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methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate

PubChem CID: 145957978

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Compound Synonyms CHEMBL4162237
Topological Polar Surface Area 139.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 56.0
Isotope Atom Count 0.0
Molecular Complexity 1650.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob 0.0
Xlogp 4.5
Molecular Formula C44H50N4O8
Prediction Swissadme 0.0
Inchi Key YBDCTPKCACZFLY-GYVKKGGISA-N
Fcsp3 0.5681818181818182
Logs -4.627
Rotatable Bond Count 7.0
Logd 1.352
Compound Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,15R,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-14-oxo-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 762.363
Formal Charge 0.0
Monoisotopic Mass 762.363
Hydrogen Bond Acceptor Count 9.0
Molecular Weight 762.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 11.0
Total Bond Stereocenter Count 0.0
Esol -7.1808619428571445
Inchi InChI=1S/C44H50N4O8/c1-7-22-16-23-19-42(40(50)53-5)36-26(14-15-48(37(22)42)38(23)49)25-12-13-30(52-4)33(35(25)46-36)28-17-31-43(41(51)54-6)20-55-39(44(31)21(2)56-44)47(3)32(43)18-27-24-10-8-9-11-29(24)45-34(27)28/h8-13,21-23,28,31-32,37,39,45-46H,7,14-20H2,1-6H3/t21-,22-,23+,28-,31-,32-,37-,39-,42+,43-,44-/m0/s1
Smiles CC[C@H]1C[C@@H]2C[C@@]3([C@H]1N(C2=O)CCC4=C3NC5=C4C=CC(=C5[C@@H]6C[C@H]7[C@]8(CO[C@@H]([C@]79[C@@H](O9)C)N([C@H]8CC1=C6NC2=CC=CC=C12)C)C(=O)OC)OC)C(=O)OC
Nring 6.0
Defined Bond Stereocenter Count 0.0