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methyl (1S,12R,14R,15E,18S)-15-ethylidene-12-[(1R,15S,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-6-yl]-18-(hydroxymethyl)-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate

PubChem CID: 122179185

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Compound Synonyms CHEMBL3581903
Prediction Swissadme 0.0
Topological Polar Surface Area 93.8
Hydrogen Bond Donor Count 3.0
Inchi Key FEQZUIYQDAAUOE-UMXRBDIUSA-N
Fcsp3 0.5476190476190477
Rotatable Bond Count 6.0
Heavy Atom Count 50.0
Compound Name methyl (1S,12R,14R,15E,18S)-15-ethylidene-12-[(1R,15S,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-6-yl]-18-(hydroxymethyl)-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate
Prediction Hob Swissadme 0.0
Exact Mass 676.399
Formal Charge 0.0
Monoisotopic Mass 676.399
Isotope Atom Count 0.0
Molecular Complexity 1310.0
Hydrogen Bond Acceptor Count 6.0
Molecular Weight 676.9
Database Name cmaup_ingredients;pubchem
Covalent Unit Count 1.0
Defined Atom Stereocenter Count 8.0
Iupac Name methyl (1S,12R,14R,15E,18S)-15-ethylidene-12-[(1R,15S,17S,18S)-17-ethyl-7-methoxy-3,13-diazapentacyclo[13.3.1.02,10.04,9.013,18]nonadeca-2(10),4,6,8-tetraen-6-yl]-18-(hydroxymethyl)-17-methyl-10,17-diazatetracyclo[12.3.1.03,11.04,9]octadeca-3(11),4,6,8-tetraene-18-carboxylate
Total Atom Stereocenter Count 8.0
Total Bond Stereocenter Count 1.0
Prediction Hob 0.0
Esol -7.441492400000001
Inchi InChI=1S/C42H52N4O4/c1-6-24-14-23-15-32-38-27(12-13-46(20-23)40(24)32)28-18-36(49-4)29(17-35(28)44-38)30-16-33-25(7-2)21-45(3)37(42(33,22-47)41(48)50-5)19-31-26-10-8-9-11-34(26)43-39(30)31/h7-11,17-18,23-24,30,32-33,37,40,43-44,47H,6,12-16,19-22H2,1-5H3/b25-7-/t23-,24-,30+,32-,33+,37-,40-,42-/m0/s1
Smiles CC[C@H]1C[C@H]2C[C@@H]3[C@H]1N(C2)CCC4=C3NC5=CC(=C(C=C45)OC)[C@H]6C[C@@H]7/C(=C\C)/CN([C@H]([C@@]7(CO)C(=O)OC)CC8=C6NC9=CC=CC=C89)C
Xlogp 5.6
Defined Bond Stereocenter Count 1.0
Molecular Formula C42H52N4O4