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5,7,8,15-Tetrahydro-4-hydroxy-3-methoxy-6-methyl[1,3]benzodioxolo[5,6-e][2]benzazecin-14(6H)-one

PubChem CID: 1275589

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Compound Synonyms HUNNEMANINE, 490-52-8, 5,7,8,15-Tetrahydro-4-hydroxy-3-methoxy-6-methyl[1,3]benzodioxolo[5,6-e][2]benzazecin-14(6H)-one, EINECS 207-711-7, 5,7,8,15-Tetrahydro-4-hydroxy-3-methoxy-6-methyl(1,3)benzodioxolo(5,6-e)(2)benzazecin-14(6H)-one, 8-hydroxy-7-methoxy-11-methyl-17,19-dioxa-11-azatetracyclo[12.7.0.04,9.016,20]henicosa-1(21),4(9),5,7,14,16(20)-hexaen-2-one, Benzo(e)(1,3)dioxolo(4,5-k)(3)benzazecin-14(6H)-one, 5,7,8,15-tetrahydro-4-hydroxy-3-methoxy-6-methyl-, S9TC6BMK2V, Oprea1_819797, MEGxp0_001728, SCHEMBL3368057, ACon1_000791, DTXSID90197655, RSMSJQDBPYSXHH-UHFFFAOYSA-N, AKOS024281760, FH66061, NS00031848, BRD-K24867927-001-01-7, [1,3]Benzodioxolo[5,6-e][2]benzazecin-14(6H)-one, 5,7,8,15-tetrahydro-4-hydroxy-3-methoxy-6-methyl-, 30334-59-9, 5,7,8,15-Tetrahydro-4-hydroxy-3-methoxy-6-methylbenzo[c][1,3]benzodioxolo[5,6-g]azecin-14(6H)-one, Benzo[c][1,3]benzodioxolo[5,6-g]azecin-14(6H)-one, 5,7,8,15-tetrahydro-4-hydroxy-3-methoxy-6-methyl-
Ghose Rule True
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 68.2
Hydrogen Bond Donor Count 1.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC1CC2CCCCC2CCCCC2CC3CCCC3CC12
Np Classifier Class Protopine alkaloids
Deep Smiles COcccccc6O))CNC)CCccC=O)C%10))ccOCOc5c9
Heavy Atom Count 26.0
Classyfire Class Protopine alkaloids
Scaffold Graph Node Level OC1CC2CCCCC2CNCCC2CC3OCOC3CC12
Isotope Atom Count 0.0
Molecular Complexity 514.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 0.0
Iupac Name 8-hydroxy-7-methoxy-11-methyl-17,19-dioxa-11-azatetracyclo[12.7.0.04,9.016,20]henicosa-1(21),4(9),5,7,14,16(20)-hexaen-2-one
Veber Rule True
Classyfire Superclass Alkaloids and derivatives
Xlogp 2.6
Gsk 4 400 Rule True
Molecular Formula C20H21NO5
Scaffold Graph Node Bond Level O=C1Cc2ccccc2CNCCc2cc3c(cc21)OCO3
Inchi Key RSMSJQDBPYSXHH-UHFFFAOYSA-N
Silicos It Class Moderately soluble
Rotatable Bond Count 1.0
Synonyms hunnemanine
Esol Class Soluble
Functional Groups CN(C)C, c1cOCO1, cC(C)=O, cO, cOC
Compound Name 5,7,8,15-Tetrahydro-4-hydroxy-3-methoxy-6-methyl[1,3]benzodioxolo[5,6-e][2]benzazecin-14(6H)-one
Exact Mass 355.142
Formal Charge 0.0
Monoisotopic Mass 355.142
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 355.4
Gi Absorption True
Covalent Unit Count 1.0
Total Atom Stereocenter Count 0.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Inchi InChI=1S/C20H21NO5/c1-21-6-5-13-8-18-19(26-11-25-18)9-14(13)16(22)7-12-3-4-17(24-2)20(23)15(12)10-21/h3-4,8-9,23H,5-7,10-11H2,1-2H3
Smiles CN1CCC2=CC3=C(C=C2C(=O)CC4=C(C1)C(=C(C=C4)OC)O)OCO3
Np Classifier Biosynthetic Pathway Alkaloids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Tyrosine alkaloids