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methyl (3S,4S,10E,11R,13S)-13-[(1S,14S,15R,17S,18S)-17-ethyl-14-(hydroxymethyl)-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-10-ethylidene-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate

PubChem CID: 145954403

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Compound Synonyms CHEMBL4169145
Topological Polar Surface Area 129.0
Hydrogen Bond Donor Count 3.0
Heavy Atom Count 56.0
Isotope Atom Count 0.0
Molecular Complexity 1560.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name methyl (3S,4S,10E,11R,13S)-13-[(1S,14S,15R,17S,18S)-17-ethyl-14-(hydroxymethyl)-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-10-ethylidene-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob 0.0
Xlogp 5.0
Molecular Formula C45H54N4O7
Prediction Swissadme 0.0
Inchi Key VYHSLRQXIWJYSY-QMPWSHTISA-N
Fcsp3 0.5555555555555556
Logs -4.871
Rotatable Bond Count 8.0
Logd 4.871
Compound Name methyl (3S,4S,10E,11R,13S)-13-[(1S,14S,15R,17S,18S)-17-ethyl-14-(hydroxymethyl)-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4(9),5,7-tetraen-5-yl]-10-ethylidene-6-oxa-8,15-diazapentacyclo[12.7.0.03,8.04,11.016,21]henicosa-1(14),16,18,20-tetraene-4-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 762.399
Formal Charge 0.0
Monoisotopic Mass 762.399
Hydrogen Bond Acceptor Count 9.0
Molecular Weight 762.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 1.0
Esol -7.423834742857144
Inchi InChI=1S/C45H54N4O7/c1-6-24-16-26-19-44(42(51)54-4)40-29(14-15-49(41(24)44)34(26)21-50)28-12-13-35(53-3)37(39(28)47-40)31-17-32-25(7-2)20-48-23-56-22-45(32,43(52)55-5)36(48)18-30-27-10-8-9-11-33(27)46-38(30)31/h7-13,24,26,31-32,34,36,41,46-47,50H,6,14-23H2,1-5H3/b25-7-/t24-,26+,31-,32+,34+,36-,41-,44+,45-/m0/s1
Smiles CC[C@H]1C[C@@H]2C[C@@]3([C@H]1N([C@@H]2CO)CCC4=C3NC5=C4C=CC(=C5[C@@H]6C[C@@H]7/C(=C\C)/CN8COC[C@]7([C@@H]8CC9=C6NC1=CC=CC=C91)C(=O)OC)OC)C(=O)OC
Nring 11.0
Defined Bond Stereocenter Count 1.0