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methyl (3S,4R,10E,11R,13S)-10-ethylidene-13-[(1S,15S,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate

PubChem CID: 145956640

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Compound Synonyms CHEMBL4159965
Topological Polar Surface Area 109.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 54.0
Isotope Atom Count 0.0
Molecular Complexity 1510.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name methyl (3S,4R,10E,11R,13S)-10-ethylidene-13-[(1S,15S,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob 0.0
Xlogp 5.6
Molecular Formula C44H52N4O6
Prediction Swissadme 0.0
Inchi Key SSPOBKKQGNARSJ-PIZRZXSPSA-N
Fcsp3 0.5454545454545454
Logs -5.434
Rotatable Bond Count 7.0
Logd 5.17
Compound Name methyl (3S,4R,10E,11R,13S)-10-ethylidene-13-[(1S,15S,17S,18S)-17-ethyl-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-7-yl]-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 732.389
Formal Charge 0.0
Monoisotopic Mass 732.389
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 732.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 1.0
Esol -7.703083066666669
Inchi InChI=1S/C44H52N4O6/c1-6-25-14-24-19-43(41(49)52-4)39-28(12-13-47(20-24)40(25)43)29-15-30(36(51-3)18-35(29)46-39)31-16-33-26(7-2)21-48-23-54-22-44(33,42(50)53-5)37(48)17-32-27-10-8-9-11-34(27)45-38(31)32/h7-11,15,18,24-25,31,33,37,40,45-46H,6,12-14,16-17,19-23H2,1-5H3/b26-7-/t24-,25-,31-,33+,37-,40-,43+,44+/m0/s1
Smiles CC[C@H]1C[C@H]2C[C@@]3([C@H]1N(C2)CCC4=C3NC5=CC(=C(C=C45)[C@@H]6C[C@@H]7/C(=C\C)/CN8COC[C@@]7([C@@H]8CC9=C6NC1=CC=CC=C91)C(=O)OC)OC)C(=O)OC
Nring 11.0
Defined Bond Stereocenter Count 1.0