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(S)-autumnaline

PubChem CID: 13878324

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Compound Synonyms (S)-autumnaline, 23068-65-7, (1S)-1-[2-(3-hydroxy-4,5-dimethoxyphenyl)ethyl]-6-methoxy-2-methyl-3,4-dihydro-1H-isoquinolin-7-ol, Autumnaline, CHEBI:80672, DTXSID50551719, Q27149714, (1S)-1-[2-(3-Hydroxy-4,5-dimethoxyphenyl)ethyl]-6-methoxy-2-methyl-1,2,3,4-tetrahydroisoquinolin-7-ol
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 71.4
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule False
Scaffold Graph Level C1CCC(CCC2CCCC3CCCCC32)CC1
Np Classifier Class Isoquinoline alkaloids, Phenethylisoquinoline alkaloids
Deep Smiles COcccCC[C@@H]NC)CCcc6ccO)cc6)OC)))))))))))))ccc6OC)))O
Heavy Atom Count 27.0
Classyfire Class Phenethylisoquinoline alkaloids
Scaffold Graph Node Level C1CCC(CCC2NCCC3CCCCC32)CC1
Isotope Atom Count 0.0
Molecular Complexity 464.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 1.0
Iupac Name (1S)-1-[2-(3-hydroxy-4,5-dimethoxyphenyl)ethyl]-6-methoxy-2-methyl-3,4-dihydro-1H-isoquinolin-7-ol
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 3.3
Gsk 4 400 Rule True
Molecular Formula C21H27NO5
Scaffold Graph Node Bond Level c1ccc(CCC2NCCc3ccccc32)cc1
Inchi Key GZUNPCNPOLOTLX-INIZCTEOSA-N
Silicos It Class Moderately soluble
Rotatable Bond Count 6.0
Synonyms autumnaline
Esol Class Moderately soluble
Functional Groups CN(C)C, cO, cOC
Compound Name (S)-autumnaline
Exact Mass 373.189
Formal Charge 0.0
Monoisotopic Mass 373.189
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 373.4
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 1.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C21H27NO5/c1-22-8-7-14-11-19(25-2)17(23)12-15(14)16(22)6-5-13-9-18(24)21(27-4)20(10-13)26-3/h9-12,16,23-24H,5-8H2,1-4H3/t16-/m0/s1
Smiles CN1CCC2=CC(=C(C=C2[C@@H]1CCC3=CC(=C(C(=C3)OC)OC)O)O)OC
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Tyrosine alkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Colchicum Autumnale (Plant) Rel Props:Reference:https://doi.org/10.15482/usda.adc/1239279