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methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,10S,15R,17S,18S)-17-ethyl-10-hydroxy-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate

PubChem CID: 145951434

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Compound Synonyms CHEMBL4173635
Topological Polar Surface Area 138.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 56.0
Isotope Atom Count 0.0
Molecular Complexity 1680.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 12.0
Iupac Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,10S,15R,17S,18S)-17-ethyl-10-hydroxy-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob 0.0
Xlogp 4.2
Molecular Formula C44H52N4O8
Prediction Swissadme 0.0
Inchi Key RZPZCABJWQYDNJ-ZDPMTFHJSA-N
Fcsp3 0.6136363636363636
Logs -4.384
Rotatable Bond Count 7.0
Logd 3.626
Compound Name methyl (1S,3'S,12S,14S,15R,16S,19S)-12-[(1S,10S,15R,17S,18S)-17-ethyl-10-hydroxy-6-methoxy-1-methoxycarbonyl-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2,4(9),5,7-tetraen-7-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 764.379
Formal Charge 0.0
Monoisotopic Mass 764.379
Hydrogen Bond Acceptor Count 11.0
Molecular Weight 764.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 12.0
Total Bond Stereocenter Count 0.0
Esol -6.958418285714287
Inchi InChI=1S/C44H52N4O8/c1-7-24-14-23-19-41(39(49)53-5)36(24)48(20-23)13-12-43(51)29-15-26(32(52-4)18-31(29)46-37(41)43)27-16-33-42(40(50)54-6)21-55-38(44(33)22(2)56-44)47(3)34(42)17-28-25-10-8-9-11-30(25)45-35(27)28/h8-11,15,18,22-24,27,33-34,36,38,45,51H,7,12-14,16-17,19-21H2,1-6H3/t22-,23+,24-,27-,33-,34-,36-,38-,41-,42-,43-,44-/m0/s1
Smiles CC[C@H]1C[C@@H]2C[C@@]3([C@H]1N(C2)CC[C@]4(C3=NC5=C4C=C(C(=C5)OC)[C@@H]6C[C@H]7[C@]8(CO[C@@H]([C@]79[C@@H](O9)C)N([C@H]8CC1=C6NC2=CC=CC=C12)C)C(=O)OC)O)C(=O)OC
Nring 13.0
Defined Bond Stereocenter Count 0.0