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Solifenacin

PubChem CID: 154059

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Compound Synonyms Solifenacin, 242478-37-1, Soliten, (+)-Solifenacin, solifenacine, Solifenacina, UNII-A8910SQJ1U, Solifenacin (INN), A8910SQJ1U, YM-905, [(3R)-1-azabicyclo[2.2.2]octan-3-yl] (1S)-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylate, NSC-759144, DTXSID3048289, YM 905, NSC 759144, SOLIFENACIN [INN], (S)-(R)-Quinuclidin-3-yl 1-phenyl-3,4-dihydroisoquinoline-2(1H)-carboxylate, (3R)-1-azabicyclo[2.2.2]octan-3-yl (1S)-1-phenyl-1,2,3,4-tetrahydroisoquinoline-2-carboxylate, Solifenacin [INN:BAN], CHEMBL1200803, 2(1H)-Isoquinolinecarboxylic acid, 3,4-dihydro-1-phenyl-,1-azabicyclo(2.2.2)oct-3-yl ester, (R-(R*,S*))-, YM905 (free base), NCGC00168778-01, solifenacinum, solifenacin-succinate, MFCD18910847, Solifenacin (Standard), Solifenacin (YM905), SOLIFENACIN [MI], SOLIFENACIN [VANDF], CHEMBL1734, SOLIFENACIN [WHO-DD], SCHEMBL188493, GTPL7483, SCHEMBL9971260, DTXCID8028264, HY-A0034R, G04BD08, CHEBI:135530, FBOUYBDGKBSUES-VXKWHMMOSA-N, HMS3886O15, HY-A0034, BDBM50344284, BDBM50370682, s5238, AKOS015896445, CCG-268199, CS-8096, DB01591, NCGC00168778-06, DB-001095, NS00098872, D08522, D95831, AB01565949_02, EN300-20176688, EN300-20343692, BRD-K24723746-001-01-1, BRD-K24723746-036-02-5, ((8R)-1-azabicyclo(2.2.2)octan-8-yl)(1S)-1-phenyl-3,4-dihydro-1h-isoquinoline-2-carboxylate, (1S)-(3R)-1-azabicyclo[2.2.2]oct-3-yl-3,4-dihydro-1-phenyl-2(1H)-isoquinolinecarboxylate, [(3r)-1-azabicyclo[2.2.2]octan-3-yl](1s)-1-phenyl-3,4-dihydro-1hisoquinoline-2-carboxylate, [(8R)-1-azabicyclo[2.2.2]octan-8-yl] (1S)-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylate, 1172613-99-8
Topological Polar Surface Area 32.8
Hydrogen Bond Donor Count 0.0
Heavy Atom Count 27.0
Isotope Atom Count 0.0
Molecular Complexity 524.0
Database Name cmaup_ingredients;npass_chem_all;pubchem
Defined Atom Stereocenter Count 2.0
Uniprot Id P08482, P10980, P08483, n.a., P25094, Q12809, Q13936, Q14524, P15382, Q9UK17, O60840, P11229, P08172, P20309, P08173, P08912
Iupac Name [(3R)-1-azabicyclo[2.2.2]octan-3-yl] (1S)-1-phenyl-3,4-dihydro-1H-isoquinoline-2-carboxylate
Prediction Hob 1.0
Target Id NPT98, NPT2691, NPT2856, NPT5891, NPT262, NPT263, NPT264, NPT265, NPT266
Xlogp 4.0
Molecular Formula C23H26N2O2
Prediction Swissadme 1.0
Inchi Key FBOUYBDGKBSUES-VXKWHMMOSA-N
Fcsp3 0.4347826086956521
Logs -3.907
Rotatable Bond Count 3.0
Logd 3.777
Compound Name Solifenacin
Prediction Hob Swissadme 1.0
Exact Mass 362.199
Formal Charge 0.0
Monoisotopic Mass 362.199
Hydrogen Bond Acceptor Count 3.0
Molecular Weight 362.5
Covalent Unit Count 1.0
Total Atom Stereocenter Count 2.0
Total Bond Stereocenter Count 0.0
Esol -4.6533214888888885
Inchi InChI=1S/C23H26N2O2/c26-23(27-21-16-24-13-10-18(21)11-14-24)25-15-12-17-6-4-5-9-20(17)22(25)19-7-2-1-3-8-19/h1-9,18,21-22H,10-16H2/t21-,22-/m0/s1
Smiles C1CN2CCC1[C@H](C2)OC(=O)N3CCC4=CC=CC=C4[C@@H]3C5=CC=CC=C5
Nring 6.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Eucommia Ulmoides (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all
  • 2. Outgoing r'ship FOUND_IN to/from Jatropha Curcas (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all