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Phorbol acetate, caprate

PubChem CID: 124027

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Compound Synonyms Phorbol acetate, caprate, 20839-15-0, 12-o-acetylphorbol-13-decanoate, 16561-28-7, [(1S,2S,6R,10S,11R,13S,14R,15R)-14-acetyloxy-1,6-dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] decanoate, 12-O-Acetyl-phorbol-13-decanoate, BRN 2610782, CHEMBL2375785, Phorbol monoacetate monodecanoate, DTXSID40937109, 12-O-Acetylphorbol 13-decanoate, Phorbol 12-acetate 13-decanoate, Decanoic acid, 9a-ester with 1,1a-alpha,1b-beta,4,4a,7a-alpha,7b,8,9,9a-decahydro-3-(hydroxymethyl)-4a-beta,7b-alpha,9-beta,9a-alpha-tetrahydroxy-1,1,6,8-alpha-tetramethyl-5H-cyclopropa(3,4)benz(1,2-e)azulen-5-one 9-acetate, Decanoic acid, ester with phorbol acetate, [acetoxy-dihydroxy-(hydroxymethyl)-tetramethyl-oxo-[?]yl] decanoate, (1aR)-1,1,6,8alpha-Tetramethyl-3-(hydroxymethyl)-5-oxo-1,1aalpha,1bbeta,4,4a,7aalpha,7b,8,9,9a-decahydro-5H-cyclopr, 28878-88-8, 5H-Cyclopropa(3,4)benz(1,2-e)azulen-5-one, 1,1a,1b,4,4a,7a,7b,8,9,9a-decahydro-4a,7b,9,9a-tetrahydroxy-3-(hydroxymethyl)-1,1,6,8-tetramethyl-, monoacetate monodecanoate, 9-(Acetyloxy)-4a,7b-dihydroxy-3-(hydroxymethyl)-1,1,6,8-tetramethyl-5-oxo-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-9aH-cyclopropa[3,4]benzo[1,2-e]azulen-9a-yl decanoate, Decanoic acid, (1aR,1bS,4aR,7aS,7bS,8R,9R,9aS)-9-(acetyloxy)-1,1a,1b,4,4a,5,7a,7b,8,9-decahydro-4a,7b-dihydroxy-3-(hydroxymethyl)-1,1,6,8-tetramethyl-5-oxo-9aH-cyclopropa[3,4]benz[1,2-e]azulen-9a-yl ester
Ghose Rule False
Classyfire Kingdom Organic compounds
Topological Polar Surface Area 130.0
Hydrogen Bond Donor Count 3.0
Pfizer 3 75 Rule False
Scaffold Graph Level CC1CCC2C1CCCC1C3CC3CCC21
Np Classifier Class Tetracyclic diterpenoids, Tigliane diterpenoids
Deep Smiles CCCCCCCCCC=O)O[C@@][C@H]OC=O)C)))[C@@H]C)[C@][C@H][C@@H]6C7C)C)))C=CCO))C[C@][C@H]7C=CC5=O))C))))O))))))O
Heavy Atom Count 40.0
Classyfire Class Prenol lipids
Scaffold Graph Node Level OC1CCC2C1CCCC1C3CC3CCC21
Classyfire Subclass Diterpenoids
Isotope Atom Count 0.0
Molecular Complexity 1090.0
Database Name cmaup_ingredients;imppat_phytochem;npass_chem_all;pubchem
Defined Atom Stereocenter Count 8.0
Iupac Name [(1S,2S,6R,10S,11R,13S,14R,15R)-14-acetyloxy-1,6-dihydroxy-8-(hydroxymethyl)-4,12,12,15-tetramethyl-5-oxo-13-tetracyclo[8.5.0.02,6.011,13]pentadeca-3,8-dienyl] decanoate
Prediction Hob 0.0
Veber Rule False
Classyfire Superclass Lipids and lipid-like molecules
Xlogp 4.4
Gsk 4 400 Rule False
Molecular Formula C32H48O8
Scaffold Graph Node Bond Level O=C1C=CC2C1CC=CC1C3CC3CCC21
Prediction Swissadme 0.0
Inchi Key CSJWNHJJHIAAIG-SVOQZPEWSA-N
Silicos It Class Moderately soluble
Fcsp3 0.78125
Logs -4.624
Rotatable Bond Count 13.0
Logd 3.687
Synonyms 12-o-acetylphorbol-13-decanoate
Esol Class Moderately soluble
Functional Groups CC(=O)OC, CC(C)=CC, CC1=CCCC1=O, CO
Compound Name Phorbol acetate, caprate
Prediction Hob Swissadme 0.0
Exact Mass 560.335
Formal Charge 0.0
Monoisotopic Mass 560.335
Hydrogen Bond Acceptor Count 8.0
Molecular Weight 560.7
Gi Absorption False
Covalent Unit Count 1.0
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 0.0
Lipinski Rule Of 5 True
Esol -5.217913600000001
Inchi InChI=1S/C32H48O8/c1-7-8-9-10-11-12-13-14-25(35)40-32-26(29(32,5)6)23-16-22(18-33)17-30(37)24(15-19(2)27(30)36)31(23,38)20(3)28(32)39-21(4)34/h15-16,20,23-24,26,28,33,37-38H,7-14,17-18H2,1-6H3/t20-,23+,24-,26-,28-,30-,31-,32-/m1/s1
Smiles CCCCCCCCCC(=O)O[C@@]12[C@@H](C1(C)C)[C@@H]3C=C(C[C@]4([C@H]([C@]3([C@@H]([C@H]2OC(=O)C)C)O)C=C(C4=O)C)O)CO
Nring 4.0
Np Classifier Biosynthetic Pathway Terpenoids
Defined Bond Stereocenter Count 0.0
Egan Rule True
Np Classifier Superclass Diterpenoids

  • 1. Outgoing r'ship FOUND_IN to/from Croton Tiglium (Plant) Rel Props:Source_db:cmaup_ingredients;npass_chem_all