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[(1S,2S,4S,5S,6R,10S)-5-hydroxy-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-3,9-dioxatricyclo[4.4.0.02,4]dec-7-en-2-yl]methyl 4-hydroxy-3-methoxybenzoate

PubChem CID: 129011779

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Compound Synonyms Kutkosid, beta-D-Glucopyranoside, (1aS,1bS,2S,5aR,6S)-1a,1b,2,5a,6,6a-hexahydro-6-hydroxy-1a-(((4-hydroxy-3-methoxybenzoyl)oxy)methyl)oxireno(4,5)cyclopenta(1,2-c)pyran-2-yl
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 197.0
Hydrogen Bond Donor Count 6.0
Pfizer 3 75 Rule True
Scaffold Graph Level CC(CCC12CC1CC1CCCC(CC3CCCCC3)C12)C1CCCCC1
Np Classifier Class Iridoids monoterpenoids
Deep Smiles OC[C@H]O[C@H]O[C@@H]OC=C[C@@H][C@H]6[C@@]COC=O)cccccc6)OC)))O))))))))O[C@H]3[C@H]6O))))))))))))[C@@H][C@H][C@@H]6O))O))O
Heavy Atom Count 36.0
Classyfire Class Tannins
Scaffold Graph Node Level OC(OCC12OC1CC1CCOC(OC3CCCCO3)C12)C1CCCCC1
Classyfire Subclass Hydrolyzable tannins
Isotope Atom Count 0.0
Molecular Complexity 839.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 11.0
Iupac Name [(1S,2S,4S,5S,6R,10S)-5-hydroxy-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-3,9-dioxatricyclo[4.4.0.02,4]dec-7-en-2-yl]methyl 4-hydroxy-3-methoxybenzoate
Veber Rule False
Classyfire Superclass Phenylpropanoids and polyketides
Xlogp -1.4
Gsk 4 400 Rule False
Molecular Formula C23H28O13
Scaffold Graph Node Bond Level O=C(OCC12OC1CC1C=COC(OC3CCCCO3)C12)c1ccccc1
Inchi Key JANLDILJJLTVDB-NGOGGKKYSA-N
Silicos It Class Soluble
Rotatable Bond Count 8.0
Synonyms 10-o-vaniloylcatalpol (kutkoside), kutkosid, kutkoside
Esol Class Very soluble
Functional Groups CO, CO[C@@H](C)O[C@H]1CCC=CO1, C[C@]1(C)O[C@H]1C, cC(=O)OC, cO, cOC
Compound Name [(1S,2S,4S,5S,6R,10S)-5-hydroxy-10-[(2R,3R,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-3,9-dioxatricyclo[4.4.0.02,4]dec-7-en-2-yl]methyl 4-hydroxy-3-methoxybenzoate
Exact Mass 512.153
Formal Charge 0.0
Monoisotopic Mass 512.153
Hydrogen Bond Acceptor Count 13.0
Molecular Weight 512.5
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 11.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Inchi InChI=1S/C23H28O13/c1-31-12-6-9(2-3-11(12)25)20(30)33-8-23-14-10(15(26)19(23)36-23)4-5-32-21(14)35-22-18(29)17(28)16(27)13(7-24)34-22/h2-6,10,13-19,21-22,24-29H,7-8H2,1H3/t10-,13-,14-,15+,16-,17+,18-,19+,21+,22-,23-/m1/s1
Smiles COC1=C(C=CC(=C1)C(=O)OC[C@@]23[C@@H]4[C@@H](C=CO[C@H]4O[C@@H]5[C@@H]([C@H]([C@@H]([C@H](O5)CO)O)O)O)[C@@H]([C@@H]2O3)O)O
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Monoterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Picrorhiza Kurroa (Plant) Rel Props:Reference:https://www.ncbi.nlm.nih.gov/pubmed/20821813
  • 2. Outgoing r'ship FOUND_IN to/from Picrorhiza Kurrooa (Plant) Rel Props:Reference:ISBN:9788185042084