This website is for informational and educational purposes only. Please do not self-medicate; contact a medical professional for advice before administration. This website is for informational and educational purposes only. Please do not self-medicate; contact a medical professional for advice before administration.

Ajacusine

PubChem CID: 124201531

Connections displayed (default: 10).
Loading graph...

Compound Synonyms Ajacusine, Aconitane-7,8,14-triol, 20-ethyl-1,6,16-trimethoxy-4-(((2-(3-methyl-2,5-dioxo-1-pyrrolidinyl)benzoyl)oxy)methyl)-, 14-benzoate, (1beta,14alpha,16beta)-, 66731-39-3
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 161.0
Hydrogen Bond Donor Count 2.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC(CC1C2CCC3C4CC5C6(CCC(C)C7CCCCC7C7C(C)CCC7C)CCCC5(C4CC6)C(C2)C13)C1CCCCC1
Np Classifier Class Terpenoid alkaloids
Deep Smiles CCNC[C@@]CC[C@H][C@]C8[C@]O)[C@H][C@H]95)OC)))[C@@][C@@H][C@H]6C[C@@H][C@@H]5OC=O)cccccc6)))))))))CC7)OC)))))))O)))))OC)))))COC=O)cccccc6NC=O)C[C@@H]C5=O))C
Heavy Atom Count 56.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC(OC1C2CCC3C4CC5C6(COC(O)C7CCCCC7N7C(O)CCC7O)CCCC5(C(C2)C31)C4NC6)C1CCCCC1
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1600.0
Database Name imppat_phytochem;pubchem
Defined Atom Stereocenter Count 12.0
Iupac Name [(1S,2R,3R,4S,5R,8R,9S,13S,16R,17R,18S)-4-benzoyloxy-11-ethyl-8,9-dihydroxy-6,16,18-trimethoxy-11-azahexacyclo[7.7.2.12,5.01,10.03,8.013,17]nonadecan-13-yl]methyl 2-[(3S)-3-methyl-2,5-dioxopyrrolidin-1-yl]benzoate
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 2.7
Gsk 4 400 Rule False
Molecular Formula C43H52N2O11
Scaffold Graph Node Bond Level O=C(OC1C2CCC3C4CC5C6(COC(=O)c7ccccc7N7C(=O)CCC7=O)CCCC5(C(C2)C31)C4NC6)c1ccccc1
Inchi Key UTXPEZCSRQUREP-USXLYEPZSA-N
Silicos It Class Poorly soluble
Rotatable Bond Count 12.0
Synonyms ajacusine
Esol Class Moderately soluble
Functional Groups CN(C)C, CO, COC, cC(=O)OC, cN1C(=O)CCC1=O
Compound Name Ajacusine
Exact Mass 772.357
Formal Charge 0.0
Monoisotopic Mass 772.357
Hydrogen Bond Acceptor Count 12.0
Molecular Weight 772.9
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 14.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 False
Inchi InChI=1S/C43H52N2O11/c1-6-44-21-40(22-55-38(49)25-14-10-11-15-28(25)45-31(46)18-23(2)36(45)47)17-16-30(53-4)42-27-19-26-29(52-3)20-41(50,43(51,39(42)44)35(54-5)34(40)42)32(27)33(26)56-37(48)24-12-8-7-9-13-24/h7-15,23,26-27,29-30,32-35,39,50-51H,6,16-22H2,1-5H3/t23-,26+,27+,29?,30+,32+,33-,34+,35-,39?,40-,41+,42-,43+/m0/s1
Smiles CCN1C[C@@]2(CC[C@H]([C@@]34[C@@H]2[C@@H]([C@@](C31)([C@]5(CC([C@H]6C[C@@H]4[C@@H]5[C@H]6OC(=O)C7=CC=CC=C7)OC)O)O)OC)OC)COC(=O)C8=CC=CC=C8N9C(=O)C[C@@H](C9=O)C
Np Classifier Biosynthetic Pathway Alkaloids, Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule False
Np Classifier Superclass Pseudoalkaloids

  • 1. Outgoing r'ship FOUND_IN to/from Consolida Ajacis (Plant) Rel Props:Reference:https://doi.org/10.15482/usda.adc/1239279