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methyl (1R,9R,16R,18R,21S)-5-[(15S,17S,19R)-15-[(1R)-1-hydroxyethyl]-1,11-diazapentacyclo[9.6.2.02,7.08,18.015,19]nonadeca-2,4,6,8(18)-tetraen-17-yl]-2,12-diazahexacyclo[14.2.2.19,12.01,9.03,8.016,21]henicosa-3(8),4,6-triene-18-carboxylate

PubChem CID: 127031361

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Compound Synonyms CHEMBL3780787
Topological Polar Surface Area 70.0
Hydrogen Bond Donor Count 2.0
Heavy Atom Count 47.0
Isotope Atom Count 0.0
Molecular Complexity 1330.0
Database Name cmaup_ingredients;pubchem
Defined Atom Stereocenter Count 9.0
Iupac Name methyl (1R,9R,16R,18R,21S)-5-[(15S,17S,19R)-15-[(1R)-1-hydroxyethyl]-1,11-diazapentacyclo[9.6.2.02,7.08,18.015,19]nonadeca-2,4,6,8(18)-tetraen-17-yl]-2,12-diazahexacyclo[14.2.2.19,12.01,9.03,8.016,21]henicosa-3(8),4,6-triene-18-carboxylate
Prediction Hob 0.0
Xlogp 5.1
Molecular Formula C40H48N4O3
Prediction Swissadme 0.0
Inchi Key NWRSTXLPBGHFPP-CKUBTQRQSA-N
Fcsp3 0.625
Logs -4.268
Rotatable Bond Count 4.0
Logd 3.669
Compound Name methyl (1R,9R,16R,18R,21S)-5-[(15S,17S,19R)-15-[(1R)-1-hydroxyethyl]-1,11-diazapentacyclo[9.6.2.02,7.08,18.015,19]nonadeca-2,4,6,8(18)-tetraen-17-yl]-2,12-diazahexacyclo[14.2.2.19,12.01,9.03,8.016,21]henicosa-3(8),4,6-triene-18-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 632.373
Formal Charge 0.0
Monoisotopic Mass 632.373
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 632.8
Covalent Unit Count 1.0
Total Atom Stereocenter Count 9.0
Total Bond Stereocenter Count 0.0
Esol -6.92993401276596
Inchi InChI=1S/C40H48N4O3/c1-24(45)38-13-6-17-42-19-11-27-26-7-3-4-8-31(26)44(33(27)34(38)42)32(23-38)25-9-10-28-30(21-25)41-40-15-14-37(22-29(40)35(46)47-2)12-5-18-43-20-16-39(28,40)36(37)43/h3-4,7-10,21,24,29,32,34,36,41,45H,5-6,11-20,22-23H2,1-2H3/t24-,29+,32+,34+,36+,37-,38-,39-,40-/m1/s1
Smiles C[C@H]([C@]12CCCN3[C@H]1C4=C(CC3)C5=CC=CC=C5N4[C@@H](C2)C6=CC7=C(C=C6)[C@]89CCN1[C@H]8[C@]2(CCC1)CC[C@@]9(N7)[C@@H](C2)C(=O)OC)O
Nring 12.0
Defined Bond Stereocenter Count 0.0

  • 1. Outgoing r'ship FOUND_IN to/from Kopsia Pauciflora (Plant) Rel Props:Source_db:cmaup_ingredients