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methyl (1S,3'S,12R,14S,15R,16S,19S)-12-[(2R,3E,5R,12bS)-3-ethylidene-9-hydroxy-2-(2-hydroxyethyl)-5-methyl-2,4,6,7,12,12b-hexahydro-1H-indolo[2,3-a]quinolizin-5-ium-8-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate

PubChem CID: 137644588

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Compound Synonyms CHEMBL4087014
Topological Polar Surface Area 123.0
Hydrogen Bond Donor Count 4.0
Heavy Atom Count 52.0
Isotope Atom Count 0.0
Molecular Complexity 1460.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 10.0
Iupac Name methyl (1S,3'S,12R,14S,15R,16S,19S)-12-[(2R,3E,5R,12bS)-3-ethylidene-9-hydroxy-2-(2-hydroxyethyl)-5-methyl-2,4,6,7,12,12b-hexahydro-1H-indolo[2,3-a]quinolizin-5-ium-8-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob 0.0
Xlogp 3.8
Molecular Formula C42H51N4O6+
Prediction Swissadme 0.0
Inchi Key UIGSHRJIOMTGLF-CSJIKXFCSA-O
Fcsp3 0.5476190476190477
Logs -1.387
Rotatable Bond Count 5.0
Logd 2.75
Compound Name methyl (1S,3'S,12R,14S,15R,16S,19S)-12-[(2R,3E,5R,12bS)-3-ethylidene-9-hydroxy-2-(2-hydroxyethyl)-5-methyl-2,4,6,7,12,12b-hexahydro-1H-indolo[2,3-a]quinolizin-5-ium-8-yl]-3',20-dimethylspiro[17-oxa-10,20-diazapentacyclo[14.3.1.03,11.04,9.014,19]icosa-3(11),4,6,8-tetraene-15,2'-oxirane]-19-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 707.381
Formal Charge 1.0
Monoisotopic Mass 707.381
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 707.9
Covalent Unit Count 1.0
Total Atom Stereocenter Count 10.0
Total Bond Stereocenter Count 1.0
Esol -6.561684246153846
Inchi InChI=1S/C42H50N4O6/c1-6-23-20-46(4)15-13-26-35-30(44-38(26)31(46)17-24(23)14-16-47)11-12-32(48)36(35)28-18-33-41(40(49)50-5)21-51-39(42(33)22(2)52-42)45(3)34(41)19-27-25-9-7-8-10-29(25)43-37(27)28/h6-12,22,24,28,31,33-34,39,43-44,47H,13-21H2,1-5H3/p+1/b23-6-/t22-,24-,28+,31-,33-,34-,39-,41-,42-,46+/m0/s1
Smiles C/C=C\1/C[N@+]2(CCC3=C([C@@H]2C[C@@H]1CCO)NC4=C3C(=C(C=C4)O)[C@H]5C[C@H]6[C@]7(CO[C@@H]([C@]68[C@@H](O8)C)N([C@H]7CC9=C5NC1=CC=CC=C91)C)C(=O)OC)C
Nring 11.0
Defined Bond Stereocenter Count 1.0

  • 1. Outgoing r'ship FOUND_IN to/from Hunteria Zeylanica (Plant) Rel Props:Source_db:cmaup_ingredients