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Tamsulosin

PubChem CID: 129211

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Compound Synonyms TAMSULOSIN, 106133-20-4, (R)-5-(2-((2-(2-Ethoxyphenoxy)ethyl)amino)propyl)-2-methoxybenzenesulfonamide, Tamsulosine, Tamsulosina, Tamsulosinum, (-)-Tamsulosin, Tamsulon, Flowmax, Tamsulosine [INN-French], Tamsulosinum [INN-Latin], Tamsulosina [INN-Spanish], Contiflo OD, Amsulosin, (r)-(-)-tamsulosin, UNII-G3P28OML5I, G3P28OML5I, Tamsulosin (INN), CHEBI:9398, HSDB 7744, HIP1402, 5-[(2R)-2-[2-(2-ethoxyphenoxy)ethylamino]propyl]-2-methoxybenzenesulfonamide, HGP-0412, HIP-1402, Flomax (TN), CHEMBL836, DTXSID3023631, (R)-5-(2-((2-(2-Ethoxyphenoxy)ethyl)amino)-propyl)-2-methoxybenzenesulfonamide, 5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]-2-methoxybenzenesulfonamide, Benzenesulfonamide, 5-(2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-2-methoxy-, (R)-, (-)-YM617, TAMSULOSIN [INN], Tamsulosine (INN-French), Tamsulosinum (INN-Latin), Tamsulosin [INN:BAN], Tamsulosina (INN-Spanish), Harnal-D, 5-((2R)-2-(2-(2-ethoxyphenoxy)ethylamino)propyl)-2-methoxy-benzenesulfonamide, 5-[(2R)-2-[2-(2-ethoxyphenoxy)ethylamino]propyl]-2-methoxy-benzenesulfonamide, 5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]-2-methoxybenzene-1-sulfonamide, Tamsulon (TN), NCGC00167442-01, HSDB-7744, C20H28N2O5S, 5-((2R)-2-((2-(2-ethoxyphenoxy)ethyl)amino)propyl)-2-methoxybenzenesulfonamide, JGX, Tamsulosin (Standard), TAMSULOSIN [MI], TAMSULOSIN [HSDB], TAMSULOSIN [VANDF], 5-[2-[2-(2-ethoxyphenoxy)ethylamino]propyl]-2-methoxy-benzenesulfonamide, TAMSULOSIN [WHO-DD], SCHEMBL34378, GTPL488, MLS006011810, BIDD:GT0261, DTXCID803631, HY-B0661R, G04CA02, (r)-5-(2-(2-(2-ethoxyphenoxy)ethylamino)propyl)-2-methoxybenzenesulfonamide, HMS2090P15, HMS3884M15, HY-B0661, BDBM50060964, s1435, STK626950, AKOS005266643, CCG-268745, DB00706, 5-{(2R)-2-[(2-{[2-(ethyloxy)phenyl]oxy}ethyl)amino]propyl}-2-(methyloxy)benzenesulfonamide, NCGC00167442-02, NCGC00167442-08, AS-82157, SMR004703489, NS00001206, YM-12617-2, (R)-5-, C07124, D08560, F15143, SBI-0653937.0001, AB01275521-01, EN300-7417041, A835382, Q418480, SR-05000001519, SR-05000001519-1, BRD-K74339692-001-01-9, (-)-(R)-5-(2-((2-(O-ETHOXYPHENOXY)ETHYL)AMINO)PROPYL)-2-METHOXYBENZENESULFONAMIDE, (r)-5-[2-[[2-(2-ethoxyphenoxy)ethyl]amino]propyl]-2-methoxy-benzenesulfonamide, 5-[(2R)-2-[[2-(2-ethoxyphenoxy)ethyl]amino]propyl]-2-methoxybenzene-sulfonamide
Topological Polar Surface Area 108.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 28.0
Isotope Atom Count 0.0
Molecular Complexity 539.0
Database Name cmaup_ingredients;npass_chem_all;pubchem
Defined Atom Stereocenter Count 1.0
Uniprot Id P35348, P35368, P25100, P08913, P19328, P18825, P43140, P15823, P23944, P14416, P35462, P21917, P27732, P31389, P28565, P08908, P34969, P18089, P18841, P18130, O02824, n.a., P25094, P97718, P08684, P10635, P11712, P0DTD1
Iupac Name 5-[(2R)-2-[2-(2-ethoxyphenoxy)ethylamino]propyl]-2-methoxybenzenesulfonamide
Prediction Hob 1.0
Target Id NPT1788, NPT1789, NPT221, NPT222, NPT224, NPT243, NPT244, NPT92, NPT1785
Xlogp 2.7
Molecular Formula C20H28N2O5S
Prediction Swissadme 0.0
Inchi Key DRHKJLXJIQTDTD-OAHLLOKOSA-N
Fcsp3 0.4
Logs -3.226
Rotatable Bond Count 11.0
Logd 2.127
Compound Name Tamsulosin
Prediction Hob Swissadme 0.0
Exact Mass 408.172
Formal Charge 0.0
Monoisotopic Mass 408.172
Hydrogen Bond Acceptor Count 7.0
Molecular Weight 408.5
Covalent Unit Count 1.0
Total Atom Stereocenter Count 1.0
Total Bond Stereocenter Count 0.0
Esol -3.6838668571428577
Inchi InChI=1S/C20H28N2O5S/c1-4-26-17-7-5-6-8-18(17)27-12-11-22-15(2)13-16-9-10-19(25-3)20(14-16)28(21,23)24/h5-10,14-15,22H,4,11-13H2,1-3H3,(H2,21,23,24)/t15-/m1/s1
Smiles CCOC1=CC=CC=C1OCCN[C@H](C)CC2=CC(=C(C=C2)OC)S(=O)(=O)N
Nring 2.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Piper Nigrum (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all