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methyl (1R,12S,14R,15S,18R)-15-ethyl-12-[(1R,10S,15R,17S,18S)-17-ethyl-10-hydroxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-6-yl]-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate

PubChem CID: 145971027

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Compound Synonyms CHEMBL4218921
Topological Polar Surface Area 81.2
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 47.0
Isotope Atom Count 0.0
Molecular Complexity 1240.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 10.0
Iupac Name methyl (1R,12S,14R,15S,18R)-15-ethyl-12-[(1R,10S,15R,17S,18S)-17-ethyl-10-hydroxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-6-yl]-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate
Prediction Hob 0.0
Xlogp 5.9
Molecular Formula C40H50N4O3
Prediction Swissadme 0.0
Inchi Key TYIAIWRCGUDFJW-HLBWWQBFSA-N
Fcsp3 0.6
Logs -5.162
Rotatable Bond Count 5.0
Logd 5.282
Compound Name methyl (1R,12S,14R,15S,18R)-15-ethyl-12-[(1R,10S,15R,17S,18S)-17-ethyl-10-hydroxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-6-yl]-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 634.388
Formal Charge 0.0
Monoisotopic Mass 634.388
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 634.8
Covalent Unit Count 1.0
Total Atom Stereocenter Count 10.0
Total Bond Stereocenter Count 0.0
Esol -7.399333212765958
Inchi InChI=1S/C40H50N4O3/c1-5-23-15-22-16-30-37(23)44(20-22)14-13-40(46)31-12-11-25(17-33(31)42-38(30)40)28-18-27-24(6-2)21-43(3)34(35(27)39(45)47-4)19-29-26-9-7-8-10-32(26)41-36(28)29/h7-12,17,22-24,27-28,30,34-35,37,41,46H,5-6,13-16,18-21H2,1-4H3/t22-,23+,24-,27-,28+,30-,34-,35-,37+,40+/m1/s1
Smiles CC[C@H]1C[C@@H]2C[C@@H]3[C@H]1N(C2)CC[C@]4(C3=NC5=C4C=CC(=C5)[C@@H]6C[C@@H]7[C@@H](CN([C@@H]([C@@H]7C(=O)OC)CC8=C6NC9=CC=CC=C89)C)CC)O
Nring 10.0
Defined Bond Stereocenter Count 0.0