI=1S/C25H22O10/c1-32-17-6-11(2-4-14(17)28)24-20(10-26)33-16-5-3-12(7-18(16)34-24)25-23(31)22(30)21-15(29)8-13(27)9-19(21)35-25/h2-9,20,23-29,31H,10H2,1H3/t20-,23-,24-,25+/m0/s1
Smiles COC1=C(C=CC(=C1)[C@H]2[C@@H](OC3=C(O2)C=C(C=C3)[C@@H]4[C@H](C(=O)C5=C(C=C(C=C5O4)O)O)O)CO)O
Nring 5.0
Np Classifier Biosynthetic Pathway Shikimates and Phenylpropanoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Lignans, Flavonoids

  • 1. Outgoing r'ship FOUND_IN to/from Anastatica Hierochuntica (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Silybum Marianum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all